CN102471290B - 手性3-三唑基亚砜衍生物的制备方法 - Google Patents

手性3-三唑基亚砜衍生物的制备方法 Download PDF

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Publication number
CN102471290B
CN102471290B CN201080031476.1A CN201080031476A CN102471290B CN 102471290 B CN102471290 B CN 102471290B CN 201080031476 A CN201080031476 A CN 201080031476A CN 102471290 B CN102471290 B CN 102471290B
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alkyl
chiral
independently
hydrogen
fluorine
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Chinese (zh)
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CN102471290A (zh
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S·安托斯
N·吕
W·A·莫拉迪
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Bayer Pharma AG
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Bayer Pharma AG
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J31/00—Catalysts comprising hydrides, coordination complexes or organic compounds
    • B01J31/02—Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides
    • B01J31/12—Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides containing organo-metallic compounds or metal hydrides

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
CN201080031476.1A 2009-07-16 2010-07-14 手性3-三唑基亚砜衍生物的制备方法 Expired - Fee Related CN102471290B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE102009027771.4 2009-07-16
DE102009027771 2009-07-16
PCT/EP2010/004288 WO2011006646A1 (de) 2009-07-16 2010-07-14 Verfahren zur herstellung von chiralen 3-triazolyl-sulfoxid-derivaten

Publications (2)

Publication Number Publication Date
CN102471290A CN102471290A (zh) 2012-05-23
CN102471290B true CN102471290B (zh) 2016-02-03

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CN201080031476.1A Expired - Fee Related CN102471290B (zh) 2009-07-16 2010-07-14 手性3-三唑基亚砜衍生物的制备方法

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Country Link
US (3) US8314133B2 (enExample)
EP (1) EP2454242B1 (enExample)
JP (1) JP5676602B2 (enExample)
KR (1) KR20120037993A (enExample)
CN (1) CN102471290B (enExample)
BR (1) BR112012001078A8 (enExample)
DK (1) DK2454242T3 (enExample)
ES (1) ES2525535T3 (enExample)
IL (1) IL217136A0 (enExample)
IN (1) IN2012DN00422A (enExample)
MX (1) MX2012000583A (enExample)
RU (1) RU2012105122A (enExample)
TW (1) TWI471314B (enExample)
WO (1) WO2011006646A1 (enExample)

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EP2274982A1 (de) * 2009-07-16 2011-01-19 Bayer CropScience AG Verwendung von Phenyltriazolen zur Bekämpfung von Insekten und Spinnmilben durch Angiessen, Tröpfchen- oder Tauchapplikation oder durch Behandlung von Saatgut
RU2012105122A (ru) 2009-07-16 2013-08-27 Байер Кропсайенс Аг Способ получения хиральных производных 3-триазолилсульфоксида
WO2011009552A1 (de) * 2009-07-23 2011-01-27 Bayer Cropscience Ag Neue alkoxyenone und enaminoketone und ein verfahren zu deren herstellung
US8242313B2 (en) 2009-07-23 2012-08-14 Bayer Cropscience Ag Alkoxy enones and enamino ketones and a process for preparation thereof
BR112012003870B1 (pt) * 2009-08-20 2018-11-21 Bayer Intellectual Property Gmbh derivados de sulfeto substituídos com 3-triazolilfenila, seu uso, seu processo de preparação e seus intermediários, composições agroquímicas, seu processo de preparação, e processo para combate de parasitas animais
WO2011029506A1 (de) * 2009-08-20 2011-03-17 Bayer Cropscience Ag 3-[1-(3-haloalkyl)-triazolyl]-phenyl-sulfid-derivate als akarizide und insektizide
EP2578575B1 (en) * 2010-06-01 2016-05-04 Kumiai Chemical Industry CO., LTD. Triazole compound having pest-controlling activity
EP2606726A1 (de) 2011-12-21 2013-06-26 Bayer CropScience AG N-Arylamidine-substituierte trifluoroethylsulfid-Derivate als Akarizide und Insektizide
CN104619683B (zh) 2012-09-27 2017-05-10 拜耳农作物科学股份公司 用于制备任选地取代的苯基和吡啶基吡咯烷类的方法
WO2014090765A1 (en) 2012-12-12 2014-06-19 Bayer Cropscience Ag Use of 1-[2-fluoro-4-methyl-5-(2,2,2-trifluoroethylsulfinyl)phenyl]-5-amino-3-trifluoromethyl)-1 h-1,2,4 tfia zole for controlling nematodes in nematode-resistant crops
WO2015036380A1 (de) 2013-09-13 2015-03-19 Bayer Cropscience Ag Verfahren zur reduktion von arylsulfoxiden zu arylthioethern
WO2015135984A1 (de) 2014-03-13 2015-09-17 Bayer Cropscience Ag Verfahren zur herstellung von chiralen 3-(5-aminotriazolyl)-sulfoxid-derivaten
JP7260532B2 (ja) * 2017-10-18 2023-04-18 バイエル・アクチエンゲゼルシヤフト 殺虫／殺ダニ特性を有する活性化合物の組合せ
WO2021084074A1 (en) 2019-10-30 2021-05-06 Solvay Sa Compositions and films comprising a polymer and tis2 particles, and their preparation and uses
JP7657783B2 (ja) 2020-04-30 2025-04-07 クミアイ化学工業株式会社 モノスルホキシド誘導体の製造方法
CN116981659A (zh) 2021-03-26 2023-10-31 拜耳公司 制备对映体富集的(2z)-2-(苯基亚氨基)-1,3-噻唑烷-4-酮亚砜衍生物的方法

Citations (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1076053A1 (en) * 1998-04-27 2001-02-14 Kumiai Chemical Industry Co., Ltd. 3-arylphenyl sulfide derivatives and insecticides and miticides
WO2006040635A1 (en) * 2004-10-11 2006-04-20 Ranbaxy Laboratories Limited Processes for the preparation of substituted sulfoxides
CN1823065A (zh) * 2003-03-28 2006-08-23 希德姆医药公司 用于对映选择性制备亚砜衍生物的方法
CN1867544A (zh) * 2003-09-19 2006-11-22 塞弗伦法国公司 通过不对称氧化而对映选择性合成莫达非尼的单一对映异构体的方法
CN101012141A (zh) * 2007-02-02 2007-08-08 沈阳药科大学 手性亚砜类化合物的制备方法
CN101035787A (zh) * 2004-10-05 2007-09-12 希德姆医药股份公司 亚砜衍生物的对映选择性制备方法
CN101039922A (zh) * 2004-10-20 2007-09-19 组合化学工业株式会社 3－三唑基苯基硫醚衍生物及含其作为有效成分的杀虫·杀螨·杀线虫剂
CN101429192A (zh) * 2008-08-22 2009-05-13 扬子江药业集团有限公司 生产手性亚砜衍生物的新方法
WO2009069312A1 (ja) * 2007-11-30 2009-06-04 Ihara Chemical Industry Co., Ltd. （１ｈ－１，２，４－トリアゾール－１－イル）アリール化合物及びその製造方法

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2863611B1 (fr) * 2003-12-15 2006-03-24 Sidem Pharma Sa Procede de preparation enantioselective de derives de sulfoxydes
EP1608649A2 (fr) * 2003-03-28 2005-12-28 Sidem Pharma SA Procede de preparation enantioselective de derives de sulfoxydes.
CN101323582A (zh) * 2008-07-30 2008-12-17 大连理工大学 一类手性西佛碱配体及其在硫醚不对称氧化反应中的应用
EP2274982A1 (de) 2009-07-16 2011-01-19 Bayer CropScience AG Verwendung von Phenyltriazolen zur Bekämpfung von Insekten und Spinnmilben durch Angiessen, Tröpfchen- oder Tauchapplikation oder durch Behandlung von Saatgut
RU2012105122A (ru) 2009-07-16 2013-08-27 Байер Кропсайенс Аг Способ получения хиральных производных 3-триазолилсульфоксида
WO2011029506A1 (de) * 2009-08-20 2011-03-17 Bayer Cropscience Ag 3-[1-(3-haloalkyl)-triazolyl]-phenyl-sulfid-derivate als akarizide und insektizide
BR112012003870B1 (pt) * 2009-08-20 2018-11-21 Bayer Intellectual Property Gmbh derivados de sulfeto substituídos com 3-triazolilfenila, seu uso, seu processo de preparação e seus intermediários, composições agroquímicas, seu processo de preparação, e processo para combate de parasitas animais

Patent Citations (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1076053A1 (en) * 1998-04-27 2001-02-14 Kumiai Chemical Industry Co., Ltd. 3-arylphenyl sulfide derivatives and insecticides and miticides
CN1823065A (zh) * 2003-03-28 2006-08-23 希德姆医药公司 用于对映选择性制备亚砜衍生物的方法
CN1867544A (zh) * 2003-09-19 2006-11-22 塞弗伦法国公司 通过不对称氧化而对映选择性合成莫达非尼的单一对映异构体的方法
CN101035787A (zh) * 2004-10-05 2007-09-12 希德姆医药股份公司 亚砜衍生物的对映选择性制备方法
WO2006040635A1 (en) * 2004-10-11 2006-04-20 Ranbaxy Laboratories Limited Processes for the preparation of substituted sulfoxides
CN101039922A (zh) * 2004-10-20 2007-09-19 组合化学工业株式会社 3－三唑基苯基硫醚衍生物及含其作为有效成分的杀虫·杀螨·杀线虫剂
CN101012141A (zh) * 2007-02-02 2007-08-08 沈阳药科大学 手性亚砜类化合物的制备方法
WO2009069312A1 (ja) * 2007-11-30 2009-06-04 Ihara Chemical Industry Co., Ltd. （１ｈ－１，２，４－トリアゾール－１－イル）アリール化合物及びその製造方法
CN101429192A (zh) * 2008-08-22 2009-05-13 扬子江药业集团有限公司 生产手性亚砜衍生物的新方法

Also Published As

Publication number Publication date
EP2454242A1 (de) 2012-05-23
IL217136A0 (en) 2012-02-29
KR20120037993A (ko) 2012-04-20
JP5676602B2 (ja) 2015-02-25
TWI471314B (zh) 2015-02-01
DK2454242T3 (en) 2015-02-02
MX2012000583A (es) 2012-02-13
WO2011006646A1 (de) 2011-01-20
CN102471290A (zh) 2012-05-23
RU2012105122A (ru) 2013-08-27
US20140256953A1 (en) 2014-09-11
IN2012DN00422A (enExample) 2015-05-15
US20130172573A1 (en) 2013-07-04
BR112012001078A2 (pt) 2015-09-01
TW201116517A (en) 2011-05-16
EP2454242B1 (de) 2014-10-15
US8765970B2 (en) 2014-07-01
US8314133B2 (en) 2012-11-20
ES2525535T3 (es) 2014-12-26
BR112012001078A8 (pt) 2016-05-03
JP2012532906A (ja) 2012-12-20
US20110015405A1 (en) 2011-01-20

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