CN102083806A - 用于治疗急性和慢性炎性疾病的5-(4-甲基磺酰基-苯基)-噻唑衍生物 - Google Patents

用于治疗急性和慢性炎性疾病的5-(4-甲基磺酰基-苯基)-噻唑衍生物 Download PDF

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Publication number
CN102083806A
CN102083806A CN2009801226820A CN200980122682A CN102083806A CN 102083806 A CN102083806 A CN 102083806A CN 2009801226820 A CN2009801226820 A CN 2009801226820A CN 200980122682 A CN200980122682 A CN 200980122682A CN 102083806 A CN102083806 A CN 102083806A
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compound
disease
cell
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tnf
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Chinese (zh)
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维克特·鲁华欧罗佑
安东尼奥·迪拉西拉马门尼兹
梅尔秋·奥瓦兹迪默索托
安娜·慕诺兹慕诺兹
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Faes Farma SA
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Faes Farma SA
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Priority claimed from US12/139,661 external-priority patent/US7781594B2/en
Priority claimed from EP08380177A external-priority patent/EP2135864A1/en
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Publication of CN102083806A publication Critical patent/CN102083806A/zh
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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CN2009801226820A 2008-06-16 2009-06-15 用于治疗急性和慢性炎性疾病的5-(4-甲基磺酰基-苯基)-噻唑衍生物 Pending CN102083806A (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US12/139,661 US7781594B2 (en) 2008-06-16 2008-06-16 5-(4-methanesulfonyl-phenyl)-thiazole derivatives for the treatment of acute and chronic inflammatory diseases
US12/139,661 2008-06-16
EP08380177.9 2008-06-16
EP08380177A EP2135864A1 (en) 2008-06-16 2008-06-16 5-(4-methanesulfonyl-phenyl)-thiazole derivatives for the treatment of acute and chronic inflammatory diseases
PCT/EP2009/057324 WO2009153226A1 (en) 2008-06-16 2009-06-15 5-(4-methanesulfonyl-phenyl)-thiazole derivatives for the treatment of acute and chronic inflammatory diseases

Publications (1)

Publication Number Publication Date
CN102083806A true CN102083806A (zh) 2011-06-01

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CN2009801226820A Pending CN102083806A (zh) 2008-06-16 2009-06-15 用于治疗急性和慢性炎性疾病的5-(4-甲基磺酰基-苯基)-噻唑衍生物

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EP (1) EP2313382A1 (enExample)
JP (1) JP2011524352A (enExample)
KR (1) KR20110022679A (enExample)
CN (1) CN102083806A (enExample)
AR (1) AR072113A1 (enExample)
AU (1) AU2009259451B2 (enExample)
BR (1) BRPI0915325A2 (enExample)
CA (1) CA2728139A1 (enExample)
CO (1) CO6331429A2 (enExample)
IL (1) IL209801A0 (enExample)
MA (1) MA32473B1 (enExample)
MX (1) MX2010013978A (enExample)
NZ (1) NZ589894A (enExample)
RU (1) RU2495031C2 (enExample)
SA (1) SA109300384B1 (enExample)
TW (1) TWI403506B (enExample)
UY (1) UY31896A (enExample)
WO (1) WO2009153226A1 (enExample)
ZA (1) ZA201008877B (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111343975A (zh) * 2017-11-23 2020-06-26 埃慕尼克股份公司 用于预防或治疗慢性炎性疾病和/或自身免疫疾病的维多地莫的剂量方案
CN115484959A (zh) * 2020-04-16 2022-12-16 米内尔瓦有限公司 用于治疗炎症的3-氮杂-双环[3.2.1]辛烷羧酸及其衍生物

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2961695B1 (fr) * 2010-06-29 2012-07-06 Galderma Res & Dev Utilisation de composes dans le traitement ou la prevention de troubles cutanes
RU2502513C2 (ru) * 2012-01-11 2013-12-27 Государственное бюджетное учреждение здравоохранения Свердловской области "Свердловский областной клинический психоневрологический госпиталь для ветеранов войн" (ГБУЗ СО "СОКП Госпиталь для ветеранов войн") Способ лечения больных с полиорганной патологией озонотерапией
KR102076936B1 (ko) * 2019-08-12 2020-02-13 연세대학교 산학협력단 티아졸 또는 이의 염을 유효성분으로 포함하는 알러지성 질환 또는 아토피 피부염 예방 또는 치료용 조성물

Family Cites Families (6)

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Publication number Priority date Publication date Assignee Title
EP0457803A4 (en) * 1989-02-08 1991-12-04 Abbott Laboratories 4-hydroxythiazoles as 5-lipoxygenase inhibitors
AU3201095A (en) * 1994-07-27 1996-02-22 G.D. Searle & Co. Substituted thiazoles for the treatment of inflammation
JPH11507670A (ja) * 1995-06-12 1999-07-06 ジー．ディー．サール アンド カンパニー シクロオキシゲナーゼ−２インヒビターと５−リポキシゲナーゼインヒビターの組合せによる炎症と炎症関連疾患の治療
AU7559200A (en) * 1999-10-12 2001-04-23 Japan Tobacco Inc. Hypertriglyceridemia remedies and antiobestics
HRP20040098B1 (en) * 2001-08-13 2012-08-31 Janssen Pharmaceutica N.V. 2,4,5-TRlSUBSTITUTED THIAZOLYL DERIVATIVES AND THEIR ANTIINFLAMMATORY ACTIVITY
US20050026902A1 (en) * 2003-01-31 2005-02-03 Timothy Maziasz Methods and compositions for the treatment or prevention of human immunodeficiency virus and related conditions using cyclooxygenase-2 selective inhibitors and antiviral agents

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111343975A (zh) * 2017-11-23 2020-06-26 埃慕尼克股份公司 用于预防或治疗慢性炎性疾病和/或自身免疫疾病的维多地莫的剂量方案
CN115484959A (zh) * 2020-04-16 2022-12-16 米内尔瓦有限公司 用于治疗炎症的3-氮杂-双环[3.2.1]辛烷羧酸及其衍生物

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AR072113A1 (es) 2010-08-04
JP2011524352A (ja) 2011-09-01
NZ589894A (en) 2011-08-26
MX2010013978A (es) 2011-03-29
UY31896A (es) 2010-01-29
KR20110022679A (ko) 2011-03-07
IL209801A0 (en) 2011-02-28
CA2728139A1 (en) 2009-12-23
TW201010988A (en) 2010-03-16
EP2313382A1 (en) 2011-04-27
TWI403506B (zh) 2013-08-01
RU2495031C2 (ru) 2013-10-10
RU2011101439A (ru) 2012-07-27
ZA201008877B (en) 2012-02-29
SA109300384B1 (ar) 2013-04-20
BRPI0915325A2 (pt) 2015-10-27
CO6331429A2 (es) 2011-10-20
WO2009153226A1 (en) 2009-12-23
AU2009259451B2 (en) 2013-03-14
MA32473B1 (fr) 2011-07-03
AU2009259451A1 (en) 2009-12-23

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