KR20110022679A - 급성 및 만성 염증성 질환 치료용 5-(4-메탄설포닐-페닐)-티아졸 유도체 - Google Patents

급성 및 만성 염증성 질환 치료용 5-(4-메탄설포닐-페닐)-티아졸 유도체 Download PDF

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KR20110022679A
KR20110022679A KR1020117001228A KR20117001228A KR20110022679A KR 20110022679 A KR20110022679 A KR 20110022679A KR 1020117001228 A KR1020117001228 A KR 1020117001228A KR 20117001228 A KR20117001228 A KR 20117001228A KR 20110022679 A KR20110022679 A KR 20110022679A
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compound
substituted
disease
formula
unsubstituted
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Korean (ko)
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로요 빅터 루비오
라 헤라 마르티네즈 안토니오 데
데 몬 소토 멜코르 알바레즈
무노즈 아나 무노즈
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파에스 파마, 에스.에이.
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Priority claimed from US12/139,661 external-priority patent/US7781594B2/en
Priority claimed from EP08380177A external-priority patent/EP2135864A1/en
Application filed by 파에스 파마, 에스.에이. filed Critical 파에스 파마, 에스.에이.
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33Heterocyclic compounds
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
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    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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KR1020117001228A 2008-06-16 2009-06-15 급성 및 만성 염증성 질환 치료용 5-(4-메탄설포닐-페닐)-티아졸 유도체 Ceased KR20110022679A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US12/139,661 US7781594B2 (en) 2008-06-16 2008-06-16 5-(4-methanesulfonyl-phenyl)-thiazole derivatives for the treatment of acute and chronic inflammatory diseases
US12/139,661 2008-06-16
EP08380177.9 2008-06-16
EP08380177A EP2135864A1 (en) 2008-06-16 2008-06-16 5-(4-methanesulfonyl-phenyl)-thiazole derivatives for the treatment of acute and chronic inflammatory diseases

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KR20110022679A true KR20110022679A (ko) 2011-03-07

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KR1020117001228A Ceased KR20110022679A (ko) 2008-06-16 2009-06-15 급성 및 만성 염증성 질환 치료용 5-(4-메탄설포닐-페닐)-티아졸 유도체

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EP (1) EP2313382A1 (enExample)
JP (1) JP2011524352A (enExample)
KR (1) KR20110022679A (enExample)
CN (1) CN102083806A (enExample)
AR (1) AR072113A1 (enExample)
AU (1) AU2009259451B2 (enExample)
BR (1) BRPI0915325A2 (enExample)
CA (1) CA2728139A1 (enExample)
CO (1) CO6331429A2 (enExample)
IL (1) IL209801A0 (enExample)
MA (1) MA32473B1 (enExample)
MX (1) MX2010013978A (enExample)
NZ (1) NZ589894A (enExample)
RU (1) RU2495031C2 (enExample)
SA (1) SA109300384B1 (enExample)
TW (1) TWI403506B (enExample)
UY (1) UY31896A (enExample)
WO (1) WO2009153226A1 (enExample)
ZA (1) ZA201008877B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102076936B1 (ko) * 2019-08-12 2020-02-13 연세대학교 산학협력단 티아졸 또는 이의 염을 유효성분으로 포함하는 알러지성 질환 또는 아토피 피부염 예방 또는 치료용 조성물

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2961695B1 (fr) * 2010-06-29 2012-07-06 Galderma Res & Dev Utilisation de composes dans le traitement ou la prevention de troubles cutanes
RU2502513C2 (ru) * 2012-01-11 2013-12-27 Государственное бюджетное учреждение здравоохранения Свердловской области "Свердловский областной клинический психоневрологический госпиталь для ветеранов войн" (ГБУЗ СО "СОКП Госпиталь для ветеранов войн") Способ лечения больных с полиорганной патологией озонотерапией
CN111343975A (zh) * 2017-11-23 2020-06-26 埃慕尼克股份公司 用于预防或治疗慢性炎性疾病和/或自身免疫疾病的维多地莫的剂量方案
IT202000008125A1 (it) * 2020-04-16 2021-10-16 Minerva Srl Acidi carbossilici 3-aza-biciclo[3.2.1]ottani e loro derivati per l’uso nel trattamento di infiammazioni

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0457803A4 (en) * 1989-02-08 1991-12-04 Abbott Laboratories 4-hydroxythiazoles as 5-lipoxygenase inhibitors
AU3201095A (en) * 1994-07-27 1996-02-22 G.D. Searle & Co. Substituted thiazoles for the treatment of inflammation
JPH11507670A (ja) * 1995-06-12 1999-07-06 ジー.ディー.サール アンド カンパニー シクロオキシゲナーゼ−2インヒビターと5−リポキシゲナーゼインヒビターの組合せによる炎症と炎症関連疾患の治療
AU7559200A (en) * 1999-10-12 2001-04-23 Japan Tobacco Inc. Hypertriglyceridemia remedies and antiobestics
HRP20040098B1 (en) * 2001-08-13 2012-08-31 Janssen Pharmaceutica N.V. 2,4,5-TRlSUBSTITUTED THIAZOLYL DERIVATIVES AND THEIR ANTIINFLAMMATORY ACTIVITY
US20050026902A1 (en) * 2003-01-31 2005-02-03 Timothy Maziasz Methods and compositions for the treatment or prevention of human immunodeficiency virus and related conditions using cyclooxygenase-2 selective inhibitors and antiviral agents

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR102076936B1 (ko) * 2019-08-12 2020-02-13 연세대학교 산학협력단 티아졸 또는 이의 염을 유효성분으로 포함하는 알러지성 질환 또는 아토피 피부염 예방 또는 치료용 조성물

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AR072113A1 (es) 2010-08-04
JP2011524352A (ja) 2011-09-01
NZ589894A (en) 2011-08-26
MX2010013978A (es) 2011-03-29
UY31896A (es) 2010-01-29
IL209801A0 (en) 2011-02-28
CN102083806A (zh) 2011-06-01
CA2728139A1 (en) 2009-12-23
TW201010988A (en) 2010-03-16
EP2313382A1 (en) 2011-04-27
TWI403506B (zh) 2013-08-01
RU2495031C2 (ru) 2013-10-10
RU2011101439A (ru) 2012-07-27
ZA201008877B (en) 2012-02-29
SA109300384B1 (ar) 2013-04-20
BRPI0915325A2 (pt) 2015-10-27
CO6331429A2 (es) 2011-10-20
WO2009153226A1 (en) 2009-12-23
AU2009259451B2 (en) 2013-03-14
MA32473B1 (fr) 2011-07-03
AU2009259451A1 (en) 2009-12-23

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