CN101426780B - 作为11-β-羟基甾族化合物脱氢酶1的抑制剂的环己基咪唑内酰胺衍生物 - Google Patents

作为11-β-羟基甾族化合物脱氢酶1的抑制剂的环己基咪唑内酰胺衍生物 Download PDF

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CN101426780B
CN101426780B CN2007800142250A CN200780014225A CN101426780B CN 101426780 B CN101426780 B CN 101426780B CN 2007800142250 A CN2007800142250 A CN 2007800142250A CN 200780014225 A CN200780014225 A CN 200780014225A CN 101426780 B CN101426780 B CN 101426780B
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pyrrolidin
chloro
tetrahydrochysene
benzoglyoxaline
bis
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CN101426780A (zh
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R·L·金瑟
T·E·马布里
A·萨伊德
N·J·斯奈德
O·B·怀莱士
徐彦平
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Eli Lilly and Co
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems

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CN2007800142250A 2006-04-21 2007-04-19 作为11-β-羟基甾族化合物脱氢酶1的抑制剂的环己基咪唑内酰胺衍生物 Expired - Fee Related CN101426780B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US74532106P 2006-04-21 2006-04-21
US60/745,321 2006-04-21
PCT/US2007/066907 WO2007124329A1 (en) 2006-04-21 2007-04-19 Cyclohexylimidazole lactam derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1

Publications (2)

Publication Number Publication Date
CN101426780A CN101426780A (zh) 2009-05-06
CN101426780B true CN101426780B (zh) 2013-06-26

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US (1) US7820659B2 (https=)
EP (1) EP2029576B1 (https=)
JP (1) JP5236628B2 (https=)
CN (1) CN101426780B (https=)
AU (1) AU2007240450B2 (https=)
BR (1) BRPI0710273A2 (https=)
CA (1) CA2646678C (https=)
EA (1) EA014717B1 (https=)
ES (1) ES2422165T3 (https=)
MX (1) MX2008013328A (https=)
WO (1) WO2007124329A1 (https=)

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WO2007124329A1 (en) 2007-11-01
EP2029576A1 (en) 2009-03-04
US7820659B2 (en) 2010-10-26
JP5236628B2 (ja) 2013-07-17
MX2008013328A (es) 2008-10-27
EA014717B1 (ru) 2011-02-28
AU2007240450A1 (en) 2007-11-01
CA2646678C (en) 2014-02-11
EP2029576B1 (en) 2013-06-19
CA2646678A1 (en) 2007-11-01
ES2422165T3 (es) 2013-09-09
US20090088428A1 (en) 2009-04-02
AU2007240450B2 (en) 2011-12-22
EA200870461A1 (ru) 2009-04-28
BRPI0710273A2 (pt) 2011-08-09
CN101426780A (zh) 2009-05-06

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