CN100579960C - 邻位取代的五氟化硫基苯、其制备方法和其作为有价值的合成中间体阶段形式的用途 - Google Patents

邻位取代的五氟化硫基苯、其制备方法和其作为有价值的合成中间体阶段形式的用途 Download PDF

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Publication number
CN100579960C
CN100579960C CN200480033240A CN200480033240A CN100579960C CN 100579960 C CN100579960 C CN 100579960C CN 200480033240 A CN200480033240 A CN 200480033240A CN 200480033240 A CN200480033240 A CN 200480033240A CN 100579960 C CN100579960 C CN 100579960C
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carbon atoms
formula
hydrogen
alkyl
independently
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CN200480033240A
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English (en)
Chinese (zh)
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CN1878753A (zh
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H-W·克勒曼
R·韦克
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Sanofi Aventis Deutschland GmbH
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Sanofi Aventis Deutschland GmbH
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C381/00—Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/00 - C07C337/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Indole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
CN200480033240A 2003-11-13 2004-11-03 邻位取代的五氟化硫基苯、其制备方法和其作为有价值的合成中间体阶段形式的用途 Expired - Fee Related CN100579960C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10353205A DE10353205A1 (de) 2003-11-13 2003-11-13 Ortho-substituierte Pentafluorsulfuranyl-Benzole, Verfahren zu ihrer Herstellung sowie ihre Verwendung als wertvolle Synthese-Zwischenstufen
DE10353205.6 2003-11-13

Publications (2)

Publication Number Publication Date
CN1878753A CN1878753A (zh) 2006-12-13
CN100579960C true CN100579960C (zh) 2010-01-13

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CN200480033240A Expired - Fee Related CN100579960C (zh) 2003-11-13 2004-11-03 邻位取代的五氟化硫基苯、其制备方法和其作为有价值的合成中间体阶段形式的用途

Country Status (24)

Country Link
EP (1) EP1685098B1 (https=)
JP (1) JP4516968B2 (https=)
KR (1) KR101165583B1 (https=)
CN (1) CN100579960C (https=)
AR (1) AR046619A1 (https=)
AT (1) ATE464288T1 (https=)
AU (1) AU2004288759B2 (https=)
BR (1) BRPI0416031A (https=)
CA (1) CA2545452C (https=)
CO (1) CO5690545A2 (https=)
DE (2) DE10353205A1 (https=)
DK (1) DK1685098T3 (https=)
ES (1) ES2344296T3 (https=)
IL (1) IL175239A (https=)
MY (1) MY143530A (https=)
NO (1) NO20062701L (https=)
NZ (1) NZ547171A (https=)
PE (1) PE20050493A1 (https=)
PT (1) PT1685098E (https=)
RU (1) RU2372332C2 (https=)
TW (1) TWI334412B (https=)
UY (1) UY28615A1 (https=)
WO (1) WO2005047240A1 (https=)
ZA (1) ZA200602578B (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107108490A (zh) * 2014-12-25 2017-08-29 宇部兴产株式会社 含氮五氟硫基苯化合物的制造方法

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102006036023A1 (de) 2006-08-02 2008-02-07 Sanofi-Aventis Imino-imidazo-pyridinderivate mit antithrombotischer Aktivität
KR20110098012A (ko) * 2007-02-09 2011-08-31 화이자 리미티드 구충제
SI2242740T1 (sl) 2008-02-05 2013-03-29 Sanofi SF5-derivati kot PAR1 inhibitorji, njihova priprava in uporaba kot zdravila
US8030512B2 (en) 2008-10-20 2011-10-04 Ube Industries, Ltd. Polycyclic pentafluorosulfanylbenzene compound and process for producing the compound
CN111454186B (zh) * 2019-01-18 2022-11-08 山东省联合农药工业有限公司 一种含五氟硫基的芳基甲酰苯胺类化合物及其制备方法与用途

Citations (2)

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WO1994022817A1 (en) * 1993-04-07 1994-10-13 Zeneca Limited Process for the preparation of aryl- and heteroarylsulphurpentafluorides
DE19748109A1 (de) * 1997-10-31 1999-05-06 Merck Patent Gmbh Schwefelpentafluorid-Derivate und flüssigkristallines Medium

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US5045554A (en) * 1988-11-29 1991-09-03 Monsanto Company Substituted thiazoles and their use as fungicides
US5220070A (en) * 1991-09-05 1993-06-15 The United States Of America As Represented By The Administrator National Aeronautics And Space Administration 1,3-diamino-5-pentafluorosulfanylbenzene
GB9120641D0 (en) * 1991-09-27 1991-11-06 Ici Plc Heterocyclic compounds
GB9306183D0 (en) * 1993-03-25 1993-05-19 Zeneca Ltd Novel compounds
GB9306184D0 (en) * 1993-03-25 1993-05-19 Zeneca Ltd Heteroaromatic compounds
WO1995016676A1 (en) * 1993-12-17 1995-06-22 E.I. Du Pont De Nemours And Company Arthropodicidal pentafluorothio substituted anilides
GB9515599D0 (en) * 1995-07-29 1995-09-27 British Nuclear Fuels Plc The preparation of fluorinated organic compounds
GB9606015D0 (en) * 1996-03-22 1996-05-22 Rhone Poulenc Agriculture New herbicides
KR20010034302A (ko) * 1998-01-22 2001-04-25 한스 루돌프 하우스 유기 니트릴 유도체 및 살충제로서의 이의 용도
AU7200300A (en) * 1999-12-16 2001-06-21 Rohm And Haas Company 5-carboxanilido-haloalkylthiazoles as antimicrobial and marine antifouling agents
US7151195B2 (en) * 2002-05-02 2006-12-19 Bayer Cropscience Lp Phthalamide derivative, agricultural or horticultural insecticide, and method of use thereof
JP4389243B2 (ja) * 2002-05-02 2009-12-24 日本農薬株式会社 フタルアミド誘導体及び農園芸用殺虫剤並びにその使用方法
DE10222192A1 (de) * 2002-05-18 2003-11-27 Aventis Pharma Gmbh Pentafluorsulfuranyl-benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
JP2004059452A (ja) * 2002-07-25 2004-02-26 Asahi Glass Co Ltd ペンタフルオロサルファー置換ベンズイミダゾール化合物およびその製造方法
JP2004067524A (ja) * 2002-08-01 2004-03-04 Asahi Glass Co Ltd ペンタフルオロサルファー置換インドール化合物の製造方法、ペンタフルオロサルファー置換インドール化合物およびその中間体
JP2004067525A (ja) * 2002-08-01 2004-03-04 Asahi Glass Co Ltd ペンタフルオロサルファー置換アントラニル酸誘導体の製造方法およびペンタフルオロサルファー置換アントラニル酸誘導体

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1994022817A1 (en) * 1993-04-07 1994-10-13 Zeneca Limited Process for the preparation of aryl- and heteroarylsulphurpentafluorides
DE19748109A1 (de) * 1997-10-31 1999-05-06 Merck Patent Gmbh Schwefelpentafluorid-Derivate und flüssigkristallines Medium

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
preparation of the first ortho-subsitutedpentafluorosulfanylbenzenes. journal of fluorine chemistry,Vol.112. 2001 *

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107108490A (zh) * 2014-12-25 2017-08-29 宇部兴产株式会社 含氮五氟硫基苯化合物的制造方法
CN107108490B (zh) * 2014-12-25 2019-12-31 宇部兴产株式会社 含氮五氟硫基苯化合物的制造方法

Also Published As

Publication number Publication date
DK1685098T3 (da) 2011-01-10
JP2007512246A (ja) 2007-05-17
NO20062701L (no) 2006-08-10
EP1685098A1 (de) 2006-08-02
ZA200602578B (en) 2007-06-27
KR101165583B1 (ko) 2012-07-23
AU2004288759A1 (en) 2005-05-26
AU2004288759B2 (en) 2011-04-07
CA2545452A1 (en) 2005-05-26
PT1685098E (pt) 2010-06-22
JP4516968B2 (ja) 2010-08-04
TW200530168A (en) 2005-09-16
TWI334412B (en) 2010-12-11
DE502004011054D1 (de) 2010-05-27
IL175239A (en) 2011-07-31
BRPI0416031A (pt) 2007-01-02
AR046619A1 (es) 2005-12-14
RU2006120474A (ru) 2007-12-27
UY28615A1 (es) 2005-06-30
CA2545452C (en) 2013-01-08
RU2372332C2 (ru) 2009-11-10
MY143530A (en) 2011-05-31
IL175239A0 (en) 2006-09-05
NZ547171A (en) 2009-12-24
CN1878753A (zh) 2006-12-13
KR20060111507A (ko) 2006-10-27
DE10353205A1 (de) 2005-06-16
EP1685098B1 (de) 2010-04-14
ES2344296T3 (es) 2010-08-24
CO5690545A2 (es) 2006-10-31
HK1095583A1 (zh) 2007-05-11
PE20050493A1 (es) 2005-10-07
ATE464288T1 (de) 2010-04-15
WO2005047240A1 (de) 2005-05-26

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