CL2014002034A1 - Compuestos derivados de isoxazol-fenil-azetidina fenil sustituidos; y compuestos intermediarios. - Google Patents

Compuestos derivados de isoxazol-fenil-azetidina fenil sustituidos; y compuestos intermediarios.

Info

Publication number
CL2014002034A1
CL2014002034A1 CL2014002034A CL2014002034A CL2014002034A1 CL 2014002034 A1 CL2014002034 A1 CL 2014002034A1 CL 2014002034 A CL2014002034 A CL 2014002034A CL 2014002034 A CL2014002034 A CL 2014002034A CL 2014002034 A1 CL2014002034 A1 CL 2014002034A1
Authority
CL
Chile
Prior art keywords
phenyl
compounds
isoxazol
intermediary
substituted phenyl
Prior art date
Application number
CL2014002034A
Other languages
English (en)
Spanish (es)
Inventor
Denis Billen
Sean David William Greenwood
Timothy Lee Stuk
Original Assignee
Zoetis Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zoetis Llc filed Critical Zoetis Llc
Publication of CL2014002034A1 publication Critical patent/CL2014002034A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CL2014002034A 2012-02-03 2014-07-30 Compuestos derivados de isoxazol-fenil-azetidina fenil sustituidos; y compuestos intermediarios. CL2014002034A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261594614P 2012-02-03 2012-02-03

Publications (1)

Publication Number Publication Date
CL2014002034A1 true CL2014002034A1 (es) 2014-11-14

Family

ID=47679107

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2014002034A CL2014002034A1 (es) 2012-02-03 2014-07-30 Compuestos derivados de isoxazol-fenil-azetidina fenil sustituidos; y compuestos intermediarios.

Country Status (13)

Country Link
US (1) US20140371464A1 (enExample)
EP (1) EP2809667A1 (enExample)
JP (1) JP2015505560A (enExample)
CN (1) CN104169276A (enExample)
AR (1) AR092793A1 (enExample)
AU (1) AU2013215374A1 (enExample)
BR (1) BR112014019212A8 (enExample)
CA (1) CA2863629A1 (enExample)
CL (1) CL2014002034A1 (enExample)
MX (1) MX2014009388A (enExample)
RU (1) RU2014131950A (enExample)
UY (1) UY34612A (enExample)
WO (1) WO2013116236A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2872989A1 (en) * 2012-05-09 2013-11-14 Zoetis Llc Azetidine derivatives as antiparasitic agents
UY37137A (es) 2016-02-24 2017-09-29 Merial Inc Compuestos antiparasitarios de isoxazolina, formulaciones inyectables de acción prolongada que los comprenden, métodos y usos de los mismos
DK3440062T3 (da) 2016-04-06 2022-01-03 Boehringer Ingelheim Animal Health Usa Inc Fremgangsmåde til fremstillingen af enantiomerisk berigede isoxazolinforbindelser - krystallinsk toluensolvat af (s)-afoxolaner
MX380497B (es) 2016-10-14 2025-03-11 Boehringer Ingelheim Animal Health Usa Inc Compuestos de vinil isoxazolina pesticidas y parasiticidas.
MX2020001724A (es) 2017-08-14 2020-07-29 Boehringer Ingelheim Animal Health Usa Inc Compuestos de pirazol-isoxazolina plaguicidas y parasiticidas.
EP3986878B1 (en) * 2019-06-19 2024-09-25 NMD Pharma A/S Process for the preparation of clc-1 chloride channel inhibitors
KR20230043904A (ko) 2020-07-24 2023-03-31 엘랑코 유에스 인코포레이티드 이속사졸린 화합물 및 이의 중간체의 제조 공정
MX2023014962A (es) 2021-08-11 2024-02-13 Elanco Us Inc Proceso para elaborar derivado de diaril isoxazolina.

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200803740A (en) 2005-12-16 2008-01-16 Du Pont 5-aryl isoxazolines for controlling invertebrate pests
CN101331127B (zh) * 2005-12-16 2012-05-23 杜邦公司 用于防治无脊椎害虫的5-芳基异噁唑啉
WO2007105814A1 (ja) 2006-03-10 2007-09-20 Nissan Chemical Industries, Ltd. 置換イソキサゾリン化合物及び有害生物防除剤
JP2008044880A (ja) * 2006-08-15 2008-02-28 Bayer Cropscience Ag 殺虫性イソオキサゾリン類
US8303622B2 (en) 2007-03-14 2012-11-06 St. Jude Medical, Inc. Heart valve chordae replacement methods and apparatus
JP2008260691A (ja) * 2007-04-10 2008-10-30 Bayer Cropscience Ag 殺虫性アリールイソオキサゾリン誘導体
JP5365806B2 (ja) 2007-09-10 2013-12-11 日産化学工業株式会社 置換イソキサゾリン化合物及び有害生物防除剤
WO2009063910A1 (ja) 2007-11-12 2009-05-22 Nissan Chemical Industries, Ltd. 光学活性イソキサゾリン化合物の触媒的不斉合成方法
BRPI0923009B1 (pt) * 2008-12-19 2018-07-17 Elanco Tiergesundheit Ag compostos de isoxazolina, composição para o controle de parasitas e uso de compostos de isoxazolina para o preparo de composição para o controle de parasitas
CN102822168B (zh) 2010-02-25 2016-10-26 先正达参股股份有限公司 制备异恶唑啉衍生物的方法
PH12013500164A1 (en) * 2010-08-05 2015-07-08 Zoetis Services Llc Isoxazoline derivatives as antiparasitic agents

Also Published As

Publication number Publication date
US20140371464A1 (en) 2014-12-18
AU2013215374A1 (en) 2014-08-21
BR112014019212A8 (pt) 2017-07-11
UY34612A (es) 2013-09-30
AR092793A1 (es) 2015-05-06
RU2014131950A (ru) 2016-03-27
WO2013116236A1 (en) 2013-08-08
JP2015505560A (ja) 2015-02-23
CA2863629A1 (en) 2013-08-08
CN104169276A (zh) 2014-11-26
MX2014009388A (es) 2014-08-27
EP2809667A1 (en) 2014-12-10
BR112014019212A2 (enExample) 2017-06-20

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