CL2012000314A1 - Compuesto derivado de n1-sustituido-5-fluoro-2-oxopirimidina-1(2h)-carboxamida; composición que lo comprende; y método para el control y prevención de un ataque fúngico en una planta. - Google Patents

Compuesto derivado de n1-sustituido-5-fluoro-2-oxopirimidina-1(2h)-carboxamida; composición que lo comprende; y método para el control y prevención de un ataque fúngico en una planta.

Info

Publication number
CL2012000314A1
CL2012000314A1 CL2012000314A CL2012000314A CL2012000314A1 CL 2012000314 A1 CL2012000314 A1 CL 2012000314A1 CL 2012000314 A CL2012000314 A CL 2012000314A CL 2012000314 A CL2012000314 A CL 2012000314A CL 2012000314 A1 CL2012000314 A1 CL 2012000314A1
Authority
CL
Chile
Prior art keywords
substituted
alkyl
oxopyrimidine
carboxamide
fluoro
Prior art date
Application number
CL2012000314A
Other languages
English (en)
Spanish (es)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Timothy Martin
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2012000314(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of CL2012000314A1 publication Critical patent/CL2012000314A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/20Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D239/22Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
CL2012000314A 2009-08-07 2012-02-06 Compuesto derivado de n1-sustituido-5-fluoro-2-oxopirimidina-1(2h)-carboxamida; composición que lo comprende; y método para el control y prevención de un ataque fúngico en una planta. CL2012000314A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23223209P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
CL2012000314A1 true CL2012000314A1 (es) 2012-10-05

Family

ID=43535293

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2012000314A CL2012000314A1 (es) 2009-08-07 2012-02-06 Compuesto derivado de n1-sustituido-5-fluoro-2-oxopirimidina-1(2h)-carboxamida; composición que lo comprende; y método para el control y prevención de un ataque fúngico en una planta.

Country Status (28)

Country Link
US (1) US8318758B2 (enFirst)
EP (1) EP2462133B1 (enFirst)
JP (1) JP5818791B2 (enFirst)
KR (1) KR101792286B1 (enFirst)
CN (1) CN102548979B (enFirst)
AU (1) AU2010279408B2 (enFirst)
BR (1) BR112012002807B1 (enFirst)
CA (1) CA2769251C (enFirst)
CL (1) CL2012000314A1 (enFirst)
CO (1) CO6491089A2 (enFirst)
CR (1) CR20120033A (enFirst)
DK (1) DK2462133T3 (enFirst)
EA (1) EA022930B1 (enFirst)
EC (1) ECSP12011651A (enFirst)
ES (1) ES2506169T3 (enFirst)
HN (1) HN2012000261A (enFirst)
IL (1) IL217954A (enFirst)
IN (1) IN2012DN00695A (enFirst)
MX (1) MX2012001623A (enFirst)
NI (1) NI201200019A (enFirst)
NZ (1) NZ597638A (enFirst)
PE (1) PE20120689A1 (enFirst)
PL (1) PL2462133T3 (enFirst)
PT (1) PT2462133E (enFirst)
RS (1) RS53658B1 (enFirst)
UA (1) UA106086C2 (enFirst)
WO (1) WO2011017544A1 (enFirst)
ZA (1) ZA201305992B (enFirst)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA022289B1 (ru) * 2009-08-07 2015-12-30 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Производные n1-сульфонил-5-фторпиримидинона
RU2015131149A (ru) 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные
DK2938194T3 (da) 2012-12-28 2020-01-02 Adama Makhteshim Ltd N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater
CN104994859B (zh) 2012-12-28 2018-10-26 阿达玛马克西姆股份有限公司 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物
WO2014105845A1 (en) 2012-12-31 2014-07-03 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
JP6585057B2 (ja) 2013-12-31 2019-10-02 アダマ・マクテシム・リミテッド 5−フルオロ−4−イミノ−3−(アルキル/置換アルキル)−1−(アリールスルホニル)−3,4−ジヒドロピリミジン−2(1h)−オンおよびそれらの調製方法
AP2016009341A0 (en) 2013-12-31 2016-07-31 Adama Makhteshim Ltd Synergistic fungicidal mixtures for fungal control in cereals
WO2016040193A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
CN108472290A (zh) 2015-11-06 2018-08-31 萨穆梅德有限公司 治疗骨关节炎
CN109476660B (zh) 2016-06-01 2023-04-04 拜斯丽治疗有限公司 N-(5-(3-(7-(3-氟苯基)-3h-咪唑并[4,5-c]吡啶-2-基)-1h-吲唑-5-基)吡啶-3-基)-3-甲基丁酰胺的制备方法
CN111094252B (zh) 2017-07-17 2024-05-24 阿达玛克西姆股份有限公司 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物
JP7701266B2 (ja) 2018-11-05 2025-07-01 アダマ・マクテシム・リミテッド 5-フルオロ-4-イミノ-3-メチル-1-トシル-3,4-ジヒドロピリミジン-2-オンを含む混合物および組成物、ならびにそれらの使用方法
US12466796B2 (en) 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
EP0888359B1 (en) * 1996-03-11 2002-05-02 Syngenta Participations AG Pyrimidin-4-one derivatives as pesticide
AU2003274652A1 (en) * 2002-10-23 2004-05-13 Obetherapy Biotechnology Compounds, compositions and methods for modulating fat metabolism
CN101730691A (zh) * 2007-04-27 2010-06-09 阿斯比奥制药株式会社 含氮芳香族六元环衍生物及含有它们的药物
US20100029482A1 (en) * 2008-08-01 2010-02-04 Benko Zoltan L Use of 5-fluorocytosine as a fungicide

Also Published As

Publication number Publication date
JP2013501726A (ja) 2013-01-17
BR112012002807A8 (pt) 2017-07-11
ES2506169T3 (es) 2014-10-13
CN102548979B (zh) 2015-05-13
WO2011017544A1 (en) 2011-02-10
CO6491089A2 (es) 2012-07-31
IL217954A0 (en) 2012-03-29
CR20120033A (es) 2012-03-22
KR101792286B1 (ko) 2017-10-31
US20110034491A1 (en) 2011-02-10
MX2012001623A (es) 2012-04-11
KR20120043069A (ko) 2012-05-03
ZA201305992B (en) 2014-10-29
PE20120689A1 (es) 2012-06-06
BR112012002807A2 (pt) 2015-10-13
CN102548979A (zh) 2012-07-04
RS53658B1 (sr) 2015-04-30
IN2012DN00695A (enFirst) 2015-06-19
BR112012002807B1 (pt) 2018-07-10
EA201270255A1 (ru) 2012-07-30
EP2462133A1 (en) 2012-06-13
EP2462133B1 (en) 2014-09-24
IL217954A (en) 2016-02-29
PL2462133T3 (pl) 2015-03-31
HK1172892A1 (en) 2013-05-03
AU2010279408A1 (en) 2012-02-09
AU2010279408B2 (en) 2015-09-10
HN2012000261A (es) 2015-01-05
NI201200019A (es) 2012-05-22
UA106086C2 (uk) 2014-07-25
PT2462133E (pt) 2014-12-26
JP5818791B2 (ja) 2015-11-18
CA2769251A1 (en) 2011-02-10
EP2462133A4 (en) 2013-01-16
DK2462133T3 (en) 2015-01-05
NZ597638A (en) 2014-06-27
CA2769251C (en) 2018-05-15
US8318758B2 (en) 2012-11-27
EA022930B1 (ru) 2016-03-31
ECSP12011651A (es) 2012-03-30

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