CL2011003302A1 - Compuestos derivados de amida del acido alquil-sulfonico; composicion farmaceutica; uso de los compuestos como moduladores de la disfuncion de glutamato para prevenir o tratar trastornos neurologicos y psiquiatricos como esquizofrenia, enfermedad de alzheimer, trastornos de deficit de atencion/hiperactividad, perdida de audicion, entre otros. - Google Patents

Compuestos derivados de amida del acido alquil-sulfonico; composicion farmaceutica; uso de los compuestos como moduladores de la disfuncion de glutamato para prevenir o tratar trastornos neurologicos y psiquiatricos como esquizofrenia, enfermedad de alzheimer, trastornos de deficit de atencion/hiperactividad, perdida de audicion, entre otros.

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Publication number
CL2011003302A1
CL2011003302A1 CL2011003302A CL2011003302A CL2011003302A1 CL 2011003302 A1 CL2011003302 A1 CL 2011003302A1 CL 2011003302 A CL2011003302 A CL 2011003302A CL 2011003302 A CL2011003302 A CL 2011003302A CL 2011003302 A1 CL2011003302 A1 CL 2011003302A1
Authority
CL
Chile
Prior art keywords
compounds
disorders
schizophrenia
pharmaceutical composition
prevent
Prior art date
Application number
CL2011003302A
Other languages
English (en)
Inventor
Anton Franz Joseph Fliri
Randall James Gallaschun
Christopher John O´Donnell
Jacob Bradley Schwarz
Barbara SEGELSTEIN
Original Assignee
Pfizer
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43127233&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2011003302(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of CL2011003302A1 publication Critical patent/CL2011003302A1/es

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    • C07C307/02—Monoamides of sulfuric acids or esters thereof, e.g. sulfamic acids
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • C07C311/07—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
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Abstract

UN COMPUESTO DERIVADO DE FORMULA 1, O UNA SAL FARMACÉUTICAMENTE ACEPTABLE DEL MISMO. SE DESCRIBE UNA COMPOSICIÓN FARMACÉUTICA QUE COMPRENDE DICHO COMPUESTO, ADEMÁS DE SU USO PARA PREVENIR O TRATAR TRASTORNOS NEUROLÓGICOS Y PSIQUIÁTRICOS COMO LA ESQUIZOFRENIA, PÉRDIDA DE AUDICIÓN, ENTRE OTROS.
CL2011003302A 2009-06-26 2011-12-26 Compuestos derivados de amida del acido alquil-sulfonico; composicion farmaceutica; uso de los compuestos como moduladores de la disfuncion de glutamato para prevenir o tratar trastornos neurologicos y psiquiatricos como esquizofrenia, enfermedad de alzheimer, trastornos de deficit de atencion/hiperactividad, perdida de audicion, entre otros. CL2011003302A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US22062509P 2009-06-26 2009-06-26

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CL2011003302A1 true CL2011003302A1 (es) 2012-07-13

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CL2011003302A CL2011003302A1 (es) 2009-06-26 2011-12-26 Compuestos derivados de amida del acido alquil-sulfonico; composicion farmaceutica; uso de los compuestos como moduladores de la disfuncion de glutamato para prevenir o tratar trastornos neurologicos y psiquiatricos como esquizofrenia, enfermedad de alzheimer, trastornos de deficit de atencion/hiperactividad, perdida de audicion, entre otros.

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WO2024033374A1 (en) 2022-08-11 2024-02-15 Syngenta Crop Protection Ag Novel arylcarboxamide or arylthioamide compounds
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