CL2007003686A1 - Compuestos derivados de indol con anillo unido en las posiciones 4,5; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para tratar una infeccion viral. - Google Patents

Compuestos derivados de indol con anillo unido en las posiciones 4,5; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para tratar una infeccion viral.

Info

Publication number
CL2007003686A1
CL2007003686A1 CL200703686A CL2007003686A CL2007003686A1 CL 2007003686 A1 CL2007003686 A1 CL 2007003686A1 CL 200703686 A CL200703686 A CL 200703686A CL 2007003686 A CL2007003686 A CL 2007003686A CL 2007003686 A1 CL2007003686 A1 CL 2007003686A1
Authority
CL
Chile
Prior art keywords
compound
indol
treat
positions
pharmaceutical composition
Prior art date
Application number
CL200703686A
Other languages
English (en)
Inventor
Kevin X Venkatraman Srika Chen
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39186835&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2007003686(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Publication of CL2007003686A1 publication Critical patent/CL2007003686A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
CL200703686A 2006-12-22 2007-12-18 Compuestos derivados de indol con anillo unido en las posiciones 4,5; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para tratar una infeccion viral. CL2007003686A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US87687706P 2006-12-22 2006-12-22

Publications (1)

Publication Number Publication Date
CL2007003686A1 true CL2007003686A1 (es) 2008-06-27

Family

ID=39186835

Family Applications (1)

Application Number Title Priority Date Filing Date
CL200703686A CL2007003686A1 (es) 2006-12-22 2007-12-18 Compuestos derivados de indol con anillo unido en las posiciones 4,5; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para tratar una infeccion viral.

Country Status (18)

Country Link
US (1) US8557848B2 (es)
EP (1) EP2064180B1 (es)
JP (1) JP5079818B2 (es)
KR (1) KR20090094154A (es)
CN (1) CN101631773A (es)
AR (1) AR064428A1 (es)
AU (1) AU2007339382B2 (es)
BR (1) BRPI0720625A2 (es)
CA (1) CA2673249C (es)
CL (1) CL2007003686A1 (es)
CO (1) CO6190515A2 (es)
EC (1) ECSP099447A (es)
MX (1) MX2009006880A (es)
NO (1) NO20092742L (es)
PE (1) PE20081608A1 (es)
RU (1) RU2009127855A (es)
TW (1) TW200831496A (es)
WO (1) WO2008082484A1 (es)

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US8404845B2 (en) * 2007-08-29 2013-03-26 Merck Sharp & Dohme Corp. 2,3-substituted azaindole derivatives for treating viral infections
US8143305B2 (en) * 2007-08-29 2012-03-27 Schering Corporation 2,3-substituted indole derivatives for treating viral infections
WO2009032124A1 (en) * 2007-08-29 2009-03-12 Schering Corporation Substituted indole derivatives and methods of use thereof
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US9457039B2 (en) 2012-10-17 2016-10-04 Merck Sharp & Dohme Corp. 2′-disubstituted nucleoside derivatives and methods of use thereof for the treatment of viral diseases
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CN106810557B (zh) * 2015-11-27 2021-05-04 南京圣和药物研发有限公司 杂环化合物及其应用
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Also Published As

Publication number Publication date
JP5079818B2 (ja) 2012-11-21
PE20081608A1 (es) 2008-11-12
EP2064180B1 (en) 2016-07-13
AU2007339382B2 (en) 2013-05-02
EP2064180A1 (en) 2009-06-03
US20100098661A1 (en) 2010-04-22
AR064428A1 (es) 2009-04-01
MX2009006880A (es) 2009-07-03
CN101631773A (zh) 2010-01-20
BRPI0720625A2 (pt) 2014-03-25
CA2673249A1 (en) 2008-07-10
WO2008082484A1 (en) 2008-07-10
KR20090094154A (ko) 2009-09-03
CA2673249C (en) 2013-04-30
RU2009127855A (ru) 2011-01-27
JP2010513490A (ja) 2010-04-30
CO6190515A2 (es) 2010-08-19
ECSP099447A (es) 2009-07-31
TW200831496A (en) 2008-08-01
AU2007339382A1 (en) 2008-07-10
US8557848B2 (en) 2013-10-15
NO20092742L (no) 2009-09-21

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