CH654209A5 - 2-pyrazolinderivate und diese enthaltende pharmazeutische zubereitung. - Google Patents

2-pyrazolinderivate und diese enthaltende pharmazeutische zubereitung. Download PDF

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Publication number
CH654209A5
CH654209A5 CH8003/81A CH800381A CH654209A5 CH 654209 A5 CH654209 A5 CH 654209A5 CH 8003/81 A CH8003/81 A CH 8003/81A CH 800381 A CH800381 A CH 800381A CH 654209 A5 CH654209 A5 CH 654209A5
Authority
CH
Switzerland
Prior art keywords
pyrazoline
substituted
trifluoromethylphenyl
phenyl
alkyl
Prior art date
Application number
CH8003/81A
Other languages
German (de)
English (en)
Inventor
Frederick Charles Copp
Albert Gordon Caldwell
David Collard
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of CH654209A5 publication Critical patent/CH654209A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/76Nitrogen atoms to which a second hetero atom is attached
    • C07D213/77Hydrazine radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH8003/81A 1980-12-16 1981-12-15 2-pyrazolinderivate und diese enthaltende pharmazeutische zubereitung. CH654209A5 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8040172 1980-12-16
US25607281A 1981-04-21 1981-04-21

Publications (1)

Publication Number Publication Date
CH654209A5 true CH654209A5 (de) 1986-02-14

Family

ID=26277856

Family Applications (1)

Application Number Title Priority Date Filing Date
CH8003/81A CH654209A5 (de) 1980-12-16 1981-12-15 2-pyrazolinderivate und diese enthaltende pharmazeutische zubereitung.

Country Status (18)

Country Link
EP (1) EP0055418B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AT (1) AT379803B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU559488B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA1180335A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CH (1) CH654209A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (2) DE3149710A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK556381A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES8307224A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (1) FI814024L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FR (1) FR2496100B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GR (1) GR76989B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HU (1) HU187392B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IE (1) IE51951B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL64555A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MC (1) MC1435A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NL (1) NL8105652A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NZ (1) NZ199288A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SE (1) SE8107524L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0070376A1 (en) * 1981-07-13 1983-01-26 American Cyanamid Company Heterocyclic substituted-amino-pyrazolines
GB8303782D0 (en) * 1983-02-11 1983-03-16 Wellcome Found Heterocyclic compounds
EP0119450A1 (en) * 1983-02-11 1984-09-26 The Wellcome Foundation Limited Preparation of aminopyrazolines and intermediates used therein
US4824859A (en) * 1983-05-21 1989-04-25 Fisons Plc. Pyrazoline compounds compositions and use
EP0178035B1 (en) * 1984-05-12 1990-01-03 FISONS plc Anti-inflammatory 1,n-diarylpyrazol-3-amines, compositions containing them and processes for their preparation
US4970210A (en) * 1987-07-17 1990-11-13 Abbott Laboratories Triazinone lipoxygenase compounds
FR2781147B1 (fr) 1998-07-20 2000-09-15 Oreal Compositions pour la teinture des fibres keratiniques contenant des derives de 3-amino pyrazolines a titre de coupleur, procede de teinture et kit de teinture
GB0603181D0 (en) * 2006-02-17 2006-03-29 Merck Sharp & Dohme Treatment of neurodegenerative and psychiatric diseases
WO2025166015A2 (en) * 2024-02-02 2025-08-07 Photys Therapeutics, Inc. Bifunctional abl1-binding compounds and uses thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES313450A1 (es) * 1964-05-27 1966-02-16 Geigy Ag J R Procedimiento para la preparacion de compuestos de pirazolina.
FR2059449A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * 1969-02-26 1971-06-04 Synthelabo
IT1207128B (it) * 1979-07-13 1989-05-17 Wellcome Found Composizioni farmaceutiche contenenti composti eterociclici derivati dalla pirazolina ad attivita'anti spasmodica e procedimento per laloro preparazione

Also Published As

Publication number Publication date
DK556381A (da) 1982-06-17
IE51951B1 (en) 1987-04-29
EP0055418B1 (en) 1986-02-26
DE3173933D1 (en) 1986-04-03
ATA537281A (de) 1985-07-15
GR76989B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1984-09-04
EP0055418A2 (en) 1982-07-07
HU187392B (en) 1985-12-28
NL8105652A (nl) 1982-07-16
FR2496100A1 (fr) 1982-06-18
CA1180335A (en) 1985-01-02
DE3149710A1 (de) 1982-08-05
ES507975A0 (es) 1983-06-16
SE8107524L (sv) 1982-06-17
AT379803B (de) 1986-03-10
MC1435A1 (fr) 1982-12-06
FI814024A7 (fi) 1982-06-17
NZ199288A (en) 1985-07-31
FR2496100B1 (fr) 1985-06-14
ES8307224A1 (es) 1983-06-16
IL64555A (en) 1986-01-31
IE812944L (en) 1982-06-16
IL64555A0 (en) 1982-03-31
FI814024L (fi) 1982-06-17
AU559488B2 (en) 1987-03-12
AU7851081A (en) 1982-06-24
EP0055418A3 (en) 1982-08-18

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PL Patent ceased