CA1180335A - 3-amino-1-aryl-2-pyrazoline compounds - Google Patents
3-amino-1-aryl-2-pyrazoline compoundsInfo
- Publication number
- CA1180335A CA1180335A CA000392319A CA392319A CA1180335A CA 1180335 A CA1180335 A CA 1180335A CA 000392319 A CA000392319 A CA 000392319A CA 392319 A CA392319 A CA 392319A CA 1180335 A CA1180335 A CA 1180335A
- Authority
- CA
- Canada
- Prior art keywords
- alkyl
- formula
- hydrogen
- compound
- pyrazoline
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/76—Nitrogen atoms to which a second hetero atom is attached
- C07D213/77—Hydrazine radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8040172 | 1980-12-16 | ||
| GB8040172 | 1980-12-16 | ||
| US25607281A | 1981-04-21 | 1981-04-21 | |
| US256,072 | 1981-04-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA1180335A true CA1180335A (en) | 1985-01-02 |
Family
ID=26277856
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA000392319A Expired CA1180335A (en) | 1980-12-16 | 1981-12-15 | 3-amino-1-aryl-2-pyrazoline compounds |
Country Status (18)
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0070376A1 (en) * | 1981-07-13 | 1983-01-26 | American Cyanamid Company | Heterocyclic substituted-amino-pyrazolines |
| GB8303782D0 (en) * | 1983-02-11 | 1983-03-16 | Wellcome Found | Heterocyclic compounds |
| EP0119450A1 (en) * | 1983-02-11 | 1984-09-26 | The Wellcome Foundation Limited | Preparation of aminopyrazolines and intermediates used therein |
| US4824859A (en) * | 1983-05-21 | 1989-04-25 | Fisons Plc. | Pyrazoline compounds compositions and use |
| EP0178035B1 (en) * | 1984-05-12 | 1990-01-03 | FISONS plc | Anti-inflammatory 1,n-diarylpyrazol-3-amines, compositions containing them and processes for their preparation |
| US4970210A (en) * | 1987-07-17 | 1990-11-13 | Abbott Laboratories | Triazinone lipoxygenase compounds |
| FR2781147B1 (fr) | 1998-07-20 | 2000-09-15 | Oreal | Compositions pour la teinture des fibres keratiniques contenant des derives de 3-amino pyrazolines a titre de coupleur, procede de teinture et kit de teinture |
| GB0603181D0 (en) * | 2006-02-17 | 2006-03-29 | Merck Sharp & Dohme | Treatment of neurodegenerative and psychiatric diseases |
| WO2025166015A2 (en) * | 2024-02-02 | 2025-08-07 | Photys Therapeutics, Inc. | Bifunctional abl1-binding compounds and uses thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES313450A1 (es) * | 1964-05-27 | 1966-02-16 | Geigy Ag J R | Procedimiento para la preparacion de compuestos de pirazolina. |
| FR2059449A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1969-02-26 | 1971-06-04 | Synthelabo | |
| IT1207128B (it) * | 1979-07-13 | 1989-05-17 | Wellcome Found | Composizioni farmaceutiche contenenti composti eterociclici derivati dalla pirazolina ad attivita'anti spasmodica e procedimento per laloro preparazione |
-
1981
- 1981-12-15 GR GR66797A patent/GR76989B/el unknown
- 1981-12-15 IE IE2944/81A patent/IE51951B1/en unknown
- 1981-12-15 ES ES507975A patent/ES8307224A1/es not_active Expired
- 1981-12-15 DE DE19813149710 patent/DE3149710A1/de not_active Withdrawn
- 1981-12-15 NZ NZ199288A patent/NZ199288A/en unknown
- 1981-12-15 AT AT0537281A patent/AT379803B/de not_active IP Right Cessation
- 1981-12-15 CA CA000392319A patent/CA1180335A/en not_active Expired
- 1981-12-15 HU HU813771A patent/HU187392B/hu unknown
- 1981-12-15 EP EP81110457A patent/EP0055418B1/en not_active Expired
- 1981-12-15 AU AU78510/81A patent/AU559488B2/en not_active Expired - Fee Related
- 1981-12-15 NL NL8105652A patent/NL8105652A/nl not_active Application Discontinuation
- 1981-12-15 FR FR8123367A patent/FR2496100B1/fr not_active Expired
- 1981-12-15 MC MC811566A patent/MC1435A1/xx unknown
- 1981-12-15 CH CH8003/81A patent/CH654209A5/de not_active IP Right Cessation
- 1981-12-15 DK DK556381A patent/DK556381A/da not_active Application Discontinuation
- 1981-12-15 DE DE8181110457T patent/DE3173933D1/de not_active Expired
- 1981-12-15 FI FI814024A patent/FI814024L/fi not_active Application Discontinuation
- 1981-12-15 IL IL64555A patent/IL64555A/xx unknown
- 1981-12-15 SE SE8107524A patent/SE8107524L/xx not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| DK556381A (da) | 1982-06-17 |
| CH654209A5 (de) | 1986-02-14 |
| IE51951B1 (en) | 1987-04-29 |
| EP0055418B1 (en) | 1986-02-26 |
| DE3173933D1 (en) | 1986-04-03 |
| ATA537281A (de) | 1985-07-15 |
| GR76989B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1984-09-04 |
| EP0055418A2 (en) | 1982-07-07 |
| HU187392B (en) | 1985-12-28 |
| NL8105652A (nl) | 1982-07-16 |
| FR2496100A1 (fr) | 1982-06-18 |
| DE3149710A1 (de) | 1982-08-05 |
| ES507975A0 (es) | 1983-06-16 |
| SE8107524L (sv) | 1982-06-17 |
| AT379803B (de) | 1986-03-10 |
| MC1435A1 (fr) | 1982-12-06 |
| FI814024A7 (fi) | 1982-06-17 |
| NZ199288A (en) | 1985-07-31 |
| FR2496100B1 (fr) | 1985-06-14 |
| ES8307224A1 (es) | 1983-06-16 |
| IL64555A (en) | 1986-01-31 |
| IE812944L (en) | 1982-06-16 |
| IL64555A0 (en) | 1982-03-31 |
| FI814024L (fi) | 1982-06-17 |
| AU559488B2 (en) | 1987-03-12 |
| AU7851081A (en) | 1982-06-24 |
| EP0055418A3 (en) | 1982-08-18 |
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| GB2093832A (en) | Pyrazoline derivatives | |
| EP0119449A1 (en) | Aminopyrazoline derivatives |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MKEX | Expiry |