CH635838A5 - Process for preparing nitrogen-containing heterocyclic carbonylpiperazinylquinazolines - Google Patents

Process for preparing nitrogen-containing heterocyclic carbonylpiperazinylquinazolines Download PDF

Info

Publication number
CH635838A5
CH635838A5 CH199477A CH199477A CH635838A5 CH 635838 A5 CH635838 A5 CH 635838A5 CH 199477 A CH199477 A CH 199477A CH 199477 A CH199477 A CH 199477A CH 635838 A5 CH635838 A5 CH 635838A5
Authority
CH
Switzerland
Prior art keywords
amino
dimethoxy
prazosin
carbonyl
quinazoline
Prior art date
Application number
CH199477A
Other languages
German (de)
English (en)
Inventor
Richard Anthony Partyka
Ronnie Ray Crenshaw
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/658,961 external-priority patent/US4001237A/en
Priority claimed from US05/658,979 external-priority patent/US4001238A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of CH635838A5 publication Critical patent/CH635838A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH199477A 1976-02-18 1977-02-17 Process for preparing nitrogen-containing heterocyclic carbonylpiperazinylquinazolines CH635838A5 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/658,961 US4001237A (en) 1976-02-18 1976-02-18 Oxazole, isoxazole, thiazole and isothiazole amides
US05/658,979 US4001238A (en) 1976-02-18 1976-02-18 1,3,4-oxadiazole amides

Publications (1)

Publication Number Publication Date
CH635838A5 true CH635838A5 (en) 1983-04-29

Family

ID=27097727

Family Applications (1)

Application Number Title Priority Date Filing Date
CH199477A CH635838A5 (en) 1976-02-18 1977-02-17 Process for preparing nitrogen-containing heterocyclic carbonylpiperazinylquinazolines

Country Status (16)

Country Link
JP (1) JPS584716B2 (xx)
CA (1) CA1081228A (xx)
CH (1) CH635838A5 (xx)
CY (1) CY1122A (xx)
DE (1) DE2707067A1 (xx)
DK (1) DK65177A (xx)
FI (1) FI770485A (xx)
FR (1) FR2348924A1 (xx)
GB (1) GB1533529A (xx)
IE (1) IE44614B1 (xx)
KE (1) KE3155A (xx)
LU (1) LU76802A1 (xx)
MY (1) MY8200110A (xx)
NL (1) NL7701753A (xx)
SE (1) SE7701732L (xx)
YU (4) YU45477A (xx)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5791987A (en) * 1980-11-26 1982-06-08 Sankyo Co Ltd Aminoquinazoline derivative and its preparation
US5932538A (en) * 1996-02-02 1999-08-03 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
US5994294A (en) * 1996-02-02 1999-11-30 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
AU2003246571B2 (en) * 2002-06-29 2008-06-26 Zentaris Gmbh Arylcarbonylpiperazines and heteroarylcarbonylpiperazines and the use thereof for treating benign and malignant tumour diseases

Also Published As

Publication number Publication date
CY1122A (en) 1981-12-04
IE44614B1 (en) 1982-01-27
SE7701732L (sv) 1977-08-19
YU45477A (en) 1982-10-31
JPS584716B2 (ja) 1983-01-27
YU267780A (en) 1983-06-30
YU161182A (en) 1982-10-31
CA1081228A (en) 1980-07-08
KE3155A (en) 1981-09-18
NL7701753A (nl) 1977-08-22
AU2242677A (en) 1978-07-06
GB1533529A (en) 1978-11-29
FI770485A (xx) 1977-08-19
DK65177A (da) 1977-08-19
DE2707067A1 (de) 1977-08-25
LU76802A1 (xx) 1977-09-12
IE44614L (en) 1977-08-18
YU161282A (en) 1982-10-31
JPS52102286A (en) 1977-08-27
FR2348924A1 (fr) 1977-11-18
MY8200110A (en) 1982-12-31
FR2348924B1 (xx) 1980-05-09

Similar Documents

Publication Publication Date Title
DE3852555T2 (de) Substituierte 2-Aminobenzothiazole und Derivate verwendbar als cerebrovasculare Mittel.
US4001238A (en) 1,3,4-oxadiazole amides
DE69431880T2 (de) Verwendung von (2-imidazolin-2-yl-amino) quinoxalinderivaten
DE2120495C2 (de) 2-Methyl-2-hydroxypropyl-4-(4-amino-6,7,8-trimethoxychinazolin-2-yl)-1-piperazincarboxylat
US4001237A (en) Oxazole, isoxazole, thiazole and isothiazole amides
DE2904445C2 (de) N↓1↓-(4-Amino-6.7-dimethoxy-2-chinazolyl)-N↓1↓-methyl-N↓2↓-(2-tetrahydrofuroyl)-1.3-propandiamin, seine Herstellung und seine pharmazeutische Verwendung
DE2807392A1 (de) Neue chinazolinverbindungen, verfahren zu deren herstellung und diese enthaltende arzneimittel
CH667268A5 (de) 1,2-benzisothiazol-3-ylpiperazine.
DE19922443A1 (de) Verwendung von Dopamin-D3-Rezeptorliganden zur Herstellung von Arzneimittel für die Behandlung von Nierenfunktionsstörungen
DE69219271T2 (de) Acridinederivat als therapeutisches Mittel
DD207913A5 (de) Verfahren zur herstellung von 2-guanidino-4-heteroarylthiazolen
DE2415082A1 (de) Disubstituierte piperazine, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel
DE69326459T2 (de) Wirkstoffe zur behandlung von suchterkrankungen
DE2720545C3 (de) Derivate des 2,4-Diamino-6,7-dimethoxychinazolins, ihre Herstellung und pharmazeutische Mittel
DE69311566T2 (de) Heterocyclische amine als calmodulin antagonisten
EP0764022B1 (de) Agonisten und antagonisten der nicotinergen acetylcholinrezeptoren von insekten als endoparasitizide
DD281596A5 (de) Verfahren zur hersteung antiarrhytmischer mittel
CH635838A5 (en) Process for preparing nitrogen-containing heterocyclic carbonylpiperazinylquinazolines
DE60009287T2 (de) Neuartige isoquinolin-derivate oder salze davon
DE3309655A1 (de) 1,2,5-thiadiazol-1-oxide und 1,1-dioxide, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
DE3233424A1 (de) Isochinolinderivate, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen und ihre verwendung
DE2845857C2 (de) Benzo [d] thiazolderivate, Verfahren zu ihrer Herstellung und sie enthaltende Arzneimittelzubereitungen
DE69426620T2 (de) Antidepressiva
DE60311233T2 (de) Chinolinderivate
CH637391A5 (de) Therapeutisch wirksame 3-(1-piperazinyl)-1,2,4-benzotriazine und ihre n-oxide.

Legal Events

Date Code Title Description
PL Patent ceased