KE3155A - 4-amino-6,7-dimethoxy-2(4-(heterocyclocarbonyl)piperazin-1-yl)quinazolines - Google Patents

4-amino-6,7-dimethoxy-2(4-(heterocyclocarbonyl)piperazin-1-yl)quinazolines

Info

Publication number
KE3155A
KE3155A KE3155A KE315581A KE3155A KE 3155 A KE3155 A KE 3155A KE 3155 A KE3155 A KE 3155A KE 315581 A KE315581 A KE 315581A KE 3155 A KE3155 A KE 3155A
Authority
KE
Kenya
Prior art keywords
heterocyclocarbonyl
quinazolines
piperazin
dimethoxy
amino
Prior art date
Application number
KE3155A
Inventor
R A Partyka
R R Crenshaw
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/658,961 external-priority patent/US4001237A/en
Priority claimed from US05/658,979 external-priority patent/US4001238A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of KE3155A publication Critical patent/KE3155A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
KE3155A 1976-02-18 1981-08-25 4-amino-6,7-dimethoxy-2(4-(heterocyclocarbonyl)piperazin-1-yl)quinazolines KE3155A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/658,961 US4001237A (en) 1976-02-18 1976-02-18 Oxazole, isoxazole, thiazole and isothiazole amides
US05/658,979 US4001238A (en) 1976-02-18 1976-02-18 1,3,4-oxadiazole amides

Publications (1)

Publication Number Publication Date
KE3155A true KE3155A (en) 1981-09-18

Family

ID=27097727

Family Applications (1)

Application Number Title Priority Date Filing Date
KE3155A KE3155A (en) 1976-02-18 1981-08-25 4-amino-6,7-dimethoxy-2(4-(heterocyclocarbonyl)piperazin-1-yl)quinazolines

Country Status (16)

Country Link
JP (1) JPS584716B2 (en)
CA (1) CA1081228A (en)
CH (1) CH635838A5 (en)
CY (1) CY1122A (en)
DE (1) DE2707067A1 (en)
DK (1) DK65177A (en)
FI (1) FI770485A (en)
FR (1) FR2348924A1 (en)
GB (1) GB1533529A (en)
IE (1) IE44614B1 (en)
KE (1) KE3155A (en)
LU (1) LU76802A1 (en)
MY (1) MY8200110A (en)
NL (1) NL7701753A (en)
SE (1) SE7701732L (en)
YU (4) YU45477A (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5791987A (en) * 1980-11-26 1982-06-08 Sankyo Co Ltd Aminoquinazoline derivative and its preparation
US5932538A (en) * 1996-02-02 1999-08-03 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
US5994294A (en) * 1996-02-02 1999-11-30 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
AU2003246571B2 (en) * 2002-06-29 2008-06-26 Zentaris Gmbh Arylcarbonylpiperazines and heteroarylcarbonylpiperazines and the use thereof for treating benign and malignant tumour diseases

Also Published As

Publication number Publication date
CY1122A (en) 1981-12-04
IE44614B1 (en) 1982-01-27
SE7701732L (en) 1977-08-19
YU45477A (en) 1982-10-31
JPS584716B2 (en) 1983-01-27
YU267780A (en) 1983-06-30
YU161182A (en) 1982-10-31
CA1081228A (en) 1980-07-08
NL7701753A (en) 1977-08-22
AU2242677A (en) 1978-07-06
GB1533529A (en) 1978-11-29
FI770485A (en) 1977-08-19
DK65177A (en) 1977-08-19
DE2707067A1 (en) 1977-08-25
LU76802A1 (en) 1977-09-12
IE44614L (en) 1977-08-18
YU161282A (en) 1982-10-31
JPS52102286A (en) 1977-08-27
FR2348924A1 (en) 1977-11-18
MY8200110A (en) 1982-12-31
FR2348924B1 (en) 1980-05-09
CH635838A5 (en) 1983-04-29

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