CH635838A5 - Process for preparing nitrogen-containing heterocyclic carbonylpiperazinylquinazolines - Google Patents

Process for preparing nitrogen-containing heterocyclic carbonylpiperazinylquinazolines Download PDF

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Publication number
CH635838A5
CH635838A5 CH199477A CH199477A CH635838A5 CH 635838 A5 CH635838 A5 CH 635838A5 CH 199477 A CH199477 A CH 199477A CH 199477 A CH199477 A CH 199477A CH 635838 A5 CH635838 A5 CH 635838A5
Authority
CH
Switzerland
Prior art keywords
amino
dimethoxy
prazosin
carbonyl
quinazoline
Prior art date
Application number
CH199477A
Other languages
German (de)
English (en)
Inventor
Richard Anthony Partyka
Ronnie Ray Crenshaw
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/658,961 external-priority patent/US4001237A/en
Priority claimed from US05/658,979 external-priority patent/US4001238A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of CH635838A5 publication Critical patent/CH635838A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH199477A 1976-02-18 1977-02-17 Process for preparing nitrogen-containing heterocyclic carbonylpiperazinylquinazolines CH635838A5 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/658,961 US4001237A (en) 1976-02-18 1976-02-18 Oxazole, isoxazole, thiazole and isothiazole amides
US05/658,979 US4001238A (en) 1976-02-18 1976-02-18 1,3,4-oxadiazole amides

Publications (1)

Publication Number Publication Date
CH635838A5 true CH635838A5 (en) 1983-04-29

Family

ID=27097727

Family Applications (1)

Application Number Title Priority Date Filing Date
CH199477A CH635838A5 (en) 1976-02-18 1977-02-17 Process for preparing nitrogen-containing heterocyclic carbonylpiperazinylquinazolines

Country Status (16)

Country Link
JP (1) JPS584716B2 (fi)
CA (1) CA1081228A (fi)
CH (1) CH635838A5 (fi)
CY (1) CY1122A (fi)
DE (1) DE2707067A1 (fi)
DK (1) DK65177A (fi)
FI (1) FI770485A (fi)
FR (1) FR2348924A1 (fi)
GB (1) GB1533529A (fi)
IE (1) IE44614B1 (fi)
KE (1) KE3155A (fi)
LU (1) LU76802A1 (fi)
MY (1) MY8200110A (fi)
NL (1) NL7701753A (fi)
SE (1) SE7701732L (fi)
YU (4) YU45477A (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5791987A (en) * 1980-11-26 1982-06-08 Sankyo Co Ltd Aminoquinazoline derivative and its preparation
US5994294A (en) * 1996-02-02 1999-11-30 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
US5932538A (en) * 1996-02-02 1999-08-03 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
MXPA04012959A (es) * 2002-06-29 2005-05-16 Zentaris Gmbh Arilcarbonilpiperacinas y heteroarilcarbonilpiperacinas y su uso para tratamiento de enfermedades de tumor benigno y maligno.

Also Published As

Publication number Publication date
DE2707067A1 (de) 1977-08-25
JPS584716B2 (ja) 1983-01-27
AU2242677A (en) 1978-07-06
CY1122A (en) 1981-12-04
SE7701732L (sv) 1977-08-19
FI770485A (fi) 1977-08-19
DK65177A (da) 1977-08-19
FR2348924B1 (fi) 1980-05-09
YU267780A (en) 1983-06-30
CA1081228A (en) 1980-07-08
IE44614B1 (en) 1982-01-27
FR2348924A1 (fr) 1977-11-18
YU161182A (en) 1982-10-31
NL7701753A (nl) 1977-08-22
LU76802A1 (fi) 1977-09-12
MY8200110A (en) 1982-12-31
GB1533529A (en) 1978-11-29
KE3155A (en) 1981-09-18
YU161282A (en) 1982-10-31
IE44614L (en) 1977-08-18
YU45477A (en) 1982-10-31
JPS52102286A (en) 1977-08-27

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PL Patent ceased