FR2348924A1 - Nouvelles carbonylpiperazinylquinazolines azoliques,leur procede de preparation et medicament les contenant - Google Patents

Nouvelles carbonylpiperazinylquinazolines azoliques,leur procede de preparation et medicament les contenant

Info

Publication number
FR2348924A1
FR2348924A1 FR7704560A FR7704560A FR2348924A1 FR 2348924 A1 FR2348924 A1 FR 2348924A1 FR 7704560 A FR7704560 A FR 7704560A FR 7704560 A FR7704560 A FR 7704560A FR 2348924 A1 FR2348924 A1 FR 2348924A1
Authority
FR
France
Prior art keywords
carbonylpiperazinylquinazolines
azolic
new
preparation process
product containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7704560A
Other languages
English (en)
French (fr)
Other versions
FR2348924B1 (fi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Co
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/658,961 external-priority patent/US4001237A/en
Priority claimed from US05/658,979 external-priority patent/US4001238A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of FR2348924A1 publication Critical patent/FR2348924A1/fr
Application granted granted Critical
Publication of FR2348924B1 publication Critical patent/FR2348924B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR7704560A 1976-02-18 1977-02-17 Nouvelles carbonylpiperazinylquinazolines azoliques,leur procede de preparation et medicament les contenant Granted FR2348924A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/658,961 US4001237A (en) 1976-02-18 1976-02-18 Oxazole, isoxazole, thiazole and isothiazole amides
US05/658,979 US4001238A (en) 1976-02-18 1976-02-18 1,3,4-oxadiazole amides

Publications (2)

Publication Number Publication Date
FR2348924A1 true FR2348924A1 (fr) 1977-11-18
FR2348924B1 FR2348924B1 (fi) 1980-05-09

Family

ID=27097727

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7704560A Granted FR2348924A1 (fr) 1976-02-18 1977-02-17 Nouvelles carbonylpiperazinylquinazolines azoliques,leur procede de preparation et medicament les contenant

Country Status (16)

Country Link
JP (1) JPS584716B2 (fi)
CA (1) CA1081228A (fi)
CH (1) CH635838A5 (fi)
CY (1) CY1122A (fi)
DE (1) DE2707067A1 (fi)
DK (1) DK65177A (fi)
FI (1) FI770485A (fi)
FR (1) FR2348924A1 (fi)
GB (1) GB1533529A (fi)
IE (1) IE44614B1 (fi)
KE (1) KE3155A (fi)
LU (1) LU76802A1 (fi)
MY (1) MY8200110A (fi)
NL (1) NL7701753A (fi)
SE (1) SE7701732L (fi)
YU (4) YU45477A (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5791987A (en) * 1980-11-26 1982-06-08 Sankyo Co Ltd Aminoquinazoline derivative and its preparation
US5994294A (en) * 1996-02-02 1999-11-30 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
US5932538A (en) * 1996-02-02 1999-08-03 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
MXPA04012959A (es) * 2002-06-29 2005-05-16 Zentaris Gmbh Arilcarbonilpiperacinas y heteroarilcarbonilpiperacinas y su uso para tratamiento de enfermedades de tumor benigno y maligno.

Also Published As

Publication number Publication date
DE2707067A1 (de) 1977-08-25
JPS584716B2 (ja) 1983-01-27
AU2242677A (en) 1978-07-06
CY1122A (en) 1981-12-04
SE7701732L (sv) 1977-08-19
CH635838A5 (en) 1983-04-29
FI770485A (fi) 1977-08-19
DK65177A (da) 1977-08-19
FR2348924B1 (fi) 1980-05-09
YU267780A (en) 1983-06-30
CA1081228A (en) 1980-07-08
IE44614B1 (en) 1982-01-27
YU161182A (en) 1982-10-31
NL7701753A (nl) 1977-08-22
LU76802A1 (fi) 1977-09-12
MY8200110A (en) 1982-12-31
GB1533529A (en) 1978-11-29
KE3155A (en) 1981-09-18
YU161282A (en) 1982-10-31
IE44614L (en) 1977-08-18
YU45477A (en) 1982-10-31
JPS52102286A (en) 1977-08-27

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Legal Events

Date Code Title Description
ST Notification of lapse