CH625524A5 - - Google Patents

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Publication number
CH625524A5
CH625524A5 CH717376A CH717376A CH625524A5 CH 625524 A5 CH625524 A5 CH 625524A5 CH 717376 A CH717376 A CH 717376A CH 717376 A CH717376 A CH 717376A CH 625524 A5 CH625524 A5 CH 625524A5
Authority
CH
Switzerland
Prior art keywords
less
atoms
group
alkyl
ring
Prior art date
Application number
CH717376A
Other languages
English (en)
Italian (it)
Inventor
Leonardo Marsili
Vittorio Rossetti
Carmine Pasqualucci
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of CH625524A5 publication Critical patent/CH625524A5/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH717376A 1975-06-13 1976-06-08 CH625524A5 (enExample)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT755174A IT1056272B (it) 1975-06-13 1975-06-13 Prodotti derivati dalle amine aromatiche

Publications (1)

Publication Number Publication Date
CH625524A5 true CH625524A5 (enExample) 1981-09-30

Family

ID=11118842

Family Applications (1)

Application Number Title Priority Date Filing Date
CH717376A CH625524A5 (enExample) 1975-06-13 1976-06-08

Country Status (28)

Country Link
US (2) US4086225A (enExample)
JP (1) JPS5236683A (enExample)
AR (1) AR211127A1 (enExample)
AU (1) AU497602B2 (enExample)
BE (1) BE842883A (enExample)
CA (1) CA1059123A (enExample)
CH (1) CH625524A5 (enExample)
CS (1) CS197271B1 (enExample)
DK (1) DK145228C (enExample)
ES (1) ES449187A1 (enExample)
FI (1) FI60208C (enExample)
FR (1) FR2314189A1 (enExample)
GB (1) GB1542063A (enExample)
HK (1) HK56083A (enExample)
HU (1) HU171396B (enExample)
IE (1) IE42998B1 (enExample)
IL (1) IL49701A (enExample)
IN (1) IN143526B (enExample)
IT (1) IT1056272B (enExample)
NL (1) NL177919C (enExample)
NO (1) NO148848C (enExample)
PH (1) PH16410A (enExample)
PL (1) PL99493B1 (enExample)
PT (1) PT65208B (enExample)
SE (1) SE434057B (enExample)
SU (1) SU680649A3 (enExample)
YU (1) YU39768B (enExample)
ZA (1) ZA763256B (enExample)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1056272B (it) * 1975-06-13 1982-01-30 Archifar Ind Chim Trentino Prodotti derivati dalle amine aromatiche
DK345977A (da) * 1976-09-30 1978-03-31 Archifar Ind Chim Trentino G rifamycinforbindelser og fremgangsmaade til deres fremstillin
BE886395A (fr) * 1980-02-13 1981-03-16 Erba Farmitalia Derives de rifamycine
IT1201963B (it) * 1983-03-24 1989-02-02 Prodotti Antibiotici Spa Derivati delle rifamicine e procedimento per la loro preparazione
US4631290A (en) * 1985-08-29 1986-12-23 American Home Products Corporation Method of treating hepatitis
ES2095772T3 (es) * 1993-05-05 1997-02-16 Palo Alto Medical Found Utilizacion de derivados de rifamicina para producir un medicamento destinado al tratamiento de la toxoplasmosis.
US5529994A (en) * 1993-05-05 1996-06-25 Palo Alto Medical Foundation Treatment for toxoplasmosis
US5981522A (en) * 1995-09-01 1999-11-09 Kaneka Corporation Treatment of disease caused by infection of Helicobacter
CA2204007A1 (en) * 1995-09-01 1997-03-13 Katsuji Yamashita Remedy for diseases caused by infection with helicobacter
US7122525B2 (en) * 2001-11-21 2006-10-17 Activbiotics, Inc. Targeted therapeutics and uses thereof
US7078399B2 (en) * 2001-12-13 2006-07-18 Activbiotics, Inc. Sulfhydryl rifamycins and uses thereof
US7820652B2 (en) * 2003-09-24 2010-10-26 Activbiotics Pharma, Llc Regimen for the administration of rifamycin-class antibiotics
US7202246B2 (en) * 2004-06-09 2007-04-10 Cumbre Pharmaceuticals Inc. Spiro-rifamycin derivatives targeting RNA polymerase
ES2246155B1 (es) * 2004-07-19 2007-03-16 Universidad De Oviedo Nuevas espiropiperidilrifamicinas.
US8404664B2 (en) 2005-08-11 2013-03-26 Targanta Therapeutics, Inc. Phosphonated Rifamycins and uses thereof for the prevention and treatment of bone and joint infections
US7678791B2 (en) * 2006-07-12 2010-03-16 Cumbre Ip Ventures, L.P. Nitroheteroaryl-containing rifamycin derivatives
CN100569778C (zh) * 2006-12-05 2009-12-16 四川明欣药业有限责任公司 一种利福布汀结晶工艺
WO2009064792A1 (en) * 2007-11-16 2009-05-22 Cumbre Pharmaceuticals Inc. Quinolone carboxylic acid-substituted rifamycin derivatives
US8524691B2 (en) 2008-08-13 2013-09-03 The Medicines Company Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections
EP3560497A1 (en) 2012-08-30 2019-10-30 The Texas A&M University System Compositions and methods for drug-sensitization or inhibition of a cancer cell
PH12013000351A1 (en) 2013-11-22 2015-05-25 Joselle A Macrohon A versatile queuing management system and method
WO2016014437A1 (en) 2014-07-21 2016-01-28 Hiroaki Serizawa Ophthalmic compositions of rifamycins and uses thereof
CN106279205B (zh) * 2015-05-12 2020-07-21 重庆华邦胜凯制药有限公司 制备利福霉素s衍生物的方法
WO2026115045A1 (en) * 2024-11-27 2026-06-04 Galapagos Nv Novel compounds and pharmaceutical compositions thereof for the treatment of infectious diseases

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL130099C (enExample) * 1963-10-11
IT1056272B (it) * 1975-06-13 1982-01-30 Archifar Ind Chim Trentino Prodotti derivati dalle amine aromatiche
DE2626296C2 (de) * 1975-06-13 1986-11-27 Farmitalia Carlo Erba S.p.A., Mailand/Milano Rifamycin-Verbindung und Verfahren zu seiner Herstellung

Also Published As

Publication number Publication date
SU680649A3 (ru) 1979-08-15
NL177919B (nl) 1985-07-16
YU140576A (en) 1982-06-30
CA1059123A (en) 1979-07-24
NO762026L (enExample) 1976-12-14
PL99493B1 (pl) 1978-07-31
IN143526B (enExample) 1977-12-17
GB1542063A (en) 1979-03-14
YU39768B (en) 1985-04-30
IE42998B1 (en) 1980-12-03
DK145228C (da) 1983-02-28
JPS6121957B2 (enExample) 1986-05-29
IT1056272B (it) 1982-01-30
HK56083A (en) 1983-11-25
CS197271B1 (en) 1980-04-30
AU1476976A (en) 1977-12-15
FI761688A7 (enExample) 1976-12-14
JPS5236683A (en) 1977-03-22
ES449187A1 (es) 1977-07-16
IE42998L (en) 1976-12-13
FI60208C (fi) 1981-12-10
HU171396B (hu) 1978-01-28
FR2314189A1 (fr) 1977-01-07
IL49701A (en) 1979-10-31
FR2314189B1 (enExample) 1980-10-31
US4219478A (en) 1980-08-26
AR211127A1 (es) 1977-10-31
NO148848C (no) 1983-12-28
DK258076A (da) 1976-12-14
NO148848B (no) 1983-09-19
ZA763256B (en) 1977-05-25
IL49701A0 (en) 1976-08-31
NL7606370A (nl) 1976-12-15
SE434057B (sv) 1984-07-02
FI60208B (fi) 1981-08-31
US4086225A (en) 1978-04-25
DK145228B (da) 1982-10-11
PT65208A (en) 1976-07-01
PH16410A (en) 1983-09-29
BE842883A (fr) 1976-10-01
AU497602B2 (en) 1978-12-21
NL177919C (nl) 1985-12-16
PT65208B (en) 1977-11-23
SE7606640L (sv) 1976-12-14

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Legal Events

Date Code Title Description
PFA Name/firm changed

Owner name: FARMITALIA CARLO ERBA S.R.L.

PL Patent ceased