CH535254A - Procédé de préparation de nouveaux dérivés de l'imidazoline - Google Patents
Procédé de préparation de nouveaux dérivés de l'imidazolineInfo
- Publication number
- CH535254A CH535254A CH17272A CH17272A CH535254A CH 535254 A CH535254 A CH 535254A CH 17272 A CH17272 A CH 17272A CH 17272 A CH17272 A CH 17272A CH 535254 A CH535254 A CH 535254A
- Authority
- CH
- Switzerland
- Prior art keywords
- preparation
- imidazoline derivatives
- novel imidazoline
- novel
- derivatives
- Prior art date
Links
- 150000002462 imidazolines Chemical class 0.000 title 1
- 229940083254 peripheral vasodilators imidazoline derivative Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB332771 | 1971-01-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH535254A true CH535254A (fr) | 1973-03-31 |
Family
ID=9756227
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH17272A CH535254A (fr) | 1971-01-27 | 1972-01-06 | Procédé de préparation de nouveaux dérivés de l'imidazoline |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US3818035A (h) |
| JP (1) | JPS4938273B1 (h) |
| AT (1) | AT311336B (h) |
| BE (1) | BE777689A (h) |
| CA (1) | CA962273A (h) |
| CH (1) | CH535254A (h) |
| DE (1) | DE2203373C3 (h) |
| DK (1) | DK138496B (h) |
| FI (1) | FI55841C (h) |
| GB (1) | GB1333471A (h) |
| HU (1) | HU162823B (h) |
| NL (1) | NL150454B (h) |
| NO (1) | NO134115C (h) |
| SE (1) | SE378426B (h) |
| SU (1) | SU474145A3 (h) |
| YU (1) | YU34694B (h) |
| ZA (1) | ZA72286B (h) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3927023A (en) * | 1974-05-24 | 1975-12-16 | Warner Lambert Co | Imidazolyl benzofurans |
| DE3049542A1 (de) * | 1980-12-31 | 1982-07-29 | Basf Ag, 6700 Ludwigshafen | Azolylalkyl-2,3-dihydrobenzofurane, diese enthaltende fungizide und verfahren zu ihrer herstellung |
| ZA825413B (en) * | 1981-08-26 | 1983-06-29 | Pfizer | Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them |
| US4851554A (en) * | 1987-04-06 | 1989-07-25 | University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
| US4806663A (en) * | 1987-04-06 | 1989-02-21 | The University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
| US4831156A (en) * | 1987-09-30 | 1989-05-16 | The University Of Tennessee Research Corp. | 3-substituted 2-alkyl indole derivatives |
| AU2003099A (en) * | 1997-12-19 | 1999-07-12 | Eli Lilly And Company | Method for treating diabetes |
| US7777035B2 (en) * | 2005-06-22 | 2010-08-17 | Chemocentryx, Inc. | Azaindazole compounds and methods of use |
| CA2637312A1 (en) * | 2006-01-27 | 2007-08-02 | F. Hoffmann-La Roche Ag | Use of substituted 2-imidazole of imidazoline derivatives |
| KR101176699B1 (ko) * | 2006-10-19 | 2012-08-23 | 에프. 호프만-라 로슈 아게 | 아미노메틸-4-이미다졸 |
| DE602007005671D1 (de) * | 2006-10-19 | 2010-05-12 | Hoffmann La Roche | Aminomethyl-2-imidazole mit affinität zu mit dem trace-amin assoziierten rezeptoren |
| ES2375578T3 (es) * | 2006-11-02 | 2012-03-02 | F. Hoffmann-La Roche Ag | 2-imidazoles sustituidos como moduladores de receptores asociados a aminas trazas. |
| EP2084152A2 (en) * | 2006-11-16 | 2009-08-05 | F. Hoffmann-Roche AG | Substituted 4-imidazoles |
| ATE509628T1 (de) * | 2006-12-13 | 2011-06-15 | Hoffmann La Roche | Neue 2-imidazole als liganden für trace amine associated receptors (taar) |
| US20080146523A1 (en) | 2006-12-18 | 2008-06-19 | Guido Galley | Imidazole derivatives |
| MX2009008255A (es) * | 2007-02-02 | 2009-08-12 | Hoffmann La Roche | Nuevas 2-aminooxazolinas como ligandos taar1. |
| JP5130305B2 (ja) * | 2007-02-15 | 2013-01-30 | エフ.ホフマン−ラ ロシュ アーゲー | Taar1リガンドとしての2−アミノオキサゾリン |
| KR101150561B1 (ko) | 2007-07-02 | 2012-06-08 | 에프. 호프만-라 로슈 아게 | 미량 아민 결합 수용체(taar)에 대한 양호한 친화도를 갖는 2-이미다졸린 |
| JP2010531836A (ja) * | 2007-07-03 | 2010-09-30 | エフ.ホフマン−ラ ロシュ アーゲー | 4−イミダゾリン及びそれらの抗うつ剤としての使用 |
| RU2010104632A (ru) * | 2007-07-27 | 2011-09-20 | Ф.Хоффманн-Ля Рош Аг (Ch) | 2-азетидинметанамины и 2-пирролидинметанамины в качестве лигандов taar |
| CN101765425A (zh) * | 2007-08-02 | 2010-06-30 | 弗·哈夫曼-拉罗切有限公司 | 苯甲酰胺衍生物用于治疗cns障碍的用途 |
| JP5341084B2 (ja) * | 2007-08-03 | 2013-11-13 | エフ.ホフマン−ラ ロシュ アーゲー | Taar1リガンドとしてのピリジンカルボキシアミド及びベンズアミド誘導体 |
| RU2513086C2 (ru) * | 2008-07-24 | 2014-04-20 | Ф.Хоффманн-Ля Рош Аг | Производные 4,5-дигидро-оксазол-2-ила |
| US8242153B2 (en) * | 2008-07-24 | 2012-08-14 | Hoffmann-La Roche Inc. | 4,5-dihydro-oxazol-2YL derivatives |
| US20100311798A1 (en) * | 2009-06-05 | 2010-12-09 | Decoret Guillaume | 2-aminooxazolines as taar1 ligands |
| US8354441B2 (en) * | 2009-11-11 | 2013-01-15 | Hoffmann-La Roche Inc. | Oxazoline derivatives |
| US9452980B2 (en) | 2009-12-22 | 2016-09-27 | Hoffmann-La Roche Inc. | Substituted benzamides |
| SI3430010T1 (sl) | 2016-03-17 | 2020-10-30 | F. Hoffmann-La Roche Ag | Derivat 5-etil-4-metil-pirazol-3-karboksamida z aktivnostjo agonista TAAR |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1121054B (de) * | 1960-11-23 | 1962-01-04 | Merck Ag E | Verfahren zur Herstellung eines neuen Imidazolinderivates und dessen Saeureadditionssalzen |
-
1971
- 1971-01-27 GB GB332771A patent/GB1333471A/en not_active Expired
-
1972
- 1972-01-05 BE BE777689A patent/BE777689A/xx not_active IP Right Cessation
- 1972-01-06 CH CH17272A patent/CH535254A/fr not_active IP Right Cessation
- 1972-01-10 US US00216795A patent/US3818035A/en not_active Expired - Lifetime
- 1972-01-17 ZA ZA720286A patent/ZA72286B/xx unknown
- 1972-01-25 DE DE2203373A patent/DE2203373C3/de not_active Expired
- 1972-01-26 SE SE7200867A patent/SE378426B/xx unknown
- 1972-01-26 NO NO192/72A patent/NO134115C/no unknown
- 1972-01-26 YU YU181/72A patent/YU34694B/xx unknown
- 1972-01-26 HU HULA791A patent/HU162823B/hu not_active IP Right Cessation
- 1972-01-26 DK DK34572AA patent/DK138496B/da unknown
- 1972-01-27 CA CA133,337A patent/CA962273A/en not_active Expired
- 1972-01-27 JP JP47010207A patent/JPS4938273B1/ja active Pending
- 1972-01-27 NL NL727201121A patent/NL150454B/xx not_active IP Right Cessation
- 1972-01-27 SU SU1742351A patent/SU474145A3/ru active
- 1972-01-27 AT AT64772A patent/AT311336B/de not_active IP Right Cessation
- 1972-01-27 FI FI219/72A patent/FI55841C/fi active
Also Published As
| Publication number | Publication date |
|---|---|
| JPS4938273B1 (h) | 1974-10-16 |
| HU162823B (h) | 1973-04-28 |
| DE2203373C3 (de) | 1978-04-13 |
| NO134115C (h) | 1976-08-18 |
| NO134115B (h) | 1976-05-10 |
| AT311336B (de) | 1973-11-12 |
| ZA72286B (en) | 1972-09-27 |
| DE2203373A1 (de) | 1972-08-17 |
| US3818035A (en) | 1974-06-18 |
| CA962273A (en) | 1975-02-04 |
| NL7201121A (h) | 1972-07-31 |
| YU18172A (en) | 1979-07-10 |
| DE2203373B2 (de) | 1977-08-11 |
| BE777689A (fr) | 1972-07-05 |
| GB1333471A (en) | 1973-10-10 |
| DK138496C (h) | 1979-02-26 |
| SE378426B (h) | 1975-09-01 |
| SU474145A3 (ru) | 1975-06-14 |
| FI55841B (fi) | 1979-06-29 |
| NL150454B (nl) | 1976-08-16 |
| AU3817772A (en) | 1973-07-26 |
| YU34694B (en) | 1979-12-31 |
| DK138496B (da) | 1978-09-18 |
| FI55841C (fi) | 1979-10-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PFA | Name/firm changed |
Owner name: SANOFI |
|
| PUE | Assignment |
Owner name: OMNIUM FINANCIER AQUITAINE POUR L HYGIENE ET LA SA |
|
| PL | Patent ceased |