DK138496B - Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf.

Info

Publication number
DK138496B
DK138496B DK34572AA DK34572A DK138496B DK 138496 B DK138496 B DK 138496B DK 34572A A DK34572A A DK 34572AA DK 34572 A DK34572 A DK 34572A DK 138496 B DK138496 B DK 138496B
Authority
DK
Denmark
Prior art keywords
preparation
acid addition
addition salts
imidazoline derivatives
analogous process
Prior art date
Application number
DK34572AA
Other languages
English (en)
Other versions
DK138496C (da
Inventor
Fernand Binon
Alex Areschka
Original Assignee
Labaz
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Labaz filed Critical Labaz
Publication of DK138496B publication Critical patent/DK138496B/da
Application granted granted Critical
Publication of DK138496C publication Critical patent/DK138496C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK34572AA 1971-01-27 1972-01-26 Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. DK138496B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB332771 1971-01-27

Publications (2)

Publication Number Publication Date
DK138496B true DK138496B (da) 1978-09-18
DK138496C DK138496C (da) 1979-02-26

Family

ID=9756227

Family Applications (1)

Application Number Title Priority Date Filing Date
DK34572AA DK138496B (da) 1971-01-27 1972-01-26 Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf.

Country Status (17)

Country Link
US (1) US3818035A (da)
JP (1) JPS4938273B1 (da)
AT (1) AT311336B (da)
BE (1) BE777689A (da)
CA (1) CA962273A (da)
CH (1) CH535254A (da)
DE (1) DE2203373C3 (da)
DK (1) DK138496B (da)
FI (1) FI55841C (da)
GB (1) GB1333471A (da)
HU (1) HU162823B (da)
NL (1) NL150454B (da)
NO (1) NO134115C (da)
SE (1) SE378426B (da)
SU (1) SU474145A3 (da)
YU (1) YU34694B (da)
ZA (1) ZA72286B (da)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3927023A (en) * 1974-05-24 1975-12-16 Warner Lambert Co Imidazolyl benzofurans
DE3049542A1 (de) * 1980-12-31 1982-07-29 Basf Ag, 6700 Ludwigshafen Azolylalkyl-2,3-dihydrobenzofurane, diese enthaltende fungizide und verfahren zu ihrer herstellung
ZA825413B (en) * 1981-08-26 1983-06-29 Pfizer Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them
US4806663A (en) * 1987-04-06 1989-02-21 The University Of Tennessee Research Corporation Certain 3-substituted 2-alkyl benzofuran derivatives
US4851554A (en) * 1987-04-06 1989-07-25 University Of Tennessee Research Corporation Certain 3-substituted 2-alkyl benzofuran derivatives
US4831156A (en) * 1987-09-30 1989-05-16 The University Of Tennessee Research Corp. 3-substituted 2-alkyl indole derivatives
WO1999032482A1 (en) * 1997-12-19 1999-07-01 Eli Lilly And Company Hypoglycemic imidazoline compounds
US7777035B2 (en) * 2005-06-22 2010-08-17 Chemocentryx, Inc. Azaindazole compounds and methods of use
CA2637312A1 (en) * 2006-01-27 2007-08-02 F. Hoffmann-La Roche Ag Use of substituted 2-imidazole of imidazoline derivatives
CA2666762C (en) * 2006-10-19 2014-12-30 F. Hoffmann-La Roche Ag Aminomethyl-4-imidazoles
WO2008046756A1 (en) * 2006-10-19 2008-04-24 F. Hoffmann-La Roche Ag Aminomethyl-2-imidazoles with affinity with the trace amine associated receptors
EP2086959B1 (en) * 2006-11-02 2011-11-16 F. Hoffmann-La Roche AG Substituted 2-imidazoles as modulators of the trace amine associated receptors
MX2009005047A (es) * 2006-11-16 2009-05-25 Hoffmann La Roche 4-imidazoles sustituidos.
MX2009005920A (es) * 2006-12-13 2009-06-16 Hoffmann La Roche Nuevos 2-imidazoles como ligandos para receptores asociados con trazas de amina.
US20080146523A1 (en) 2006-12-18 2008-06-19 Guido Galley Imidazole derivatives
MX2009008255A (es) * 2007-02-02 2009-08-12 Hoffmann La Roche Nuevas 2-aminooxazolinas como ligandos taar1.
KR101222412B1 (ko) * 2007-02-15 2013-01-15 에프. 호프만-라 로슈 아게 Taar1 리간드로서의 2-아미노옥사졸린
CN101687812A (zh) 2007-07-02 2010-03-31 弗·哈夫曼-拉罗切有限公司 对痕量胺相关受体(taar)具有良好亲和性的2-咪唑啉化合物
WO2009003867A1 (en) * 2007-07-03 2009-01-08 F. Hoffmann-La Roche Ag 4-imidazolines and their use as antidepressants
WO2009016048A1 (en) * 2007-07-27 2009-02-05 F. Hoffmann-La Roche Ag 2-azetidinemethaneamines and 2-pyrrolidinemethaneamines as taar-ligands
CN101765425A (zh) * 2007-08-02 2010-06-30 弗·哈夫曼-拉罗切有限公司 苯甲酰胺衍生物用于治疗cns障碍的用途
BRPI0814758A2 (pt) * 2007-08-03 2015-03-03 Hoffmann La Roche Piridinacarboxamida e derivados de benzamida como ligantes taar1
CN102083805A (zh) * 2008-07-24 2011-06-01 弗·哈夫曼-拉罗切有限公司 4,5-二氢-唑-2-基衍生物
US8242153B2 (en) * 2008-07-24 2012-08-14 Hoffmann-La Roche Inc. 4,5-dihydro-oxazol-2YL derivatives
US20100311798A1 (en) * 2009-06-05 2010-12-09 Decoret Guillaume 2-aminooxazolines as taar1 ligands
US8354441B2 (en) * 2009-11-11 2013-01-15 Hoffmann-La Roche Inc. Oxazoline derivatives
US9452980B2 (en) 2009-12-22 2016-09-27 Hoffmann-La Roche Inc. Substituted benzamides
JP6814814B2 (ja) 2016-03-17 2021-01-20 エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft Taarのアゴニストとしての活性を有する5−エチル−4−メチル−ピラゾール−3−カルボキサミド誘導体

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1121054B (de) * 1960-11-23 1962-01-04 Merck Ag E Verfahren zur Herstellung eines neuen Imidazolinderivates und dessen Saeureadditionssalzen

Also Published As

Publication number Publication date
BE777689A (fr) 1972-07-05
ZA72286B (en) 1972-09-27
JPS4938273B1 (da) 1974-10-16
AU3817772A (en) 1973-07-26
YU34694B (en) 1979-12-31
SE378426B (da) 1975-09-01
YU18172A (en) 1979-07-10
AT311336B (de) 1973-11-12
NL7201121A (da) 1972-07-31
SU474145A3 (ru) 1975-06-14
NO134115B (da) 1976-05-10
DE2203373A1 (de) 1972-08-17
NL150454B (nl) 1976-08-16
NO134115C (da) 1976-08-18
DE2203373C3 (de) 1978-04-13
GB1333471A (en) 1973-10-10
DK138496C (da) 1979-02-26
DE2203373B2 (de) 1977-08-11
US3818035A (en) 1974-06-18
FI55841B (fi) 1979-06-29
HU162823B (da) 1973-04-28
FI55841C (fi) 1979-10-10
CA962273A (en) 1975-02-04
CH535254A (fr) 1973-03-31

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