DK138496B - Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. - Google Patents
Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf.Info
- Publication number
- DK138496B DK138496B DK34572AA DK34572A DK138496B DK 138496 B DK138496 B DK 138496B DK 34572A A DK34572A A DK 34572AA DK 34572 A DK34572 A DK 34572A DK 138496 B DK138496 B DK 138496B
- Authority
- DK
- Denmark
- Prior art keywords
- preparation
- acid addition
- addition salts
- imidazoline derivatives
- analogous process
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000002462 imidazolines Chemical class 0.000 title 1
- 229940083254 peripheral vasodilators imidazoline derivative Drugs 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB332771 | 1971-01-27 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK138496B true DK138496B (da) | 1978-09-18 |
| DK138496C DK138496C (da) | 1979-02-26 |
Family
ID=9756227
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK34572AA DK138496B (da) | 1971-01-27 | 1972-01-26 | Analogifremgangsmåde til fremstilling af imidazolinderivater eller syreadditionssalte deraf. |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US3818035A (da) |
| JP (1) | JPS4938273B1 (da) |
| AT (1) | AT311336B (da) |
| BE (1) | BE777689A (da) |
| CA (1) | CA962273A (da) |
| CH (1) | CH535254A (da) |
| DE (1) | DE2203373C3 (da) |
| DK (1) | DK138496B (da) |
| FI (1) | FI55841C (da) |
| GB (1) | GB1333471A (da) |
| HU (1) | HU162823B (da) |
| NL (1) | NL150454B (da) |
| NO (1) | NO134115C (da) |
| SE (1) | SE378426B (da) |
| SU (1) | SU474145A3 (da) |
| YU (1) | YU34694B (da) |
| ZA (1) | ZA72286B (da) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3927023A (en) * | 1974-05-24 | 1975-12-16 | Warner Lambert Co | Imidazolyl benzofurans |
| DE3049542A1 (de) * | 1980-12-31 | 1982-07-29 | Basf Ag, 6700 Ludwigshafen | Azolylalkyl-2,3-dihydrobenzofurane, diese enthaltende fungizide und verfahren zu ihrer herstellung |
| ZA825413B (en) * | 1981-08-26 | 1983-06-29 | Pfizer | Thromboxane synthetase inhibitors, processes for their production, and pharmaceutical compositions comprising them |
| US4851554A (en) * | 1987-04-06 | 1989-07-25 | University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
| US4806663A (en) * | 1987-04-06 | 1989-02-21 | The University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzofuran derivatives |
| US4831156A (en) * | 1987-09-30 | 1989-05-16 | The University Of Tennessee Research Corp. | 3-substituted 2-alkyl indole derivatives |
| ES2198033T3 (es) * | 1997-12-19 | 2004-01-16 | Eli Lilly And Company | Compuestos de imidazolina hipoglucemicos. |
| US7777035B2 (en) * | 2005-06-22 | 2010-08-17 | Chemocentryx, Inc. | Azaindazole compounds and methods of use |
| KR20080080410A (ko) * | 2006-01-27 | 2008-09-03 | 에프. 호프만-라 로슈 아게 | 이미다졸린 유도체의 치환된 2-이미다졸의 용도 |
| WO2008046757A1 (en) * | 2006-10-19 | 2008-04-24 | F. Hoffmann-La Roche Ag | Aminomethyl-4-imidazoles |
| DE602007005671D1 (de) * | 2006-10-19 | 2010-05-12 | Hoffmann La Roche | Aminomethyl-2-imidazole mit affinität zu mit dem trace-amin assoziierten rezeptoren |
| KR101176700B1 (ko) * | 2006-11-02 | 2012-08-23 | 에프. 호프만-라 로슈 아게 | 미량 아민 결합된 수용체의 조절자로서 치환된 2-이미다졸 |
| JP2010510184A (ja) * | 2006-11-16 | 2010-04-02 | エフ.ホフマン−ラ ロシュ アーゲー | 置換4−イミダゾール類 |
| AU2007332641A1 (en) * | 2006-12-13 | 2008-06-19 | F. Hoffmann-La Roche Ag | Novel 2 -imidazoles as ligands for trace amine associated receptors (TAAR) |
| US20080146523A1 (en) * | 2006-12-18 | 2008-06-19 | Guido Galley | Imidazole derivatives |
| NZ578260A (en) * | 2007-02-02 | 2012-02-24 | Hoffmann La Roche | Novel 2-aminooxazolines as taar1 ligands for cns disorders |
| JP5130305B2 (ja) * | 2007-02-15 | 2013-01-30 | エフ.ホフマン−ラ ロシュ アーゲー | Taar1リガンドとしての2−アミノオキサゾリン |
| EP2173720A2 (en) | 2007-07-02 | 2010-04-14 | F. Hoffmann-Roche AG | 2-imidazolines having a good affinity to the trace amine associated receptors (taars) |
| EP2173719A1 (en) * | 2007-07-03 | 2010-04-14 | F. Hoffmann-Roche AG | 4-imidazolines and their use as antidepressants |
| JP2010534701A (ja) * | 2007-07-27 | 2010-11-11 | エフ.ホフマン−ラ ロシュ アーゲー | Taarリガンドとしての2−アゼチジンメタンアミン及び2−ピロリジンメタンアミン |
| KR20100039429A (ko) * | 2007-08-02 | 2010-04-15 | 에프. 호프만-라 로슈 아게 | Cns 질환의 치료를 위한 벤즈아미드 유도체의 용도 |
| JP5341084B2 (ja) * | 2007-08-03 | 2013-11-13 | エフ.ホフマン−ラ ロシュ アーゲー | Taar1リガンドとしてのピリジンカルボキシアミド及びベンズアミド誘導体 |
| US8242153B2 (en) * | 2008-07-24 | 2012-08-14 | Hoffmann-La Roche Inc. | 4,5-dihydro-oxazol-2YL derivatives |
| AU2009273324A1 (en) * | 2008-07-24 | 2010-01-28 | F. Hoffmann-La Roche Ag | 4,5-dihydro-oxazol-2-yl derivatives |
| US20100311798A1 (en) * | 2009-06-05 | 2010-12-09 | Decoret Guillaume | 2-aminooxazolines as taar1 ligands |
| US8354441B2 (en) * | 2009-11-11 | 2013-01-15 | Hoffmann-La Roche Inc. | Oxazoline derivatives |
| US9452980B2 (en) | 2009-12-22 | 2016-09-27 | Hoffmann-La Roche Inc. | Substituted benzamides |
| JP6814814B2 (ja) | 2016-03-17 | 2021-01-20 | エフ.ホフマン−ラ ロシュ アーゲーF. Hoffmann−La Roche Aktiengesellschaft | Taarのアゴニストとしての活性を有する5−エチル−4−メチル−ピラゾール−3−カルボキサミド誘導体 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1121054B (de) * | 1960-11-23 | 1962-01-04 | Merck Ag E | Verfahren zur Herstellung eines neuen Imidazolinderivates und dessen Saeureadditionssalzen |
-
1971
- 1971-01-27 GB GB332771A patent/GB1333471A/en not_active Expired
-
1972
- 1972-01-05 BE BE777689A patent/BE777689A/xx not_active IP Right Cessation
- 1972-01-06 CH CH17272A patent/CH535254A/fr not_active IP Right Cessation
- 1972-01-10 US US00216795A patent/US3818035A/en not_active Expired - Lifetime
- 1972-01-17 ZA ZA720286A patent/ZA72286B/xx unknown
- 1972-01-25 DE DE2203373A patent/DE2203373C3/de not_active Expired
- 1972-01-26 HU HULA791A patent/HU162823B/hu not_active IP Right Cessation
- 1972-01-26 YU YU181/72A patent/YU34694B/xx unknown
- 1972-01-26 DK DK34572AA patent/DK138496B/da unknown
- 1972-01-26 NO NO192/72A patent/NO134115C/no unknown
- 1972-01-26 SE SE7200867A patent/SE378426B/xx unknown
- 1972-01-27 JP JP47010207A patent/JPS4938273B1/ja active Pending
- 1972-01-27 FI FI219/72A patent/FI55841C/fi active
- 1972-01-27 CA CA133,337A patent/CA962273A/en not_active Expired
- 1972-01-27 SU SU1742351A patent/SU474145A3/ru active
- 1972-01-27 AT AT64772A patent/AT311336B/de not_active IP Right Cessation
- 1972-01-27 NL NL727201121A patent/NL150454B/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| NO134115B (da) | 1976-05-10 |
| FI55841C (fi) | 1979-10-10 |
| FI55841B (fi) | 1979-06-29 |
| SU474145A3 (ru) | 1975-06-14 |
| YU34694B (en) | 1979-12-31 |
| BE777689A (fr) | 1972-07-05 |
| AT311336B (de) | 1973-11-12 |
| CA962273A (en) | 1975-02-04 |
| ZA72286B (en) | 1972-09-27 |
| HU162823B (da) | 1973-04-28 |
| DE2203373C3 (de) | 1978-04-13 |
| DE2203373B2 (de) | 1977-08-11 |
| NO134115C (da) | 1976-08-18 |
| YU18172A (en) | 1979-07-10 |
| SE378426B (da) | 1975-09-01 |
| NL150454B (nl) | 1976-08-16 |
| JPS4938273B1 (da) | 1974-10-16 |
| DK138496C (da) | 1979-02-26 |
| NL7201121A (da) | 1972-07-31 |
| CH535254A (fr) | 1973-03-31 |
| GB1333471A (en) | 1973-10-10 |
| US3818035A (en) | 1974-06-18 |
| AU3817772A (en) | 1973-07-26 |
| DE2203373A1 (de) | 1972-08-17 |
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