CA3218977A1 - A plurality of tasquinimod particles and use thereof - Google Patents

A plurality of tasquinimod particles and use thereof Download PDF

Info

Publication number
CA3218977A1
CA3218977A1 CA3218977A CA3218977A CA3218977A1 CA 3218977 A1 CA3218977 A1 CA 3218977A1 CA 3218977 A CA3218977 A CA 3218977A CA 3218977 A CA3218977 A CA 3218977A CA 3218977 A1 CA3218977 A1 CA 3218977A1
Authority
CA
Canada
Prior art keywords
range
particles
cancer
tasquinimod
dosage unit
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CA3218977A
Other languages
English (en)
French (fr)
Inventor
Hans Wannman
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Active Biotech AB
Original Assignee
Active Biotech AB
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Active Biotech AB filed Critical Active Biotech AB
Publication of CA3218977A1 publication Critical patent/CA3218977A1/en
Pending legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/47042-Quinolinones, e.g. carbostyril
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Powder Metallurgy (AREA)
CA3218977A 2021-05-25 2022-05-23 A plurality of tasquinimod particles and use thereof Pending CA3218977A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP21175623 2021-05-25
EP21175623.4 2021-05-25
PCT/EP2022/063887 WO2022248401A1 (en) 2021-05-25 2022-05-23 A plurality of tasquinimod particles and use thereof

Publications (1)

Publication Number Publication Date
CA3218977A1 true CA3218977A1 (en) 2022-12-01

Family

ID=76098832

Family Applications (1)

Application Number Title Priority Date Filing Date
CA3218977A Pending CA3218977A1 (en) 2021-05-25 2022-05-23 A plurality of tasquinimod particles and use thereof

Country Status (14)

Country Link
US (2) US12485095B2 (https=)
EP (1) EP4346773B1 (https=)
JP (1) JP2024520307A (https=)
KR (1) KR20240012436A (https=)
CN (1) CN117295492A (https=)
AU (1) AU2022281056A1 (https=)
BR (1) BR112023023715A2 (https=)
CA (1) CA3218977A1 (https=)
ES (1) ES3048983T3 (https=)
IL (1) IL308542A (https=)
MX (1) MX2023013301A (https=)
PL (1) PL4346773T3 (https=)
WO (1) WO2022248401A1 (https=)
ZA (1) ZA202311594B (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025228998A1 (en) * 2024-04-30 2025-11-06 Institut National de la Santé et de la Recherche Médicale Use of hdac4 inhibitors for the treatment of melanoma

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9801474D0 (sv) 1998-04-27 1998-04-27 Active Biotech Ab Quinoline Derivatives
SE9802549D0 (sv) 1998-07-15 1998-07-15 Active Biotech Ab Quinoline derivatives
SE0002320D0 (sv) 1999-10-25 2000-06-21 Active Biotech Ab Malignant tumors
SE0201778D0 (sv) 2002-06-12 2002-06-12 Active Biotech Ab Process for the manufacture of quinoline derivatives
SG186430A1 (en) 2010-07-09 2013-01-30 Active Biotech Ab Method for manufacturing of quinoline-3-carboxamides
EP2537517A1 (en) 2011-06-22 2012-12-26 Active Biotech AB Deuterium-enriched 4-hydroxy-5-methoxy-n,1-dimethyl-2-oxo-n-[(4-trifluoro-methyl)phenyl]-1,2-dihydroquinoline-3-carboxamide
US10213422B2 (en) 2014-04-14 2019-02-26 Yale University Compositions and methods of inhibiting histone deacetylases
JP6647287B2 (ja) 2014-09-23 2020-02-14 アクティブ バイオテック エイビー 多発性骨髄腫の治療に使用するためのキノリンカルボキサミド
MX379401B (es) 2014-11-19 2025-03-11 Active Biotech Ab Carboxamidas de quinolina para usarse en el tratamiento de leucemia.
EP3067062A1 (en) 2015-03-13 2016-09-14 Ipsen Pharma S.A.S. Combination of tasquinimod or a pharmaceutically acceptable salt thereof and a pd1 and/or pdl1 inhibitor, for use as a medicament
WO2018105943A1 (ko) 2016-12-07 2018-06-14 순천향대학교 산학협력단 폐섬유증 또는 천식의 치료 또는 완화용 약학 조성물
BR112023000892A2 (pt) 2020-07-23 2023-02-07 Univ Erasmus Med Ct Rotterdam Inibidor de uma proteína s100 para uso na prevenção ou tratamento de uma neoplasia mieloproliferativa, agente e método para identificar um indivíduo que sofre de uma neoplasia mieloproliferativa, e, métodos para identificar um indivíduo em risco de desenvolver mielofibrose e que se beneficie de um tratamento com um inibidor
ES3057099T3 (en) 2021-01-18 2026-02-26 Active Biotech Ab Tasquinimod or a pharmaceutically acceptable salt thereof for use in the treatment of myelodysplastic syndrome

Also Published As

Publication number Publication date
ZA202311594B (en) 2025-04-30
AU2022281056A1 (en) 2023-11-30
IL308542A (en) 2024-01-01
JP2024520307A (ja) 2024-05-24
BR112023023715A2 (pt) 2024-02-20
EP4346773C0 (en) 2025-07-02
US20240285532A1 (en) 2024-08-29
EP4346773B1 (en) 2025-07-02
EP4346773A1 (en) 2024-04-10
CN117295492A (zh) 2023-12-26
WO2022248401A1 (en) 2022-12-01
ES3048983T3 (en) 2025-12-12
US12485095B2 (en) 2025-12-02
KR20240012436A (ko) 2024-01-29
US20260076908A1 (en) 2026-03-19
PL4346773T3 (pl) 2025-11-03
MX2023013301A (es) 2023-12-04

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