CA2957224A1 - Method of treating prader-willi syndrome - Google Patents
Method of treating prader-willi syndrome Download PDFInfo
- Publication number
- CA2957224A1 CA2957224A1 CA2957224A CA2957224A CA2957224A1 CA 2957224 A1 CA2957224 A1 CA 2957224A1 CA 2957224 A CA2957224 A CA 2957224A CA 2957224 A CA2957224 A CA 2957224A CA 2957224 A1 CA2957224 A1 CA 2957224A1
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- Prior art keywords
- alkyl
- substituted
- oxytocin receptor
- receptor agonist
- selective oxytocin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A61K38/095—Oxytocins; Vasopressins; Related peptides
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- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
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Landscapes
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- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Endocrinology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
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| PCT/US2015/049911 WO2016044131A1 (en) | 2014-09-19 | 2015-09-14 | Method of treating prader-willi syndrome |
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| CA2957224A1 true CA2957224A1 (en) | 2016-03-24 |
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| CN110997697A (zh) | 2017-08-11 | 2020-04-10 | 辉凌公司 | 制备药物组合物的方法 |
| US20190135859A1 (en) | 2017-08-11 | 2019-05-09 | Ferring B.V. | Method of manufacturing a pharmaceutical composition |
| US10736894B2 (en) | 2018-02-15 | 2020-08-11 | Ovid Therapeutics Inc. | Methods of treating developmental syndromes with PDE10A inhibitors |
| WO2020061416A1 (en) * | 2018-09-20 | 2020-03-26 | Levo Therapeutics, Inc. | Carbetocin drug product and process for preparing same |
| CA3112185C (en) * | 2018-09-20 | 2025-10-07 | Acadia Pharmaceuticals Inc. | STABLE INTRANASAL FORMULATIONS OF CARBETOCINE |
| EP4262833A4 (en) * | 2020-12-18 | 2024-11-20 | The General Hospital Corporation | PROBIOTICS COMPOSITIONS AND METHODS OF USE THEREOF TO IMPROVE GROWTH AND SOCIAL FUNCTION IN CHILDREN |
| US20240197813A1 (en) * | 2021-03-26 | 2024-06-20 | Ot4B | Treatment of dysphagia |
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| US7544662B2 (en) | 1993-06-17 | 2009-06-09 | Carle Development Foundation | Polypeptides useful for appetite suppression |
| US6894026B1 (en) | 2000-01-11 | 2005-05-17 | Atossa Healthcare, Inc. | Long-acting oxytocin analogues for the treatment and prevention of breast cancer and psychiatric disorders |
| US20070032410A1 (en) | 2000-01-11 | 2007-02-08 | Atossa Healthcare, Inc. | Compositions and methods for the treatment of psychiatric disorders |
| US9023793B2 (en) | 2006-09-29 | 2015-05-05 | Retrophin, Inc. | Intranasal carbetocin formulations and methods for the treatment of autism |
| WO2008150305A1 (en) * | 2007-06-07 | 2008-12-11 | Nastech Pharmaceutical Company Inc. | Intranasal carbetocin formulations and methods for the treatment of autism |
| EP2190459A1 (en) | 2007-09-11 | 2010-06-02 | Mondobiotech Laboratories AG | Use of cnp-22, alone1 or in combination with physalemin, as a therapeutic agent |
| KR20100061680A (ko) | 2007-09-11 | 2010-06-08 | 몬도바이오테크 래보래토리즈 아게 | 치료제로서의 ｇｌｙ－ｐｒｏ－ｇｌｕ－ｏｈ（ｇｐｅ）의 용도 |
| WO2009033820A2 (en) | 2007-09-11 | 2009-03-19 | Mondobiotech Laboratories Ag | Use of a peptide as a therapeutic agent |
| US20100204112A1 (en) | 2007-09-11 | 2010-08-12 | Dorian Bevec | Use of tyr-w-mif-1 and urocortin 2 as therapeutic agents |
| WO2009122285A1 (en) * | 2008-03-31 | 2009-10-08 | Ferring B.V. | Oxitocin analogues |
| CA2731020A1 (en) | 2008-07-18 | 2010-01-21 | Zafgen, Inc. | Use of antiangiogenic fumagillins in the treatment of obesity |
| TWI463990B (zh) * | 2009-09-21 | 2014-12-11 | Ferring Bv | 催產素受體促進劑 |
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| EP2575853B1 (en) | 2010-05-25 | 2016-08-24 | INSERM - Institut National de la Santé et de la Recherche Médicale | Methods and pharmaceutical composition for the treatment of a feeding disorder with early-onset in a patient |
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| DK2935312T3 (en) | 2012-12-21 | 2018-10-22 | Hoffmann La Roche | Peptides as oxytocin agonists |
| CA2898015A1 (en) * | 2013-01-17 | 2014-07-24 | F. Hoffmann-La Roche Ag | Oxytocin receptor agonists for the treatment of cns diseases |
| EA030091B1 (ru) | 2014-06-03 | 2018-06-29 | Ф. Хоффманн-Ля Рош Аг | Пептиды, выполняющие роль агонистов окситоцина |
| CR20160562A (es) | 2014-06-06 | 2017-01-06 | Hoffmann La Roche | Péptidos como agonistas de la oxitocina |
| CN106573958A (zh) | 2014-08-07 | 2017-04-19 | 豪夫迈·罗氏有限公司 | 用于制备催产素类似物的方法 |
| CN112773765A (zh) * | 2014-09-19 | 2021-05-11 | 辉凌公司 | 治疗普拉德-威利综合征的方法 |
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- 2015-09-14 HU HUE19216650A patent/HUE065829T2/hu unknown
- 2015-09-14 PT PT192166502T patent/PT3666258T/pt unknown
- 2015-09-14 RS RS20240134A patent/RS65144B1/sr unknown
- 2015-09-14 EP EP19216650.2A patent/EP3666258B1/en active Active
- 2015-09-14 CN CN201580049147.2A patent/CN106714819A/zh active Pending
- 2015-09-14 CA CA2957224A patent/CA2957224A1/en active Pending
- 2015-09-14 JP JP2017515228A patent/JP6599447B2/ja active Active
- 2015-09-14 US US15/510,781 patent/US10441627B2/en active Active
- 2015-09-14 ES ES15772107T patent/ES2775425T3/es active Active
- 2015-09-14 WO PCT/US2015/049911 patent/WO2016044131A1/en not_active Ceased
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2019
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2021
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2022
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| CN106714819A (zh) | 2017-05-24 |
| JP6599447B2 (ja) | 2019-10-30 |
| JP2017532316A (ja) | 2017-11-02 |
| HUE065829T2 (hu) | 2024-06-28 |
| US20240082344A1 (en) | 2024-03-14 |
| US10441627B2 (en) | 2019-10-15 |
| FI3666258T3 (fi) | 2024-02-09 |
| PT3666258T (pt) | 2024-02-01 |
| RS65144B1 (sr) | 2024-02-29 |
| JP6921154B2 (ja) | 2021-08-18 |
| EP3666258B1 (en) | 2023-11-15 |
| LT3666258T (lt) | 2024-01-10 |
| DK3666258T3 (da) | 2024-02-05 |
| US20170326200A1 (en) | 2017-11-16 |
| HRP20240166T1 (hr) | 2024-04-26 |
| PL3666258T3 (pl) | 2024-04-08 |
| ES2970059T3 (es) | 2024-05-24 |
| JP2020019790A (ja) | 2020-02-06 |
| US20200129584A1 (en) | 2020-04-30 |
| CN112773765A (zh) | 2021-05-11 |
| EP3193907A1 (en) | 2017-07-26 |
| JP2021098745A (ja) | 2021-07-01 |
| EP3666258A1 (en) | 2020-06-17 |
| ES2775425T3 (es) | 2020-07-27 |
| WO2016044131A1 (en) | 2016-03-24 |
| SI3666258T1 (sl) | 2024-04-30 |
| EP3193907B1 (en) | 2020-01-01 |
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