CA2943979A1 - Substituted heteroaryl compounds and methods of use - Google Patents
Substituted heteroaryl compounds and methods of use Download PDFInfo
- Publication number
- CA2943979A1 CA2943979A1 CA2943979A CA2943979A CA2943979A1 CA 2943979 A1 CA2943979 A1 CA 2943979A1 CA 2943979 A CA2943979 A CA 2943979A CA 2943979 A CA2943979 A CA 2943979A CA 2943979 A1 CA2943979 A1 CA 2943979A1
- Authority
- CA
- Canada
- Prior art keywords
- cr6r7
- compound
- cycloalkyl
- disease
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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Applications Claiming Priority (3)
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| US201461971552P | 2014-03-28 | 2014-03-28 | |
| US61/971,552 | 2014-03-28 | ||
| PCT/US2015/022864 WO2015148869A1 (en) | 2014-03-28 | 2015-03-27 | Substituted heteroaryl compounds and methods of use |
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| CA2943979A1 true CA2943979A1 (en) | 2015-10-01 |
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| EP (5) | EP3312164B1 (enExample) |
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| AU (1) | AU2015235880B2 (enExample) |
| CA (1) | CA2943979A1 (enExample) |
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| EP3312164B1 (en) * | 2014-03-28 | 2020-12-09 | Calitor Sciences, LLC | Substituted heteroaryl compounds and methods of use |
| RU2653762C1 (ru) | 2014-09-11 | 2018-05-14 | Конинклейке Филипс Н.В. | Способ управления процессом обжарки кофейных зерен и устройство для использования в процессе обжарки кофейных зерен |
| CN106478651B (zh) * | 2015-08-31 | 2019-07-09 | 广东东阳光药业有限公司 | 取代的杂芳基化合物及其组合物和用途 |
| WO2017044434A1 (en) | 2015-09-11 | 2017-03-16 | Sunshine Lake Pharma Co., Ltd. | Substituted heteroaryl compounds and methods of use |
| WO2017048675A1 (en) * | 2015-09-17 | 2017-03-23 | Sunshine Lake Pharma Co., Ltd. | Substituted heteroaryl compounds and methods of use |
| US11214565B2 (en) | 2015-11-20 | 2022-01-04 | Denali Therapeutics Inc. | Compound, compositions, and methods |
| JP6453794B2 (ja) * | 2016-03-07 | 2019-01-16 | Ckd株式会社 | 検査装置、ブリスタ包装機、ｐｔｐシートの製造方法および錠剤 |
| PT3472153T (pt) | 2016-06-16 | 2021-12-31 | Denali Therapeutics Inc | Pirimidin-2-ilamino-1h-pirazóis como inibidores de lrrk2 para uso no tratamento de distúrbios neurodegenerativos |
| US11289643B2 (en) | 2016-12-09 | 2022-03-29 | Koninklijke Philips N.V. | Actuator device and method |
| WO2018169700A1 (en) * | 2017-03-14 | 2018-09-20 | Sunshine Lake Pharma Co., Ltd. | Substituted heteroaryl compounds and methods of use |
| JP7254076B2 (ja) | 2017-11-19 | 2023-04-07 | サンシャイン・レイク・ファーマ・カンパニー・リミテッド | 置換ヘテロアリール化合物及び使用方法 |
| CN110833553A (zh) * | 2018-08-15 | 2020-02-25 | 广西梧州制药（集团）股份有限公司 | 吡唑并嘧啶衍生物在治疗Arthus反应的用途 |
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| CN118976029A (zh) * | 2019-12-16 | 2024-11-19 | 韩国化学研究院 | 用于预防或治疗帕金森病或非酒精性脂肪性肝炎的药学组合物 |
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| CN116157388A (zh) * | 2020-09-10 | 2023-05-23 | 四川海思科制药有限公司 | 一种碳环酰胺衍生物及其在医药上的应用 |
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- 2015-03-27 US US14/670,421 patent/US9403801B2/en active Active
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- 2015-03-27 MX MX2016012574A patent/MX2016012574A/es unknown
- 2015-03-27 JP JP2017502934A patent/JP6538148B2/ja active Active
- 2015-03-27 WO PCT/US2015/022862 patent/WO2015148867A1/en not_active Ceased
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- 2015-03-27 AU AU2015235880A patent/AU2015235880B2/en active Active
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|---|---|
| EP3122730A4 (en) | 2017-08-09 |
| EP3122729A1 (en) | 2017-02-01 |
| US9399637B2 (en) | 2016-07-26 |
| EP3122730A1 (en) | 2017-02-01 |
| WO2015148867A1 (en) | 2015-10-01 |
| EP3312164B1 (en) | 2020-12-09 |
| EP3122730B1 (en) | 2020-03-25 |
| JP2017510642A (ja) | 2017-04-13 |
| EP3122728A1 (en) | 2017-02-01 |
| EP3312164A1 (en) | 2018-04-25 |
| JP6517318B2 (ja) | 2019-05-22 |
| AU2015235880A1 (en) | 2016-09-15 |
| WO2015148869A1 (en) | 2015-10-01 |
| US20150274747A1 (en) | 2015-10-01 |
| JP2017510643A (ja) | 2017-04-13 |
| JP6517319B2 (ja) | 2019-05-22 |
| MX2016012574A (es) | 2017-09-26 |
| AU2015235880B2 (en) | 2018-11-01 |
| US9403801B2 (en) | 2016-08-02 |
| EP3122729A4 (en) | 2017-11-15 |
| EP3327006A1 (en) | 2018-05-30 |
| JP2017510644A (ja) | 2017-04-13 |
| EP3122728A4 (en) | 2017-10-25 |
| US20150274705A1 (en) | 2015-10-01 |
| US20150274704A1 (en) | 2015-10-01 |
| WO2015148868A1 (en) | 2015-10-01 |
| US9394281B2 (en) | 2016-07-19 |
| JP6538148B2 (ja) | 2019-07-03 |
| EP3327006B1 (en) | 2020-05-20 |
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