CA2826871A1 - 3-hydroxy-6h-benzo [c] chromene-6-one derivative and manufacturing method thereof - Google Patents

3-hydroxy-6h-benzo [c] chromene-6-one derivative and manufacturing method thereof Download PDF

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Publication number
CA2826871A1
CA2826871A1 CA2826871A CA2826871A CA2826871A1 CA 2826871 A1 CA2826871 A1 CA 2826871A1 CA 2826871 A CA2826871 A CA 2826871A CA 2826871 A CA2826871 A CA 2826871A CA 2826871 A1 CA2826871 A1 CA 2826871A1
Authority
CA
Canada
Prior art keywords
group
formula
salt
compound
hydroxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2826871A
Other languages
English (en)
French (fr)
Inventor
Kazuhiro Kudou
Noriyoshi Yamamoto
Masakazu Ban
Atsushi Ohno
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ayumi Pharmaceutical Corp
Original Assignee
Santen Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Santen Pharmaceutical Co Ltd filed Critical Santen Pharmaceutical Co Ltd
Publication of CA2826871A1 publication Critical patent/CA2826871A1/en
Abandoned legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrane Compounds (AREA)
CA2826871A 2011-02-09 2012-02-08 3-hydroxy-6h-benzo [c] chromene-6-one derivative and manufacturing method thereof Abandoned CA2826871A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2011-026188 2011-02-09
JP2011026188 2011-02-09
PCT/JP2012/052824 WO2012108455A1 (ja) 2011-02-09 2012-02-08 ３－ヒドロキシ－６Ｈ－ベンゾ［ｃ］クロメン－６－オン誘導体およびその製造方法

Publications (1)

Publication Number Publication Date
CA2826871A1 true CA2826871A1 (en) 2012-08-16

Family

ID=46638668

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2826871A Abandoned CA2826871A1 (en) 2011-02-09 2012-02-08 3-hydroxy-6h-benzo [c] chromene-6-one derivative and manufacturing method thereof

Country Status (8)

Country Link
US (2) US8802869B2 (enExample)
EP (1) EP2674422A4 (enExample)
JP (1) JP5921235B2 (enExample)
KR (1) KR20140002735A (enExample)
CN (1) CN103370310A (enExample)
CA (1) CA2826871A1 (enExample)
TW (1) TW201309663A (enExample)
WO (1) WO2012108455A1 (enExample)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9381187B2 (en) 2011-02-16 2016-07-05 Paloma Pharmaceuticals, Inc. Radiation countermeasure agents
EP3663287B1 (en) * 2013-12-23 2023-09-20 Amazentis SA Process scale synthesis of urolithins
WO2015154047A1 (en) * 2014-04-03 2015-10-08 Restorgenex Corporation Novel methods
CN105884739B (zh) * 2016-04-14 2018-04-27 广西大学 一种苯并香豆素多环化合物的合成方法
JPWO2018230713A1 (ja) 2017-06-16 2020-04-16 学校法人同志社 カスパーゼ阻害活性を有する化合物、これらの化合物を含む、角膜内皮の症状、障害または疾患を治療または予防するための医薬およびその応用
CN110944668A (zh) 2017-06-16 2020-03-31 学校法人同志社 用于治疗或预防眼部症状、障碍或疾病的包含mTOR抑制剂的药物及其应用
JP7449232B2 (ja) * 2018-02-27 2024-03-13 アマゼンティス エスアー ウロリチンａのプロセススケール合成
CN111039913A (zh) * 2018-10-15 2020-04-21 韦忠友 一种具有抗肿瘤作用的化合物的制备方法
MX2023008677A (es) 2021-01-27 2023-10-03 Vandria Sa Derivados de urolitinas y métodos para su uso.
CN120693339A (zh) 2022-10-25 2025-09-23 Artus治疗股份有限公司 用于增强上皮和/或内皮屏障功能的治疗剂
CN119661547A (zh) * 2023-09-20 2025-03-21 科辉智药(深圳)新药研究中心有限公司 作为sarm1酶活性抑制剂的三环吡啶类化合物及其应用
CN117756766B (zh) * 2023-12-20 2026-02-17 常州大学 3-羟基-8-氟-6H-苯并[c]色烯-6-酮类衍生物及其制备方法和应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004073612A2 (en) * 2003-02-13 2004-09-02 Merck & Co. Inc. Estrogen receptor modulators
US20050282781A1 (en) * 2004-06-18 2005-12-22 Shibnath Ghosal Compositions of stable bioactive metabolites of docosahexaenoic (DHA) and eicosapentaenoic (EPA) acids
EP1944290B1 (en) 2005-09-14 2013-12-04 Santen Pharmaceutical Co., Ltd. Novel 1-2-dihydroquinoline derivative having glucocorticoid receptor binding activity
PL2085387T3 (pl) 2006-11-14 2013-09-30 Ayumi Pharmaceutical Corp Nowe pochodne 1,2-dihydrochinoliny zawierające jako podstawniki fenylochalkogeno-podstawioną niższą grupę alkilową oraz wprowadzoną przez ester grupę fenylową
KR20110010634A (ko) * 2008-05-12 2011-02-01 산텐 세이야꾸 가부시키가이샤 치환 옥시기를 가지는 2,2,4-트리메틸-6-페닐-1,2-디하이드로퀴놀린 유도체를 포함하는 글루코코르티코이드 수용체 작용제

Also Published As

Publication number Publication date
WO2012108455A1 (ja) 2012-08-16
US20130310576A1 (en) 2013-11-21
JP2012180345A (ja) 2012-09-20
US20140296540A1 (en) 2014-10-02
US9029572B2 (en) 2015-05-12
TW201309663A (zh) 2013-03-01
EP2674422A1 (en) 2013-12-18
KR20140002735A (ko) 2014-01-08
CN103370310A (zh) 2013-10-23
US8802869B2 (en) 2014-08-12
EP2674422A4 (en) 2015-01-21
JP5921235B2 (ja) 2016-05-24

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Date Code Title Description
FZDE Discontinued

Effective date: 20180208