CA2791630A1 - Combination pharmaceutical agents as inhibitors of hcv replication - Google Patents
Combination pharmaceutical agents as inhibitors of hcv replication Download PDFInfo
- Publication number
- CA2791630A1 CA2791630A1 CA2791630A CA2791630A CA2791630A1 CA 2791630 A1 CA2791630 A1 CA 2791630A1 CA 2791630 A CA2791630 A CA 2791630A CA 2791630 A CA2791630 A CA 2791630A CA 2791630 A1 CA2791630 A1 CA 2791630A1
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- CA
- Canada
- Prior art keywords
- hcv
- optionally substituted
- compound
- additional agent
- composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Landscapes
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| PCT/US2010/044591 WO2011109037A1 (en) | 2010-03-04 | 2010-08-05 | Combination pharmaceutical agents as inhibitors of hcv replication |
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| MX2011006332A (es) | 2008-12-23 | 2011-06-27 | Abbott Lab | Compuestos antivirales. |
| JP2012513410A (ja) | 2008-12-23 | 2012-06-14 | アボット・ラボラトリーズ | 抗ウイルス化合物 |
| US8242156B2 (en) * | 2009-02-17 | 2012-08-14 | Enanta Pharmaceuticals, Inc. | Linked dibenzimidazole derivatives |
| US8673954B2 (en) | 2009-02-27 | 2014-03-18 | Enanta Pharmaceuticals, Inc. | Benzimidazole derivatives |
| US9765087B2 (en) | 2009-02-27 | 2017-09-19 | Enanta Pharmaceuticals, Inc. | Benzimidazole derivatives |
| US10752611B2 (en) | 2009-02-27 | 2020-08-25 | Enanta Pharmaceuticals, Inc. | Benzimidazole derivatives |
| US8101643B2 (en) * | 2009-02-27 | 2012-01-24 | Enanta Pharmaceuticals, Inc. | Benzimidazole derivatives |
| US8507522B2 (en) * | 2009-03-06 | 2013-08-13 | Enanta Pharmaceuticals, Inc. | Hepatitis C virus inhibitors |
| EP2419404B1 (en) * | 2009-04-15 | 2015-11-04 | AbbVie Inc. | Anti-viral compounds |
| US8937150B2 (en) | 2009-06-11 | 2015-01-20 | Abbvie Inc. | Anti-viral compounds |
| US9394279B2 (en) | 2009-06-11 | 2016-07-19 | Abbvie Inc. | Anti-viral compounds |
| DK2368890T3 (da) * | 2009-06-11 | 2013-07-22 | Abbvie Bahamas Ltd | Hepatitis C-virusinhibitorer |
| US8716454B2 (en) | 2009-06-11 | 2014-05-06 | Abbvie Inc. | Solid compositions |
| CN102656160A (zh) | 2009-07-16 | 2012-09-05 | 顶点制药公司 | 用于治疗或预防黄病毒感染的苯并咪唑类似物 |
| EP2512480A4 (en) * | 2009-12-14 | 2013-05-15 | Enanta Pharm Inc | HEPATITIS C-VIRUS HEMMER |
| WO2011075607A1 (en) * | 2009-12-18 | 2011-06-23 | Intermune, Inc. | Novel inhibitors of hepatitis c virus replication |
| PE20130244A1 (es) * | 2010-01-25 | 2013-03-10 | Enanta Pharm Inc | Inhibidores del virus de la hepatitis c |
| US8933110B2 (en) | 2010-01-25 | 2015-01-13 | Enanta Pharmaceuticals, Inc. | Hepatitis C virus inhibitors |
| JP2013522375A (ja) | 2010-03-24 | 2013-06-13 | バーテックス ファーマシューティカルズ インコーポレイテッド | フラビウイルス感染を処置または予防するためのアナログ |
| CA2800509A1 (en) | 2010-05-24 | 2011-12-01 | Presidio Pharmaceuticals, Inc. | Inhibitors of hcv ns5a |
| EP2575819A4 (en) | 2010-06-04 | 2013-11-27 | Enanta Pharm Inc | INHIBITORS OF HEPATITIS C VIRUS |
| NZ605440A (en) | 2010-06-10 | 2014-05-30 | Abbvie Bahamas Ltd | Solid compositions comprising an hcv inhibitor |
| EP2593565A4 (en) * | 2010-07-16 | 2013-12-04 | Bristol Myers Squibb Co | METHODS FOR IDENTIFYING COMBINATIONS OF NS5A TARGETING COMPOUNDS THAT SYNERGISTICALLY WORK TO INHIBIT THE REPLICATION OF HEPATITIS C VIRUS |
| US8697704B2 (en) | 2010-08-12 | 2014-04-15 | Enanta Pharmaceuticals, Inc. | Hepatitis C virus inhibitors |
| WO2012083170A1 (en) * | 2010-12-16 | 2012-06-21 | Abbott Laboratories | Anti-viral compounds |
| US8552047B2 (en) | 2011-02-07 | 2013-10-08 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| US9243025B2 (en) | 2011-03-31 | 2016-01-26 | Idenix Pharmaceuticals, Llc | Compounds and pharmaceutical compositions for the treatment of viral infections |
| US9546160B2 (en) | 2011-05-12 | 2017-01-17 | Bristol-Myers Squibb Company | Hepatitis C virus inhibitors |
| US10201584B1 (en) | 2011-05-17 | 2019-02-12 | Abbvie Inc. | Compositions and methods for treating HCV |
| CN103687489A (zh) | 2011-05-18 | 2014-03-26 | 埃南塔制药公司 | 制备5-氮杂螺[2.4]庚烷-6-甲酸及其衍生物的方法 |
| CN103781786A (zh) * | 2011-07-15 | 2014-05-07 | 盐野义制药株式会社 | 具有ampk活化作用的氮杂苯并咪唑衍生物 |
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| AU2013217224B2 (en) | 2012-02-10 | 2017-04-06 | Lupin Limited | Antiviral compounds with a dibenzooxaheterocycle moiety |
| KR20140145126A (ko) * | 2012-02-13 | 2014-12-22 | 프레시디오 파마슈티칼스, 인코포레이티드 | Hcv ns5a의 저해제를 포함하는 고체형태, 이의 조성물 및 이에 의한 용도 |
| EP2852605B1 (en) | 2012-05-22 | 2018-01-31 | Idenix Pharmaceuticals LLC | 3',5'-cyclic phosphate prodrugs for hcv infection |
| EP2852604B1 (en) | 2012-05-22 | 2017-04-12 | Idenix Pharmaceuticals LLC | 3',5'-cyclic phosphoramidate prodrugs for hcv infection |
| BR112014029115A8 (pt) | 2012-05-22 | 2018-04-03 | Idenix Pharmaceuticals Inc | Composto, composição farmacêutica, e, uso de um composto ou composição |
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| US20150023913A1 (en) | 2013-07-02 | 2015-01-22 | Bristol-Myers Squibb Company | Hepatitis C Virus Inhibitors |
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- 2010-08-05 EP EP10847147.5A patent/EP2542074A4/en not_active Withdrawn
- 2010-08-05 US US12/851,350 patent/US9060971B2/en not_active Expired - Fee Related
- 2010-08-05 EA EA201201235A patent/EA201201235A1/ru unknown
- 2010-08-05 MX MX2012010252A patent/MX2012010252A/es not_active Application Discontinuation
- 2010-08-05 AU AU2010347272A patent/AU2010347272A1/en not_active Abandoned
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- 2010-08-05 JP JP2012556049A patent/JP2013521279A/ja active Pending
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| EP2542074A1 (en) | 2013-01-09 |
| US9060971B2 (en) | 2015-06-23 |
| BR112012022311A2 (pt) | 2016-08-23 |
| US20110217261A1 (en) | 2011-09-08 |
| KR20120124495A (ko) | 2012-11-13 |
| CN102858157A (zh) | 2013-01-02 |
| JP2013521279A (ja) | 2013-06-10 |
| EA201201235A1 (ru) | 2013-04-30 |
| MX2012010252A (es) | 2013-02-01 |
| WO2011109037A1 (en) | 2011-09-09 |
| AU2010347272A1 (en) | 2012-09-20 |
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