CA2479453A1 - Use of benzimidazole analogs in the treatment of cell proliferation - Google Patents

Use of benzimidazole analogs in the treatment of cell proliferation Download PDF

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Publication number
CA2479453A1
CA2479453A1 CA002479453A CA2479453A CA2479453A1 CA 2479453 A1 CA2479453 A1 CA 2479453A1 CA 002479453 A CA002479453 A CA 002479453A CA 2479453 A CA2479453 A CA 2479453A CA 2479453 A1 CA2479453 A1 CA 2479453A1
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CA
Canada
Prior art keywords
substituted
group
aryl
cycloalkyl
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002479453A
Other languages
English (en)
French (fr)
Inventor
Mark L. Richards
Jagadish C. Sircar
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Avanir Pharmaceuticals Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2479453A1 publication Critical patent/CA2479453A1/en
Abandoned legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CA002479453A 2002-03-25 2003-03-06 Use of benzimidazole analogs in the treatment of cell proliferation Abandoned CA2479453A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US36768602P 2002-03-25 2002-03-25
US60/367,686 2002-03-25
PCT/US2003/006981 WO2003082186A2 (en) 2002-03-25 2003-03-06 Use of benzimidazole analogs in the treatment of cell proliferation

Publications (1)

Publication Number Publication Date
CA2479453A1 true CA2479453A1 (en) 2003-10-09

Family

ID=28675384

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002479453A Abandoned CA2479453A1 (en) 2002-03-25 2003-03-06 Use of benzimidazole analogs in the treatment of cell proliferation

Country Status (9)

Country Link
US (1) US20050197375A1 (enExample)
EP (1) EP1494668A4 (enExample)
JP (1) JP2005525389A (enExample)
AU (1) AU2003213768A1 (enExample)
CA (1) CA2479453A1 (enExample)
PE (1) PE20040165A1 (enExample)
TW (1) TW200304820A (enExample)
UY (1) UY27732A1 (enExample)
WO (1) WO2003082186A2 (enExample)

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Also Published As

Publication number Publication date
WO2003082186A2 (en) 2003-10-09
EP1494668A4 (en) 2007-03-21
WO2003082186A3 (en) 2004-03-25
JP2005525389A (ja) 2005-08-25
AU2003213768A1 (en) 2003-10-13
PE20040165A1 (es) 2004-06-11
US20050197375A1 (en) 2005-09-08
UY27732A1 (es) 2003-10-31
TW200304820A (en) 2003-10-16
EP1494668A2 (en) 2005-01-12
AU2003213768A8 (en) 2003-10-13

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