CA2250250A1 - Novel oxazolidine derivatives, process for their production and medicaments containing them - Google Patents

Novel oxazolidine derivatives, process for their production and medicaments containing them Download PDF

Info

Publication number
CA2250250A1
CA2250250A1 CA002250250A CA2250250A CA2250250A1 CA 2250250 A1 CA2250250 A1 CA 2250250A1 CA 002250250 A CA002250250 A CA 002250250A CA 2250250 A CA2250250 A CA 2250250A CA 2250250 A1 CA2250250 A1 CA 2250250A1
Authority
CA
Canada
Prior art keywords
residue
denotes
alkyl
amino
piperidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002250250A
Other languages
English (en)
French (fr)
Inventor
Christos Tsaklakidis
Liesel Dorge
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Roche Diagnostics GmbH
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19612827A external-priority patent/DE19612827A1/de
Priority claimed from DE1996154479 external-priority patent/DE19654479A1/de
Application filed by Individual filed Critical Individual
Publication of CA2250250A1 publication Critical patent/CA2250250A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
CA002250250A 1996-03-30 1997-03-26 Novel oxazolidine derivatives, process for their production and medicaments containing them Abandoned CA2250250A1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19612827A DE19612827A1 (de) 1996-03-30 1996-03-30 Neue Oxazolidinonderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel
DE19612827.7 1996-03-30
DE1996154479 DE19654479A1 (de) 1996-12-27 1996-12-27 Neue Oxazolidinderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel
DE19654479.3 1996-12-27

Publications (1)

Publication Number Publication Date
CA2250250A1 true CA2250250A1 (en) 1997-10-09

Family

ID=26024325

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002250250A Abandoned CA2250250A1 (en) 1996-03-30 1997-03-26 Novel oxazolidine derivatives, process for their production and medicaments containing them

Country Status (16)

Country Link
EP (1) EP0891359A1 (de)
JP (1) JP2000510445A (de)
KR (1) KR20000005117A (de)
CN (1) CN1219933A (de)
AR (1) AR006452A1 (de)
AU (1) AU722747B2 (de)
BR (1) BR9708475A (de)
CA (1) CA2250250A1 (de)
CZ (1) CZ305198A3 (de)
HU (1) HUP9901741A3 (de)
IL (1) IL126390A0 (de)
NO (1) NO984547L (de)
NZ (1) NZ332245A (de)
PL (1) PL329053A1 (de)
TR (1) TR199801961T2 (de)
WO (1) WO1997036899A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999032486A1 (en) * 1997-12-23 1999-07-01 Alcon Laboratories, Inc. Muscarinic agents and use thereof to treat glaucoma, myopia and various other conditions
WO2002074762A1 (fr) * 2001-03-15 2002-09-26 Takeda Chemical Industries, Ltd. Procede relatif a l'elaboration de derive sulfone
EP1598340B1 (de) * 2001-04-18 2009-03-04 Euro-Celtique S.A. 1-(4-piperidinyl)-1,3-dihydro-2h-benzoxazole-2-one derivate und verwandte verbindungen als nociceptin analoge und orl1 liganden zur behandlung von schmerz
JPWO2003095446A1 (ja) * 2002-05-09 2005-09-15 持田製薬株式会社 1−(4−ピリジル)−4−ピペリドンの製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9122016D0 (en) * 1991-10-16 1991-11-27 Glaxo Group Ltd Chemical compounds
AU2915892A (en) * 1991-11-14 1993-06-15 Glaxo Group Limited Piperidine acetic acid derivatives as inhibitors of fibrinogen-dependent blood platelet aggregation
WO1993014077A1 (en) * 1992-01-21 1993-07-22 Glaxo Group Limited Piperidineacetic acid derivatives as inhibitors of fibrinogen-dependent blood platelet aggregation
ATE181735T1 (de) * 1993-05-01 1999-07-15 Merck Patent Gmbh Substituierte 1-phenyl-oxazolidin-2-on derivate, deren herstellung und deren verwendung als adhäsionsrezeptor-antagonisten
DE19524765A1 (de) * 1995-07-07 1997-01-09 Boehringer Mannheim Gmbh Neue Oxazolidinonderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel

Also Published As

Publication number Publication date
CN1219933A (zh) 1999-06-16
NO984547D0 (no) 1998-09-29
PL329053A1 (en) 1999-03-01
NO984547L (no) 1998-11-30
AU2505697A (en) 1997-10-22
EP0891359A1 (de) 1999-01-20
HUP9901741A3 (en) 2000-03-28
HUP9901741A2 (hu) 1999-09-28
NZ332245A (en) 2000-03-27
AR006452A1 (es) 1999-08-25
KR20000005117A (ko) 2000-01-25
AU722747B2 (en) 2000-08-10
TR199801961T2 (xx) 1999-01-18
CZ305198A3 (cs) 1999-02-17
JP2000510445A (ja) 2000-08-15
IL126390A0 (en) 1999-05-09
BR9708475A (pt) 1999-04-13
WO1997036899A1 (de) 1997-10-09

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Legal Events

Date Code Title Description
FZDE Discontinued