CA2121898A1 - Synthesis of prototypes for renin inhibitors - Google Patents
Synthesis of prototypes for renin inhibitorsInfo
- Publication number
- CA2121898A1 CA2121898A1 CA002121898A CA2121898A CA2121898A1 CA 2121898 A1 CA2121898 A1 CA 2121898A1 CA 002121898 A CA002121898 A CA 002121898A CA 2121898 A CA2121898 A CA 2121898A CA 2121898 A1 CA2121898 A1 CA 2121898A1
- Authority
- CA
- Canada
- Prior art keywords
- carbon atoms
- alkyl
- mmol
- compound
- chch3
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/02—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from isocyanates with formation of carbamate groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Priority Applications (14)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CA002121898A CA2121898A1 (en) | 1994-04-21 | 1994-04-21 | Synthesis of prototypes for renin inhibitors |
EP95913311A EP0756590A1 (de) | 1994-04-21 | 1995-04-12 | Synthese von renin-inhibitor-prototypen |
CN95192655A CN1147810A (zh) | 1994-04-21 | 1995-04-12 | 原型血管紧张肽原酶抑制剂的合成 |
CZ963065A CZ306596A3 (en) | 1994-04-21 | 1995-04-12 | Process for preparing prototypes of renin inhibitors |
PCT/IB1995/000257 WO1995029150A1 (en) | 1994-04-21 | 1995-04-12 | Synthesis of prototypes for renin inhibitors |
HU9602892A HUT74743A (en) | 1994-04-21 | 1995-04-12 | Synthesis of prototypes for renin inhibitors and new intermediates |
JP7527500A JPH09512266A (ja) | 1994-04-21 | 1995-04-12 | レニン阻害剤に対するプロトタイプの合成 |
CA 2188294 CA2188294A1 (en) | 1994-04-21 | 1995-04-12 | Synthesis of prototypes for renin inhibitors |
AU20823/95A AU2082395A (en) | 1994-04-21 | 1995-04-12 | Synthesis of prototypes for renin inhibitors |
PL95316677A PL316677A1 (en) | 1994-04-21 | 1995-04-12 | Synthesis of prototypes for renin inhibitors |
IL11340195A IL113401A0 (en) | 1994-04-21 | 1995-04-17 | Synthesis of prototypes for renin inhibitors |
ZA953187A ZA953187B (en) | 1994-04-21 | 1995-04-20 | Synthesis of prototypes for renin inhibitors |
NO963831A NO963831D0 (no) | 1994-04-21 | 1996-09-13 | Syntese av prototyper for renin-inhibitorer |
FI963743A FI963743A (fi) | 1994-04-21 | 1996-09-20 | Reniini-inhibiittorien prototyyppien synteesi |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CA002121898A CA2121898A1 (en) | 1994-04-21 | 1994-04-21 | Synthesis of prototypes for renin inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2121898A1 true CA2121898A1 (en) | 1995-10-22 |
Family
ID=4153433
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002121898A Abandoned CA2121898A1 (en) | 1994-04-21 | 1994-04-21 | Synthesis of prototypes for renin inhibitors |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP0756590A1 (de) |
JP (1) | JPH09512266A (de) |
CN (1) | CN1147810A (de) |
AU (1) | AU2082395A (de) |
CA (1) | CA2121898A1 (de) |
CZ (1) | CZ306596A3 (de) |
FI (1) | FI963743A (de) |
HU (1) | HUT74743A (de) |
IL (1) | IL113401A0 (de) |
PL (1) | PL316677A1 (de) |
WO (1) | WO1995029150A1 (de) |
ZA (1) | ZA953187B (de) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10205862A1 (de) * | 2002-02-13 | 2003-08-21 | Bayer Cropscience Ag | DELTA1-Pyrroline |
GB0511686D0 (en) * | 2005-06-08 | 2005-07-13 | Novartis Ag | Organic compounds |
CN109422664B (zh) * | 2017-08-23 | 2022-02-18 | 中国科学院福建物质结构研究所 | 一类干扰素调节剂及其制备方法和用途 |
-
1994
- 1994-04-21 CA CA002121898A patent/CA2121898A1/en not_active Abandoned
-
1995
- 1995-04-12 AU AU20823/95A patent/AU2082395A/en not_active Abandoned
- 1995-04-12 EP EP95913311A patent/EP0756590A1/de not_active Withdrawn
- 1995-04-12 PL PL95316677A patent/PL316677A1/xx unknown
- 1995-04-12 JP JP7527500A patent/JPH09512266A/ja active Pending
- 1995-04-12 HU HU9602892A patent/HUT74743A/hu unknown
- 1995-04-12 CN CN95192655A patent/CN1147810A/zh active Pending
- 1995-04-12 WO PCT/IB1995/000257 patent/WO1995029150A1/en not_active Application Discontinuation
- 1995-04-12 CZ CZ963065A patent/CZ306596A3/cs unknown
- 1995-04-17 IL IL11340195A patent/IL113401A0/xx unknown
- 1995-04-20 ZA ZA953187A patent/ZA953187B/xx unknown
-
1996
- 1996-09-20 FI FI963743A patent/FI963743A/fi not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP0756590A1 (de) | 1997-02-05 |
CZ306596A3 (en) | 1997-01-15 |
HU9602892D0 (en) | 1996-12-30 |
AU2082395A (en) | 1995-11-16 |
WO1995029150A1 (en) | 1995-11-02 |
HUT74743A (en) | 1997-02-28 |
ZA953187B (en) | 1995-10-23 |
FI963743A0 (fi) | 1996-09-20 |
FI963743A (fi) | 1996-09-20 |
JPH09512266A (ja) | 1997-12-09 |
PL316677A1 (en) | 1997-02-03 |
IL113401A0 (en) | 1995-07-31 |
CN1147810A (zh) | 1997-04-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FZDE | Discontinued | ||
FZDE | Discontinued |
Effective date: 19970421 |