CA2121898A1 - Synthese de prototypes d'inhibiteurs de la renine - Google Patents

Synthese de prototypes d'inhibiteurs de la renine

Info

Publication number
CA2121898A1
CA2121898A1 CA002121898A CA2121898A CA2121898A1 CA 2121898 A1 CA2121898 A1 CA 2121898A1 CA 002121898 A CA002121898 A CA 002121898A CA 2121898 A CA2121898 A CA 2121898A CA 2121898 A1 CA2121898 A1 CA 2121898A1
Authority
CA
Canada
Prior art keywords
carbon atoms
alkyl
mmol
compound
chch3
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002121898A
Other languages
English (en)
Inventor
Stephen Hanessian
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Priority to CA002121898A priority Critical patent/CA2121898A1/fr
Priority to PL95316677A priority patent/PL316677A1/xx
Priority to PCT/IB1995/000257 priority patent/WO1995029150A1/fr
Priority to CA 2188294 priority patent/CA2188294A1/fr
Priority to AU20823/95A priority patent/AU2082395A/en
Priority to CN95192655A priority patent/CN1147810A/zh
Priority to CZ963065A priority patent/CZ306596A3/cs
Priority to EP95913311A priority patent/EP0756590A1/fr
Priority to JP7527500A priority patent/JPH09512266A/ja
Priority to HU9602892A priority patent/HUT74743A/hu
Priority to IL11340195A priority patent/IL113401A0/xx
Priority to ZA953187A priority patent/ZA953187B/xx
Publication of CA2121898A1 publication Critical patent/CA2121898A1/fr
Priority to NO963831A priority patent/NO963831D0/no
Priority to FI963743A priority patent/FI963743A/fi
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/02—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from isocyanates with formation of carbamate groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
CA002121898A 1994-04-21 1994-04-21 Synthese de prototypes d'inhibiteurs de la renine Abandoned CA2121898A1 (fr)

Priority Applications (14)

Application Number Priority Date Filing Date Title
CA002121898A CA2121898A1 (fr) 1994-04-21 1994-04-21 Synthese de prototypes d'inhibiteurs de la renine
EP95913311A EP0756590A1 (fr) 1994-04-21 1995-04-12 Synthese des prototypes des inhibiteurs de la renine
JP7527500A JPH09512266A (ja) 1994-04-21 1995-04-12 レニン阻害剤に対するプロトタイプの合成
CA 2188294 CA2188294A1 (fr) 1994-04-21 1995-04-12 Synthese des prototypes des inhibiteurs de la renine
AU20823/95A AU2082395A (en) 1994-04-21 1995-04-12 Synthesis of prototypes for renin inhibitors
CN95192655A CN1147810A (zh) 1994-04-21 1995-04-12 原型血管紧张肽原酶抑制剂的合成
CZ963065A CZ306596A3 (en) 1994-04-21 1995-04-12 Process for preparing prototypes of renin inhibitors
PL95316677A PL316677A1 (en) 1994-04-21 1995-04-12 Synthesis of prototypes for renin inhibitors
PCT/IB1995/000257 WO1995029150A1 (fr) 1994-04-21 1995-04-12 Synthese des prototypes des inhibiteurs de la renine
HU9602892A HUT74743A (en) 1994-04-21 1995-04-12 Synthesis of prototypes for renin inhibitors and new intermediates
IL11340195A IL113401A0 (en) 1994-04-21 1995-04-17 Synthesis of prototypes for renin inhibitors
ZA953187A ZA953187B (en) 1994-04-21 1995-04-20 Synthesis of prototypes for renin inhibitors
NO963831A NO963831D0 (no) 1994-04-21 1996-09-13 Syntese av prototyper for renin-inhibitorer
FI963743A FI963743A (fi) 1994-04-21 1996-09-20 Reniini-inhibiittorien prototyyppien synteesi

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CA002121898A CA2121898A1 (fr) 1994-04-21 1994-04-21 Synthese de prototypes d'inhibiteurs de la renine

Publications (1)

Publication Number Publication Date
CA2121898A1 true CA2121898A1 (fr) 1995-10-22

Family

ID=4153433

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002121898A Abandoned CA2121898A1 (fr) 1994-04-21 1994-04-21 Synthese de prototypes d'inhibiteurs de la renine

Country Status (12)

Country Link
EP (1) EP0756590A1 (fr)
JP (1) JPH09512266A (fr)
CN (1) CN1147810A (fr)
AU (1) AU2082395A (fr)
CA (1) CA2121898A1 (fr)
CZ (1) CZ306596A3 (fr)
FI (1) FI963743A (fr)
HU (1) HUT74743A (fr)
IL (1) IL113401A0 (fr)
PL (1) PL316677A1 (fr)
WO (1) WO1995029150A1 (fr)
ZA (1) ZA953187B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10205862A1 (de) * 2002-02-13 2003-08-21 Bayer Cropscience Ag DELTA1-Pyrroline
GB0511686D0 (en) * 2005-06-08 2005-07-13 Novartis Ag Organic compounds
CN109422664B (zh) * 2017-08-23 2022-02-18 中国科学院福建物质结构研究所 一类干扰素调节剂及其制备方法和用途

Also Published As

Publication number Publication date
AU2082395A (en) 1995-11-16
IL113401A0 (en) 1995-07-31
JPH09512266A (ja) 1997-12-09
HUT74743A (en) 1997-02-28
FI963743A0 (fi) 1996-09-20
CN1147810A (zh) 1997-04-16
WO1995029150A1 (fr) 1995-11-02
PL316677A1 (en) 1997-02-03
ZA953187B (en) 1995-10-23
FI963743A (fi) 1996-09-20
EP0756590A1 (fr) 1997-02-05
CZ306596A3 (en) 1997-01-15
HU9602892D0 (en) 1996-12-30

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Legal Events

Date Code Title Description
FZDE Discontinued
FZDE Discontinued

Effective date: 19970421