CA1060345A - Spermicidal vaginal composition comprising 1,2-benzisothiazole derivatives - Google Patents

Spermicidal vaginal composition comprising 1,2-benzisothiazole derivatives

Info

Publication number
CA1060345A
CA1060345A CA256,023A CA256023A CA1060345A CA 1060345 A CA1060345 A CA 1060345A CA 256023 A CA256023 A CA 256023A CA 1060345 A CA1060345 A CA 1060345A
Authority
CA
Canada
Prior art keywords
benzisothiazole
composition
radical
derivative
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA256,023A
Other languages
English (en)
French (fr)
Inventor
Adriano Butti
Giovanni Gazzani
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Prephar Prospection de Recherches Pharmaceutiques
Original Assignee
Prephar Prospection de Recherches Pharmaceutiques
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Prephar Prospection de Recherches Pharmaceutiques filed Critical Prephar Prospection de Recherches Pharmaceutiques
Application granted granted Critical
Publication of CA1060345A publication Critical patent/CA1060345A/en
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S424/00—Drug, bio-affecting and body treating compositions
    • Y10S424/14—Topical contraceptives and spermacides

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Separation Of Suspended Particles By Flocculating Agents (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Debugging And Monitoring (AREA)
CA256,023A 1975-07-03 1976-06-30 Spermicidal vaginal composition comprising 1,2-benzisothiazole derivatives Expired CA1060345A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT25051/75A IT1039699B (it) 1975-07-03 1975-07-03 Composizione spermicida a base di derivati benzisotiazolici

Publications (1)

Publication Number Publication Date
CA1060345A true CA1060345A (en) 1979-08-14

Family

ID=11215541

Family Applications (1)

Application Number Title Priority Date Filing Date
CA256,023A Expired CA1060345A (en) 1975-07-03 1976-06-30 Spermicidal vaginal composition comprising 1,2-benzisothiazole derivatives

Country Status (12)

Country Link
US (1) US4093730A (enExample)
JP (1) JPS527444A (enExample)
BE (1) BE843745A (enExample)
CA (1) CA1060345A (enExample)
DE (1) DE2629018A1 (enExample)
DK (1) DK298676A (enExample)
FR (1) FR2315927A1 (enExample)
GB (1) GB1495909A (enExample)
IL (1) IL49922A0 (enExample)
IT (1) IT1039699B (enExample)
NO (1) NO762311L (enExample)
SE (1) SE7607597L (enExample)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU522792B2 (en) * 1977-07-19 1982-06-24 Fisons Plc Pressure pack formulation
DE3041036A1 (de) * 1980-10-31 1982-06-09 A. Nattermann & Cie GmbH, 5000 Köln Verwendung von benzisothiazolen
JPS58177982A (ja) * 1982-04-09 1983-10-18 Green Cross Corp:The ベンズイソチアゾリン誘導体及び抗白癬菌剤
JPS58177915A (ja) * 1982-04-12 1983-10-18 Green Cross Corp:The 抗血栓剤
JPS6086541U (ja) * 1983-11-22 1985-06-14 株式会社幸袋工作所 コ−クス炉々蓋掃除装置
JPS6093745U (ja) * 1983-12-02 1985-06-26 株式会社幸袋工作所 コ−クス炉々蓋掃除装置
CA1340759C (en) * 1988-07-01 1999-09-21 James P. Albarella Isobenzothiazolone chromogenic thiol indicators and their derivatives
US5620997A (en) * 1995-05-31 1997-04-15 Warner-Lambert Company Isothiazolones
US6001863A (en) * 1996-11-26 1999-12-14 Warner-Lambert Company Isothiazolones
US6355648B1 (en) 1999-05-04 2002-03-12 American Home Products Corporation Thio-oxindole derivatives
US6462032B1 (en) 1999-05-04 2002-10-08 Wyeth Cyclic regimens utilizing indoline derivatives
US6423699B1 (en) 1999-05-04 2002-07-23 American Home Products Corporation Combination therapies using benzimidazolones
US6417214B1 (en) 1999-05-04 2002-07-09 Wyeth 3,3-substituted indoline derivatives
US6380235B1 (en) 1999-05-04 2002-04-30 American Home Products Corporation Benzimidazolones and analogues
US6498154B1 (en) 1999-05-04 2002-12-24 Wyeth Cyclic regimens using quinazolinone and benzoxazine derivatives
US6306851B1 (en) 1999-05-04 2001-10-23 American Home Products Corporation Cyclocarbamate and cyclic amide derivatives
US6369056B1 (en) 1999-05-04 2002-04-09 American Home Products Corporation Cyclic urea and cyclic amide derivatives
US6399593B1 (en) 1999-05-04 2002-06-04 Wyeth Cyclic regimens using cyclic urea and cyclic amide derivatives
US6407101B1 (en) 1999-05-04 2002-06-18 American Home Products Corporation Cyanopyrroles
US6358948B1 (en) 1999-05-04 2002-03-19 American Home Products Corporation Quinazolinone and benzoxazine derivatives as progesterone receptor modulators
US6444668B1 (en) 1999-05-04 2002-09-03 Wyeth Combination regimens using progesterone receptor modulators
US6319912B1 (en) 1999-05-04 2001-11-20 American Home Products Corporation Cyclic regimens using 2,1-benzisothiazoline 2,2-dioxides
US6391907B1 (en) 1999-05-04 2002-05-21 American Home Products Corporation Indoline derivatives
US6358947B1 (en) 1999-05-04 2002-03-19 American Home Products Corporation Tetracyclic progesterone receptor modulator compounds and methods
US6329416B1 (en) 1999-05-04 2001-12-11 American Home Products Corporation Combination regimens using 3,3-substituted indoline derivatives
US6339098B1 (en) 1999-05-04 2002-01-15 American Home Products Corporation 2,1-benzisothiazoline 2,2-dioxides
US6380178B1 (en) 1999-05-04 2002-04-30 American Home Products Corporation Cyclic regimens using cyclocarbamate and cyclic amide derivatives
US6509334B1 (en) 1999-05-04 2003-01-21 American Home Products Corporation Cyclocarbamate derivatives as progesterone receptor modulators
UA73119C2 (en) 2000-04-19 2005-06-15 American Home Products Corpoir Derivatives of cyclic thiocarbamates, pharmaceutical composition including noted derivatives of cyclic thiocarbamates and active ingredients of medicines as modulators of progesterone receptors
WO2003059884A1 (en) 2001-12-21 2003-07-24 X-Ceptor Therapeutics, Inc. Modulators of lxr
WO2003060078A2 (en) * 2001-12-21 2003-07-24 X-Ceptor Therapeutics, Inc. Heterocyclic modulators of nuclear receptors
US7482366B2 (en) 2001-12-21 2009-01-27 X-Ceptor Therapeutics, Inc. Modulators of LXR
WO2004075854A2 (en) * 2003-02-26 2004-09-10 Program For Appropriate Technology In Health Microbicidal compositions and method of use
US20050037033A1 (en) * 2003-05-23 2005-02-17 Program For Appropriate Technology In Health Microbicidal compositions and methods and use
WO2005019417A2 (en) * 2003-08-14 2005-03-03 The Bio Balance Corporation Bacterial strains, compositions including same and probiotic use thereof
UA93354C2 (ru) 2004-07-09 2011-02-10 Гилиад Сайенсиз, Инк. Местный противовирусный препарат
MX2012006297A (es) 2009-12-01 2012-07-23 Seprox Biotech S L Uso topico hidroxitirosol y derivados para la prevencion de la infeccion por vih.
EP2546358A1 (en) 2011-07-15 2013-01-16 Laboratorios Del. Dr. Esteve, S.A. Methods and reagents for efficient control of HIV progression
CN109503547B (zh) * 2018-12-20 2021-03-16 江苏师范大学 苯并二硫环戊二烯衍生物的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3012039A (en) * 1958-03-14 1961-12-05 Ici Ltd 2-p-chlorobenzyl-1, 2-benzisothiazolone
GB848130A (en) * 1958-03-14 1960-09-14 Ici Ltd Benzisothiazolones
GB861379A (en) * 1958-03-14 1961-02-22 Ici Ltd Therapeutic compositions comprising 1:2-benzisothiazolone derivatives
CH395094A (de) * 1960-03-24 1965-07-15 Wander Ag Dr A Verfahren zur Herstellung von 6-Chlor-benzisothiazolon
DE1147947B (de) * 1961-07-25 1963-05-02 Knoll Ag Verfahren zur Herstellung neuer 1, 2-Benzisothiazolone
SE392103B (sv) * 1970-04-27 1977-03-14 Sherwin Williams Co Sett att framstella 1,2-bensisotiazolin-3-oner

Also Published As

Publication number Publication date
US4093730A (en) 1978-06-06
JPS527444A (en) 1977-01-20
IT1039699B (it) 1979-12-10
DE2629018A1 (de) 1977-01-27
BE843745A (fr) 1977-01-03
DK298676A (da) 1977-01-04
GB1495909A (en) 1977-12-21
NO762311L (enExample) 1977-01-04
SE7607597L (sv) 1977-01-04
IL49922A0 (en) 1976-08-31
FR2315927B1 (enExample) 1979-05-04
FR2315927A1 (fr) 1977-01-28

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