BRPI0813214A2 - Processo para a preparação de 17-(3-hidroxipropil)-17-hidroxiesteróides - Google Patents

Processo para a preparação de 17-(3-hidroxipropil)-17-hidroxiesteróides

Info

Publication number
BRPI0813214A2
BRPI0813214A2 BRPI0813214-3A2A BRPI0813214A BRPI0813214A2 BR PI0813214 A2 BRPI0813214 A2 BR PI0813214A2 BR PI0813214 A BRPI0813214 A BR PI0813214A BR PI0813214 A2 BRPI0813214 A2 BR PI0813214A2
Authority
BR
Brazil
Prior art keywords
hydroxyesteroids
hydroxypropil
preparing
Prior art date
Application number
BRPI0813214-3A2A
Other languages
English (en)
Inventor
Claus-Christian Haeselhoff
Mike Petersen
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40029248&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0813214(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of BRPI0813214A2 publication Critical patent/BRPI0813214A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • C07J53/008—3 membered carbocyclic rings in position 15/16
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BRPI0813214-3A2A 2007-06-28 2008-06-27 Processo para a preparação de 17-(3-hidroxipropil)-17-hidroxiesteróides BRPI0813214A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102007030596A DE102007030596B3 (de) 2007-06-28 2007-06-28 Verfahren zur Herstellung von 17-(3-Hydroxypropyl)-17-hydroxysteroiden
PCT/EP2008/058296 WO2009000923A2 (en) 2007-06-28 2008-06-27 Process for the preparation of 17-(3-hydroxypropyl)-17-hydroxysteroids

Publications (1)

Publication Number Publication Date
BRPI0813214A2 true BRPI0813214A2 (pt) 2014-12-23

Family

ID=40029248

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0813214-3A2A BRPI0813214A2 (pt) 2007-06-28 2008-06-27 Processo para a preparação de 17-(3-hidroxipropil)-17-hidroxiesteróides

Country Status (26)

Country Link
US (2) US8853431B2 (pt)
EP (1) EP2170926B1 (pt)
JP (2) JP5643087B2 (pt)
KR (1) KR101547365B1 (pt)
CN (1) CN101743248B (pt)
AR (1) AR067194A1 (pt)
AU (1) AU2008267145B2 (pt)
BR (1) BRPI0813214A2 (pt)
CA (1) CA2690177C (pt)
CL (1) CL2008001908A1 (pt)
DE (1) DE102007030596B3 (pt)
DK (1) DK2170926T3 (pt)
ES (1) ES2514516T3 (pt)
HK (1) HK1144822A1 (pt)
HR (1) HRP20140938T1 (pt)
IL (1) IL202205A (pt)
PA (1) PA8786201A1 (pt)
PE (1) PE20090485A1 (pt)
PL (1) PL2170926T3 (pt)
PT (1) PT2170926E (pt)
RU (1) RU2466137C2 (pt)
SI (1) SI2170926T1 (pt)
TW (1) TWI437006B (pt)
UY (1) UY31188A1 (pt)
WO (1) WO2009000923A2 (pt)
ZA (1) ZA201000636B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102007030596B3 (de) * 2007-06-28 2009-03-12 Bayer Schering Pharma Aktiengesellschaft Verfahren zur Herstellung von 17-(3-Hydroxypropyl)-17-hydroxysteroiden
CN105566032B (zh) * 2014-10-09 2017-12-22 中国石油化工股份有限公司 富炔碳四的选择加氢工艺

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3113953A (en) * 1958-11-28 1963-12-10 Sterling Drug Inc Esters of 17alpha-(3-hydroxy-1-propinyl) androst-5-ene-3beta, 17beta-diol and their preparation
FR2429056A1 (fr) * 1978-06-19 1980-01-18 Tournus Manuf Metallurg Procede de fabrication de bandes composites par coulee continue
DE3042136A1 (de) * 1980-11-03 1982-06-09 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur herstellung von 3 (beta), 7 (beta) -dihydroxy- (delta) (pfeil hoch)5(pfeil hoch) -steroiden
ATE15206T1 (de) * 1981-09-21 1985-09-15 Schering Ag 3-beta,7-beta,15-alpha-trihydroxy-5-androsten-1 - one, ihre 3,15-trimethylessigsaeure-ester und ihre herstellung.
US5106995A (en) * 1989-05-05 1992-04-21 Isp Investments Inc. Production of lactones from diols
US5693280A (en) 1996-07-31 1997-12-02 Owens-Corning Fiberglas Technology, Inc. Method of producing organic fibers from a rotary process
DE19633685C1 (de) * 1996-08-12 1997-10-09 Schering Ag Verfahren zur Herstellung von Drospirenon (6beta,7beta;15 beta,16beta-Dimethyl-en-3-oxo-17alpha-pregn-4-en-21,17-carbolacton, DRSP) sowie 7alpha-(3-Hydroxy-1-propyl)-6beta,7beta;15beta, 16beta-dimethylen-5beta-androstan-3beta,5,17beta-triol (ZK 92836) und 6beta,7beta;15beta,16beta-dimethylen-5beta-hydroxy-3-oxo-17alpha-androstan-21,17-carbolacton (90965) als Zwischenprodukte des Verfahrens
WO2001058919A2 (en) * 2000-02-11 2001-08-16 Sri International Synthesis of anti-estrogenic and other therapeutic steroids from 21-hydroxy-19-norpregna-4-en-3-one
ITMI20040367A1 (it) * 2004-03-01 2004-06-01 Ind Chimica Srl Processo per la preparazione di drospirenone
ITMI20042338A1 (it) * 2004-12-06 2005-03-06 Ind Chimica Srl Processo per la preparazione di drospirenone
US7319154B2 (en) * 2005-07-21 2008-01-15 Bayer Schering Pharma Ag Process for the production of 3-oxo-pregn-4-ene-21, 17-carbolactones by the metal free oxidation of 17-(3-hydroxypropyl)-3, 17-dihydroxyandrostanes
NZ565247A (en) * 2005-07-21 2011-02-25 Bayer Schering Pharma Ag Process for the production drospirenone utilising the metal-free oxidation of 17-(3-hydroxypropyl)-3,17-dihydroxyandrostanes with TEMPO
CN100480256C (zh) * 2006-06-21 2009-04-22 上海迪赛诺医药发展有限公司 合成曲螺酮的方法
DE102007030596B3 (de) * 2007-06-28 2009-03-12 Bayer Schering Pharma Aktiengesellschaft Verfahren zur Herstellung von 17-(3-Hydroxypropyl)-17-hydroxysteroiden
ES2419663T3 (es) * 2010-08-03 2013-08-21 Newchem S.P.A. Métodos para la preparación de Drospirenona y productos intermedios de la misma

Also Published As

Publication number Publication date
TWI437006B (zh) 2014-05-11
CN101743248A (zh) 2010-06-16
PL2170926T3 (pl) 2014-12-31
TW200918548A (en) 2009-05-01
KR101547365B1 (ko) 2015-08-25
ES2514516T3 (es) 2014-10-28
US20090012286A1 (en) 2009-01-08
IL202205A0 (en) 2010-06-16
AR067194A1 (es) 2009-09-30
EP2170926A2 (en) 2010-04-07
SI2170926T1 (sl) 2014-11-28
ZA201000636B (en) 2015-06-24
AU2008267145B2 (en) 2013-10-24
CA2690177C (en) 2015-09-15
UY31188A1 (es) 2009-01-30
HRP20140938T1 (hr) 2014-12-05
CA2690177A1 (en) 2008-12-31
RU2466137C2 (ru) 2012-11-10
JP2014198724A (ja) 2014-10-23
CN101743248B (zh) 2013-01-02
DE102007030596B3 (de) 2009-03-12
CL2008001908A1 (es) 2009-01-02
WO2009000923A3 (en) 2009-04-23
DK2170926T3 (da) 2014-10-13
IL202205A (en) 2015-06-30
PE20090485A1 (es) 2009-05-24
WO2009000923A2 (en) 2008-12-31
AU2008267145A1 (en) 2008-12-31
HK1144822A1 (pt) 2011-03-11
EP2170926B1 (en) 2014-07-23
JP5643087B2 (ja) 2014-12-17
PT2170926E (pt) 2014-10-13
US20150005488A1 (en) 2015-01-01
RU2010102134A (ru) 2011-08-10
US8853431B2 (en) 2014-10-07
KR20100027158A (ko) 2010-03-10
PA8786201A1 (es) 2009-01-23
JP2010531337A (ja) 2010-09-24
JP5898731B2 (ja) 2016-04-06

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Legal Events

Date Code Title Description
B25D Requested change of name of applicant approved

Owner name: BAYER PHARMA AKTIENGESELLSCHAFT (DE)

B25A Requested transfer of rights approved

Owner name: BAYER INTELLECTUAL PROPERTY GMBH (DE)

B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B11D Dismissal acc. art. 38, par 2 of ipl - failure to pay fee after grant in time