BRPI0806418A2 - formas de dosagem oral para picoplatina, série de granulados revestidos, processo para preparar uma forma de dosagem oral para picoplatina e métodos de tratamentos do cáncer - Google Patents
formas de dosagem oral para picoplatina, série de granulados revestidos, processo para preparar uma forma de dosagem oral para picoplatina e métodos de tratamentos do cáncer Download PDFInfo
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- BRPI0806418A2 BRPI0806418A2 BRPI0806418-0A BRPI0806418A BRPI0806418A2 BR PI0806418 A2 BRPI0806418 A2 BR PI0806418A2 BR PI0806418 A BRPI0806418 A BR PI0806418A BR PI0806418 A2 BRPI0806418 A2 BR PI0806418A2
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- Prior art keywords
- picoplatin
- dosage form
- oral dosage
- coating
- core
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- A61K9/2806—Coating materials
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/28—Compounds containing heavy metals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/24—Heavy metals; Compounds thereof
- A61K33/243—Platinum; Compounds thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K33/00—Medicinal preparations containing inorganic active ingredients
- A61K33/24—Heavy metals; Compounds thereof
- A61K33/28—Mercury; Compounds thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
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- Public Health (AREA)
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- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US88917107P | 2007-02-09 | 2007-02-09 | |
| US60/889,171 | 2007-02-09 | ||
| US88968107P | 2007-02-13 | 2007-02-13 | |
| US60/889,681 | 2007-02-13 | ||
| PCT/US2008/001752 WO2008097661A1 (en) | 2007-02-09 | 2008-02-08 | Stabilized picoplatin oral dosage form |
Publications (1)
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|---|---|
| BRPI0806418A2 true BRPI0806418A2 (pt) | 2011-09-06 |
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| BRPI0806418-0A BRPI0806418A2 (pt) | 2007-02-09 | 2008-02-08 | formas de dosagem oral para picoplatina, série de granulados revestidos, processo para preparar uma forma de dosagem oral para picoplatina e métodos de tratamentos do cáncer |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP2114418A4 (enExample) |
| JP (1) | JP2010518089A (enExample) |
| KR (1) | KR20090109129A (enExample) |
| CN (2) | CN104288119A (enExample) |
| AU (1) | AU2008214202A1 (enExample) |
| BR (1) | BRPI0806418A2 (enExample) |
| CA (1) | CA2677640A1 (enExample) |
| HK (1) | HK1206267A1 (enExample) |
| IL (1) | IL200262A0 (enExample) |
| MX (1) | MX2009008488A (enExample) |
| RU (1) | RU2009133446A (enExample) |
| WO (1) | WO2008097661A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8168662B1 (en) | 2006-11-06 | 2012-05-01 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US8173686B2 (en) | 2006-11-06 | 2012-05-08 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US8168661B2 (en) | 2006-11-06 | 2012-05-01 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US8178564B2 (en) | 2006-11-06 | 2012-05-15 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US20120148661A1 (en) * | 2009-04-15 | 2012-06-14 | Poniard Pharmaceuticals, Inc. | High bioavailability oral picoplatin anti-cancer therapy |
| US9814716B2 (en) * | 2014-05-23 | 2017-11-14 | Mingsight Pharmaceuticals, Inc. | Treatment of autoimmune disease |
| CN107778331B (zh) * | 2016-08-27 | 2020-06-30 | 鲁南制药集团股份有限公司 | 一种甲啶铂的提纯方法 |
| CN108864177B (zh) * | 2018-04-20 | 2020-07-28 | 公安部物证鉴定中心 | [2h3]-1-甲氨基-2-苯基丙烷的合成方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9502799D0 (en) * | 1995-02-14 | 1995-04-05 | Johnson Matthey Plc | Improvements in platinum complexes |
| DE60032517T2 (de) * | 2000-02-16 | 2007-10-04 | Astellas Pharma Inc. | Heilmittel gegen durch endothelin verursachte erkrankungen |
| AU2002249046A1 (en) * | 2001-04-23 | 2002-11-05 | Nucryst Pharmaceuticals Corp. | Lubricious coatings for substrates |
| DE10141528B4 (de) * | 2001-08-24 | 2006-08-10 | Faustus Forschungs Cie. Translational Cancer Research Gmbh | Platin(II)- und Platin(IV)-Komplexe und ihre Verwendung |
| AU2003220022A1 (en) * | 2002-03-01 | 2003-09-16 | Trustees Of Dartmouth College | Compositions and methods for preventing sporadic neoplasia in colon |
| TWI272273B (en) * | 2002-07-16 | 2007-02-01 | Sonus Pharma Inc | Platinum compounds |
| WO2004054499A2 (en) * | 2002-08-02 | 2004-07-01 | Transave, Inc. | Platinum aggregates and process for producing the same |
| AU2005223654A1 (en) * | 2004-03-18 | 2005-09-29 | Transave, Inc. | Administration of cisplatin by inhalation |
| US20060205810A1 (en) * | 2004-11-24 | 2006-09-14 | Schering Corporation | Platinum therapeutic combinations |
-
2008
- 2008-02-08 CN CN201410283507.2A patent/CN104288119A/zh active Pending
- 2008-02-08 EP EP08725393A patent/EP2114418A4/en not_active Withdrawn
- 2008-02-08 MX MX2009008488A patent/MX2009008488A/es not_active Application Discontinuation
- 2008-02-08 RU RU2009133446/15A patent/RU2009133446A/ru not_active Application Discontinuation
- 2008-02-08 CA CA002677640A patent/CA2677640A1/en not_active Abandoned
- 2008-02-08 AU AU2008214202A patent/AU2008214202A1/en not_active Abandoned
- 2008-02-08 WO PCT/US2008/001752 patent/WO2008097661A1/en not_active Ceased
- 2008-02-08 CN CN200880011357A patent/CN101678046A/zh active Pending
- 2008-02-08 JP JP2009549128A patent/JP2010518089A/ja active Pending
- 2008-02-08 BR BRPI0806418-0A patent/BRPI0806418A2/pt not_active IP Right Cessation
- 2008-02-08 KR KR1020097018780A patent/KR20090109129A/ko not_active Withdrawn
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2009
- 2009-08-06 IL IL200262A patent/IL200262A0/en unknown
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2015
- 2015-07-21 HK HK15106959.9A patent/HK1206267A1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| RU2009133446A (ru) | 2011-03-20 |
| AU2008214202A1 (en) | 2008-08-14 |
| CN104288119A (zh) | 2015-01-21 |
| CN101678046A (zh) | 2010-03-24 |
| IL200262A0 (en) | 2010-04-29 |
| MX2009008488A (es) | 2010-01-15 |
| WO2008097661A1 (en) | 2008-08-14 |
| HK1206267A1 (en) | 2016-01-08 |
| EP2114418A1 (en) | 2009-11-11 |
| KR20090109129A (ko) | 2009-10-19 |
| CA2677640A1 (en) | 2008-08-14 |
| EP2114418A4 (en) | 2013-01-09 |
| JP2010518089A (ja) | 2010-05-27 |
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