BRPI0718396A2 - Uso de 3-alfa-androstanodiol, opcionalmente em combinação com um inibidor de pdes, no tratamento de disfunção sexual - Google Patents
Uso de 3-alfa-androstanodiol, opcionalmente em combinação com um inibidor de pdes, no tratamento de disfunção sexual Download PDFInfo
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- BRPI0718396A2 BRPI0718396A2 BRPI0718396-8A2A BRPI0718396A BRPI0718396A2 BR PI0718396 A2 BRPI0718396 A2 BR PI0718396A2 BR PI0718396 A BRPI0718396 A BR PI0718396A BR PI0718396 A2 BRPI0718396 A2 BR PI0718396A2
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- Prior art keywords
- alpha
- androstanediol
- sexual
- sexual dysfunction
- pde5
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
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- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/40—Cyclodextrins; Derivatives thereof
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
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- A—HUMAN NECESSITIES
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
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- Veterinary Medicine (AREA)
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- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Reproductive Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Inorganic Chemistry (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06076976A EP1925307A1 (en) | 2006-11-03 | 2006-11-03 | Use of 3-alpha-androstanediol in the treatment of sexual dysfunction |
| EP06076976.7 | 2006-11-03 | ||
| PCT/NL2007/050534 WO2008054214A2 (en) | 2006-11-03 | 2007-11-02 | Use of 3-alpha-androstanediol, optionally in combination with a pde5 inhibitor, in the treatment of sexual dysfunction |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0718396A2 true BRPI0718396A2 (pt) | 2013-11-26 |
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| BRPI0718396-8A2A BRPI0718396A2 (pt) | 2006-11-03 | 2007-11-02 | Uso de 3-alfa-androstanodiol, opcionalmente em combinação com um inibidor de pdes, no tratamento de disfunção sexual |
| BRPI0717856-5A2A BRPI0717856A2 (pt) | 2006-11-03 | 2007-11-02 | Usos de testosterona e um agonista 5-ht1a, e de testosterona, um inibidor de pde5 e um agonista ht1a, composição farmacêutica, e, kit de partes |
| BRPI0717963-4A2A BRPI0717963A2 (pt) | 2006-11-03 | 2007-11-02 | Uso de 3-alfa-androstanodiol, composição farmacêutica, e, kit de partes. |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0717856-5A2A BRPI0717856A2 (pt) | 2006-11-03 | 2007-11-02 | Usos de testosterona e um agonista 5-ht1a, e de testosterona, um inibidor de pde5 e um agonista ht1a, composição farmacêutica, e, kit de partes |
| BRPI0717963-4A2A BRPI0717963A2 (pt) | 2006-11-03 | 2007-11-02 | Uso de 3-alfa-androstanodiol, composição farmacêutica, e, kit de partes. |
Country Status (27)
| Country | Link |
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| US (10) | US8575139B2 (https=) |
| EP (5) | EP1925307A1 (https=) |
| JP (8) | JP2010509211A (https=) |
| KR (6) | KR101578224B1 (https=) |
| CN (6) | CN104524580A (https=) |
| AU (3) | AU2007314736B2 (https=) |
| BR (3) | BRPI0718396A2 (https=) |
| CA (3) | CA2668320C (https=) |
| CY (1) | CY1117191T1 (https=) |
| DK (1) | DK2086544T3 (https=) |
| ES (1) | ES2561946T3 (https=) |
| HR (1) | HRP20160108T1 (https=) |
| HU (1) | HUE026752T2 (https=) |
| IL (5) | IL198459A (https=) |
| ME (1) | ME02410B (https=) |
| MX (3) | MX2009004695A (https=) |
| NO (3) | NO343597B1 (https=) |
| NZ (3) | NZ577390A (https=) |
| PH (2) | PH12014501440A1 (https=) |
| PL (1) | PL2086544T3 (https=) |
| PT (1) | PT2086544E (https=) |
| RS (1) | RS54541B1 (https=) |
| RU (4) | RU2463054C2 (https=) |
| SI (1) | SI2086544T1 (https=) |
| UA (4) | UA100119C2 (https=) |
| WO (3) | WO2008054213A2 (https=) |
| ZA (3) | ZA200903837B (https=) |
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| EP1750766B1 (en) | 2004-05-11 | 2013-07-03 | Emotional Brain B.V. | Pharmaceutical formulations and uses thereof in the treatment of female sexual dysfunction |
| EP1790343A1 (en) | 2005-11-11 | 2007-05-30 | Emotional Brain B.V. | Pharmaceuticals formulations and uses thereof in the treatment of female sexual dysfunction |
| EP1925307A1 (en) | 2006-11-03 | 2008-05-28 | Emotional Brain B.V. | Use of 3-alpha-androstanediol in the treatment of sexual dysfunction |
| EP2266567A1 (en) | 2009-05-26 | 2010-12-29 | Æterna Zentaris GmbH | Use of cetrorelix in combination with PDE V inhibitors for the treatment of sex hormone dependent disorders |
| EP2266568A1 (en) | 2009-05-26 | 2010-12-29 | Æterna Zentaris GmbH | Use of LHRH antagonists in combination with PDE V inhibitors for the treatment of sex hormone dependent disorders |
| SG10201606751XA (en) * | 2011-05-13 | 2016-10-28 | Eb Ip Hybritabs B V | Drug Delivery System |
| US8633178B2 (en) | 2011-11-23 | 2014-01-21 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
| US9180091B2 (en) | 2012-12-21 | 2015-11-10 | Therapeuticsmd, Inc. | Soluble estradiol capsule for vaginal insertion |
| JP5828923B2 (ja) | 2014-01-30 | 2015-12-09 | 国立大学法人高知大学 | ニッケル粉の製造方法 |
| WO2015125650A1 (ja) | 2014-02-21 | 2015-08-27 | 国立大学法人高知大学 | ニッケル粉の製造方法 |
| JP6406613B2 (ja) | 2014-04-15 | 2018-10-17 | 住友金属鉱山株式会社 | 含有する炭素及び硫黄の濃度を低減するニッケル粉の製造方法 |
| CN103947533B (zh) * | 2014-05-15 | 2015-12-16 | 青岛理工大学 | 生长环境可控的磁化水工厂化豆芽菜生产系统 |
| RU2600845C2 (ru) | 2014-07-04 | 2016-10-27 | Общество С Ограниченной Ответственностью "Консорциум-Пик" | Применение производных оксатриазолий-5-олата для лечения сексуальных расстройств |
| US11977085B1 (en) | 2023-09-05 | 2024-05-07 | Elan Ehrlich | Date rape drug detection device and method of using same |
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| US3251436A (en) * | 1965-03-16 | 1966-05-17 | Dayton Steel Foundry Co | Spot-type disk brake |
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| US4521421A (en) * | 1983-09-26 | 1985-06-04 | Eli Lilly And Company | Treatment of sexual dysfunction |
| AU577802B2 (en) * | 1983-10-17 | 1988-10-06 | Duphar International Research B.V. | Blood-pressure lowering piperazine derivatives |
| US4596795A (en) | 1984-04-25 | 1986-06-24 | The United States Of America As Represented By The Secretary, Dept. Of Health & Human Services | Administration of sex hormones in the form of hydrophilic cyclodextrin derivatives |
| US4640921A (en) * | 1986-02-04 | 1987-02-03 | Bristol-Myers | Treatment of sexual dysfunction with buspirone |
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| US4877774A (en) | 1987-09-09 | 1989-10-31 | The United States Of America As Represented By The Department Of Health And Human Services | Administration of steroid hormones |
| CA1335106C (en) * | 1989-02-27 | 1995-04-04 | John Mehnert Schaus | Ring-substituted 2-amino-1,2,3,4-tetra-hydronaphthalenes |
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