BRPI0715620A2 - inibidores de asmase - Google Patents

inibidores de asmase Download PDF

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Publication number
BRPI0715620A2
BRPI0715620A2 BRPI0715620-0A BRPI0715620A BRPI0715620A2 BR PI0715620 A2 BRPI0715620 A2 BR PI0715620A2 BR PI0715620 A BRPI0715620 A BR PI0715620A BR PI0715620 A2 BRPI0715620 A2 BR PI0715620A2
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BR
Brazil
Prior art keywords
amino
biphenyl
carbonyl
phenyl
octyloxy
Prior art date
Application number
BRPI0715620-0A
Other languages
English (en)
Portuguese (pt)
Inventor
Karl Baumann
Andreas Billich
Berndt Oberhauser
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BRPI0715620A2 publication Critical patent/BRPI0715620A2/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/44—Amides thereof
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BRPI0715620-0A 2006-08-23 2007-08-21 inibidores de asmase BRPI0715620A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP06119350.4 2006-08-23
EP06119350 2006-08-23
PCT/EP2007/007360 WO2008022771A1 (en) 2006-08-23 2007-08-21 Amides as sphingomyeline inhibitors

Publications (1)

Publication Number Publication Date
BRPI0715620A2 true BRPI0715620A2 (pt) 2013-07-02

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Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0715620-0A BRPI0715620A2 (pt) 2006-08-23 2007-08-21 inibidores de asmase

Country Status (12)

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US (1) US8119617B2 (OSRAM)
EP (1) EP2057173B1 (OSRAM)
JP (1) JP5328652B2 (OSRAM)
KR (1) KR20090042270A (OSRAM)
CN (1) CN101501051A (OSRAM)
AU (1) AU2007287819A1 (OSRAM)
BR (1) BRPI0715620A2 (OSRAM)
CA (1) CA2659991A1 (OSRAM)
ES (1) ES2463490T3 (OSRAM)
MX (1) MX2009001933A (OSRAM)
RU (1) RU2009110243A (OSRAM)
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RU2009110243A (ru) 2010-09-27
US20100022482A1 (en) 2010-01-28
ES2463490T3 (es) 2014-05-28
JP2010501500A (ja) 2010-01-21
KR20090042270A (ko) 2009-04-29
CN101501051A (zh) 2009-08-05
EP2057173B1 (en) 2014-02-26
WO2008022771A1 (en) 2008-02-28
EP2057173A1 (en) 2009-05-13
US8119617B2 (en) 2012-02-21
AU2007287819A1 (en) 2008-02-28
CA2659991A1 (en) 2008-02-28
MX2009001933A (es) 2009-03-06

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