BRPI0708611A2 - composto; uso do composto na preparação de um medicamento para tratamento de um transtorno neurológico em um mamìmefo; método de preparação do composto; e método de tratamento de um transtorno neurológico em um mamìfero - Google Patents
composto; uso do composto na preparação de um medicamento para tratamento de um transtorno neurológico em um mamìmefo; método de preparação do composto; e método de tratamento de um transtorno neurológico em um mamìfero Download PDFInfo
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- BRPI0708611A2 BRPI0708611A2 BRPI0708611-3A BRPI0708611A BRPI0708611A2 BR PI0708611 A2 BRPI0708611 A2 BR PI0708611A2 BR PI0708611 A BRPI0708611 A BR PI0708611A BR PI0708611 A2 BRPI0708611 A2 BR PI0708611A2
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- Brazil
- Prior art keywords
- alkyl
- compound
- substituted
- compound according
- formula
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Classifications
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
Landscapes
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- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
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| US77994006P | 2006-03-07 | 2006-03-07 | |
| US60/779,940 | 2006-03-07 | ||
| PCT/US2007/005645 WO2007103347A1 (en) | 2006-03-07 | 2007-03-05 | Meridamycin analogues for the treatment of neurodegenerative disorders |
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| EP1828203A2 (en) * | 2004-12-20 | 2007-09-05 | Wyeth | Rapamycin derivatives and the uses thereof in the treatment of neurological disorders |
| RU2394036C2 (ru) * | 2004-12-20 | 2010-07-10 | Вайет | Аналоги рапамицина и их применение при лечении неврологических, пролиферативных и воспалительных заболеваний |
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| GB9318144D0 (en) | 1993-09-01 | 1993-10-20 | Sandoz Ltd | Organic compounds |
| EP0729471A1 (en) | 1993-11-19 | 1996-09-04 | Abbott Laboratories | Semisynthetic analogs of rapamycin (macrolides) being immunomodulators |
| US20050197356A1 (en) * | 2004-03-02 | 2005-09-08 | Wyeth | Non-immunosuppressive immunophilin ligands as neuroprotective and/or neuroregenerative agents |
| BRPI0508224A (pt) | 2004-03-02 | 2007-07-17 | Wyeth Corp | composto ou um sal farmaceuticamente aceitável do mesmo, cepa de actinomiceto, isolado de uma cepa, métodos para a produção de um macrolìdeo e de um composto, produto, composição, métodos de tratamento de um mamìfero e de um distúrbio neurológico, e, uso de um composto |
| JP2008501342A (ja) | 2004-06-03 | 2008-01-24 | ワイス | 複合ポリケチドを生成するための生合成遺伝子クラスター |
| US7595187B2 (en) * | 2004-11-12 | 2009-09-29 | Wyeth | Elaiophylin biosynthetic gene cluster |
| EP1828203A2 (en) | 2004-12-20 | 2007-09-05 | Wyeth | Rapamycin derivatives and the uses thereof in the treatment of neurological disorders |
| RU2394036C2 (ru) | 2004-12-20 | 2010-07-10 | Вайет | Аналоги рапамицина и их применение при лечении неврологических, пролиферативных и воспалительных заболеваний |
-
2007
- 2007-03-05 JP JP2008558346A patent/JP2009529049A/ja active Pending
- 2007-03-05 WO PCT/US2007/005645 patent/WO2007103347A1/en not_active Ceased
- 2007-03-05 MX MX2008011312A patent/MX2008011312A/es not_active Application Discontinuation
- 2007-03-05 CN CNA2007800078343A patent/CN101426796A/zh active Pending
- 2007-03-05 RU RU2008132779/04A patent/RU2008132779A/ru not_active Application Discontinuation
- 2007-03-05 EP EP07752355A patent/EP1991551A1/en not_active Withdrawn
- 2007-03-05 CA CA002643350A patent/CA2643350A1/en not_active Abandoned
- 2007-03-05 KR KR1020087021820A patent/KR20080099317A/ko not_active Withdrawn
- 2007-03-05 TW TW096107510A patent/TW200804400A/zh unknown
- 2007-03-05 US US11/713,972 patent/US7745457B2/en not_active Expired - Fee Related
- 2007-03-05 AR ARP070100899A patent/AR059738A1/es unknown
- 2007-03-05 BR BRPI0708611-3A patent/BRPI0708611A2/pt not_active Application Discontinuation
- 2007-03-05 AU AU2007223962A patent/AU2007223962A1/en not_active Abandoned
- 2007-03-09 PE PE2007000263A patent/PE20081550A1/es not_active Application Discontinuation
-
2008
- 2008-08-12 IL IL193414A patent/IL193414A0/en unknown
- 2008-08-27 NO NO20083695A patent/NO20083695L/no not_active Application Discontinuation
- 2008-09-05 ZA ZA200807678A patent/ZA200807678B/xx unknown
- 2008-09-05 EC EC2008008718A patent/ECSP088718A/es unknown
- 2008-09-05 CR CR10272A patent/CR10272A/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200807678B (en) | 2009-08-26 |
| US7745457B2 (en) | 2010-06-29 |
| AU2007223962A1 (en) | 2007-09-13 |
| KR20080099317A (ko) | 2008-11-12 |
| RU2008132779A (ru) | 2010-04-20 |
| EP1991551A1 (en) | 2008-11-19 |
| CA2643350A1 (en) | 2007-09-13 |
| CR10272A (es) | 2008-10-03 |
| MX2008011312A (es) | 2008-09-12 |
| US20070213525A1 (en) | 2007-09-13 |
| WO2007103347A1 (en) | 2007-09-13 |
| ECSP088718A (es) | 2008-10-31 |
| TW200804400A (en) | 2008-01-16 |
| NO20083695L (no) | 2008-10-03 |
| CN101426796A (zh) | 2009-05-06 |
| PE20081550A1 (es) | 2008-12-31 |
| IL193414A0 (en) | 2009-05-04 |
| AR059738A1 (es) | 2008-04-23 |
| JP2009529049A (ja) | 2009-08-13 |
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