BRPI0617772A2 - composto, composição farmacêutica, e, uso de um composto - Google Patents
composto, composição farmacêutica, e, uso de um composto Download PDFInfo
- Publication number
- BRPI0617772A2 BRPI0617772A2 BRPI0617772-7A BRPI0617772A BRPI0617772A2 BR PI0617772 A2 BRPI0617772 A2 BR PI0617772A2 BR PI0617772 A BRPI0617772 A BR PI0617772A BR PI0617772 A2 BRPI0617772 A2 BR PI0617772A2
- Authority
- BR
- Brazil
- Prior art keywords
- diaza
- bicyclo
- nonane
- methyl
- pyridazin
- Prior art date
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Classifications
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4995—Pyrazines or piperazines forming part of bridged ring systems
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Landscapes
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- Rheumatology (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200501724 | 2005-12-06 | ||
| DKPA200501724 | 2005-12-06 | ||
| PCT/EP2006/069316 WO2007065892A1 (en) | 2005-12-06 | 2006-12-05 | Novel diazabicyclic aryl derivatives and their medical use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0617772A2 true BRPI0617772A2 (pt) | 2011-08-09 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0617772-7A BRPI0617772A2 (pt) | 2005-12-06 | 2006-12-05 | composto, composição farmacêutica, e, uso de um composto |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US8173658B2 (enExample) |
| EP (2) | EP1963323B1 (enExample) |
| JP (1) | JP2009518357A (enExample) |
| KR (1) | KR20080079250A (enExample) |
| CN (1) | CN101305004B (enExample) |
| AT (1) | ATE473978T1 (enExample) |
| AU (1) | AU2006323986A1 (enExample) |
| BR (1) | BRPI0617772A2 (enExample) |
| CA (1) | CA2632642A1 (enExample) |
| DE (1) | DE602006015523D1 (enExample) |
| DK (1) | DK1963323T3 (enExample) |
| NZ (1) | NZ567048A (enExample) |
| RU (1) | RU2008110911A (enExample) |
| WO (1) | WO2007065892A1 (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2641678A1 (en) | 2006-02-10 | 2007-08-16 | Neurosearch A/S | 3,9-diazabicyclo[3.3.1]nonane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| AU2007213670A1 (en) | 2006-02-10 | 2007-08-16 | Neurosearch A/S | 3,9-diazabicyclo[3.3.1]nonane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| EP1987031A1 (en) | 2006-02-10 | 2008-11-05 | NeuroSearch A/S | 3-heteroaryl- 3,9-diazabicyclo[3.3.1]nonane derivatives as nicotinic acetylcholine receptor agonists |
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| US3293251A (en) * | 1966-12-20 | Rearrangement process for j,b-diaza- bicyclo-(j,z,i)-octane derivatives | ||
| US5478939A (en) * | 1994-07-20 | 1995-12-26 | American Cyanamid Company | (R,R) and (S,S) 2,5-diazabicyclo [2,2,1]heptane derivatives |
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| DE69811070T2 (de) * | 1997-05-30 | 2003-10-02 | Neurosearch A/S, Ballerup | 9-azabicyclo(3.3.1)non-2-ene und nonanderivate als liganden der nicotinergen rezeptoren |
| FR2786770B1 (fr) | 1998-12-04 | 2001-01-19 | Synthelabo | Derives de 1,4-diazabicyclo[3.2.2.]nonane, leur preparation et leur application en therapeutique |
| US7265115B2 (en) * | 1999-01-29 | 2007-09-04 | Abbott Laboratories | Diazabicyclic CNS active agents |
| NZ512884A (en) | 1999-01-29 | 2004-03-26 | Abbott Lab | Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands |
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| FR2809731B1 (fr) | 2000-05-31 | 2002-07-19 | Sanofi Synthelabo | Derives de 1,4-diazabicyclo-[3.2.2] nonane-pheylisoxazole, leur preparation et leur application en therapeutique |
| FR2809732B1 (fr) | 2000-05-31 | 2002-07-19 | Sanofi Synthelabo | DERIVES DE 4(-2-PHENYLTHIAZOL-5-yl)-1,4-DIAZABICYCLO-[3.2.2] NONANE, LEUR PREPARATION ET LEUR APPLICATION ENTHERAPEUTIQUE |
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| FR2832712B1 (fr) | 2001-11-23 | 2004-02-13 | Sanofi Synthelabo | Derives de 4-(oxadiazol-3-yl)-1,4-diazabicyclo[3.2.2]nonane, leur preparation et leur application en therapeutique |
| CN1653068A (zh) * | 2002-05-07 | 2005-08-10 | 神经研究公司 | 新的二氮杂双环联芳基衍生物 |
| WO2004043960A1 (en) | 2002-11-11 | 2004-05-27 | Neurosearch A/S | 1,4-diazabicyclo (3,2,2)nonane derivatives, preparation and therapeutical use thereof |
| US7399765B2 (en) * | 2003-09-19 | 2008-07-15 | Abbott Laboratories | Substituted diazabicycloalkane derivatives |
| MXPA06005019A (es) * | 2003-11-03 | 2006-07-06 | Warner Lambert Co | Nuevos inhibidores de la recaptacion de norpinefrina para el tratamiento de transtornos del sistema nervioso central. |
| CN101035792B (zh) | 2004-10-20 | 2010-09-15 | 神经研究公司 | 新颖的二氮杂双环芳基衍生物和它们的医药用途 |
| ATE422499T1 (de) | 2004-11-30 | 2009-02-15 | Neurosearch As | Neuartige diazabicyclische arylderivate als cholinerge liganden |
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| JP5052952B2 (ja) * | 2007-05-07 | 2012-10-17 | 東芝機械株式会社 | マイクロレンズ転写成形用ロールの製造方法および製造装置 |
| AR071997A1 (es) * | 2008-06-04 | 2010-07-28 | Bristol Myers Squibb Co | Forma cristalina de 6-((4s)-2-metil-4-(2-naftil)-1,2,3,4-tetrahidroisoquinolin-7-il)piridazin-3-amina |
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- 2006-12-05 KR KR1020087013706A patent/KR20080079250A/ko not_active Withdrawn
- 2006-12-05 JP JP2008543818A patent/JP2009518357A/ja not_active Abandoned
- 2006-12-05 AU AU2006323986A patent/AU2006323986A1/en not_active Abandoned
- 2006-12-05 WO PCT/EP2006/069316 patent/WO2007065892A1/en not_active Ceased
- 2006-12-05 EP EP06830366A patent/EP1963323B1/en not_active Not-in-force
- 2006-12-05 NZ NZ567048A patent/NZ567048A/en not_active IP Right Cessation
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| NZ567048A (en) | 2010-12-24 |
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| CN101305004B (zh) | 2011-11-16 |
| JP2009518357A (ja) | 2009-05-07 |
| CN101305004A (zh) | 2008-11-12 |
| WO2007065892A1 (en) | 2007-06-14 |
| US8173658B2 (en) | 2012-05-08 |
| ATE473978T1 (de) | 2010-07-15 |
| DE602006015523D1 (de) | 2010-08-26 |
| EP2246352A1 (en) | 2010-11-03 |
| EP1963323B1 (en) | 2010-07-14 |
| DK1963323T3 (da) | 2010-10-25 |
| KR20080079250A (ko) | 2008-08-29 |
| EP1963323A1 (en) | 2008-09-03 |
| RU2008110911A (ru) | 2010-01-20 |
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