BRPI0417739A - (s)-2-n-propilamino-5-hidroxitetralina como um agonista d3 - Google Patents

(s)-2-n-propilamino-5-hidroxitetralina como um agonista d3

Info

Publication number
BRPI0417739A
BRPI0417739A BRPI0417739-8A BRPI0417739A BRPI0417739A BR PI0417739 A BRPI0417739 A BR PI0417739A BR PI0417739 A BRPI0417739 A BR PI0417739A BR PI0417739 A BRPI0417739 A BR PI0417739A
Authority
BR
Brazil
Prior art keywords
propylamino
hydroxytetraline
agonist
hydroxitetraline
dopa
Prior art date
Application number
BRPI0417739-8A
Other languages
English (en)
Inventor
Dieter Scheller
Klaus Hansen
Original Assignee
Sanol Arznei Schwarz Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanol Arznei Schwarz Gmbh filed Critical Sanol Arznei Schwarz Gmbh
Publication of BRPI0417739A publication Critical patent/BRPI0417739A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C219/00—Compounds containing amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C219/26—Compounds containing amino and esterified hydroxy groups bound to the same carbon skeleton having esterified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/14—Drugs for genital or sexual disorders; Contraceptives for lactation disorders, e.g. galactorrhoea
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34—Tobacco-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/36—Opioid-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/33—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings
    • C07C211/34—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton
    • C07C211/38—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of rings other than six-membered aromatic rings of a saturated carbon skeleton containing condensed ring systems

Abstract

"(S)-2-N-PROPILAMINO-5-HIDROXITETRALINA COMO UM AGONISTA D3". A presente invenção refere-se a um medicamento que contém a (S)-2-N-propilamino-5-hidroxitetralina, os sais ou pró-drogas da mesma. Como um agonista D3, a (S)-2-N-propilamino-5-hidroxitetralina é adequada particularmente para o tratamento de distúrbios do movimento sensíveis à Dopa.
BRPI0417739-8A 2003-12-18 2004-12-13 (s)-2-n-propilamino-5-hidroxitetralina como um agonista d3 BRPI0417739A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10359528A DE10359528A1 (de) 2003-12-18 2003-12-18 (S)-2-N-Propylamino-5-hydroxytetralin als D3-agonistisches Therapeutikum
PCT/EP2004/014143 WO2005058296A1 (de) 2003-12-18 2004-12-13 (s)-2-n-propylamino-5-hydroxytetralin als d3-agonistisches therapeutikum

Publications (1)

Publication Number Publication Date
BRPI0417739A true BRPI0417739A (pt) 2007-04-03

Family

ID=34683532

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0417739-8A BRPI0417739A (pt) 2003-12-18 2004-12-13 (s)-2-n-propilamino-5-hidroxitetralina como um agonista d3

Country Status (22)

Country Link
US (2) US8609641B2 (pt)
EP (1) EP1694318B1 (pt)
JP (1) JP5253737B2 (pt)
KR (1) KR101083568B1 (pt)
CN (1) CN1929829B (pt)
AT (1) ATE356621T1 (pt)
AU (1) AU2004298341B2 (pt)
BR (1) BRPI0417739A (pt)
CA (1) CA2547820C (pt)
CY (1) CY1106589T1 (pt)
DE (2) DE10359528A1 (pt)
DK (1) DK1694318T3 (pt)
ES (1) ES2282923T3 (pt)
HK (1) HK1094421A1 (pt)
HR (1) HRP20070175T3 (pt)
IS (1) IS2533B (pt)
MX (1) MXPA06006696A (pt)
PL (1) PL1694318T3 (pt)
PT (1) PT1694318E (pt)
RS (1) RS50536B (pt)
SI (1) SI1694318T1 (pt)
WO (1) WO2005058296A1 (pt)

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EP1987815A1 (en) 2007-05-04 2008-11-05 Schwarz Pharma Ag Oronasopharyngeally deliverable pharmaceutical compositions of dopamine agonists for the prevention and/or treatment of restless limb disorders
CN101970422B (zh) 2007-11-28 2014-10-22 Ucb制药有限公司 罗替高汀的多晶型物
EP2281559A1 (en) 2009-06-26 2011-02-09 UCB Pharma GmbH Pharmaceutical composition comprising rotigotine salts (acid or Na), especially for iontophoresis
ME03053B (me) 2009-12-22 2018-10-20 Ucb Biopharma Sprl Polivinilpirolidon za stabilizaciju čvrste disperzije nekristalnog oblika rotigotina

Also Published As

Publication number Publication date
IS2533B (is) 2009-07-15
IS8505A (is) 2006-06-12
SI1694318T1 (sl) 2007-08-31
PT1694318E (pt) 2007-05-31
CN1929829B (zh) 2010-12-15
US20140051768A1 (en) 2014-02-20
CY1106589T1 (el) 2012-01-25
EP1694318B1 (de) 2007-03-14
JP2007514674A (ja) 2007-06-07
DK1694318T3 (da) 2007-06-25
ES2282923T3 (es) 2007-10-16
PL1694318T3 (pl) 2007-07-31
AU2004298341B2 (en) 2011-03-10
HRP20070175T3 (en) 2007-06-30
ATE356621T1 (de) 2007-04-15
KR20060126500A (ko) 2006-12-07
HK1094421A1 (en) 2007-03-30
RS50536B (sr) 2010-05-07
WO2005058296A1 (de) 2005-06-30
AU2004298341A1 (en) 2005-06-30
US9108900B2 (en) 2015-08-18
US20070197480A1 (en) 2007-08-23
DE10359528A1 (de) 2005-07-28
KR101083568B1 (ko) 2011-11-14
DE502004003249D1 (en) 2007-04-26
US8609641B2 (en) 2013-12-17
CN1929829A (zh) 2007-03-14
EP1694318A1 (de) 2006-08-30
CA2547820C (en) 2013-02-19
JP5253737B2 (ja) 2013-07-31
MXPA06006696A (es) 2006-08-31
CA2547820A1 (en) 2005-06-30

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