BRPI0411921A - processo para preparar intermediários úteis para preparar determinadas hidroxilaminas de n-formila antibacterianas - Google Patents
processo para preparar intermediários úteis para preparar determinadas hidroxilaminas de n-formila antibacterianasInfo
- Publication number
- BRPI0411921A BRPI0411921A BRPI0411921-5A BRPI0411921A BRPI0411921A BR PI0411921 A BRPI0411921 A BR PI0411921A BR PI0411921 A BRPI0411921 A BR PI0411921A BR PI0411921 A BRPI0411921 A BR PI0411921A
- Authority
- BR
- Brazil
- Prior art keywords
- preparing
- certain antibacterial
- intermediates useful
- formyl
- hydroxylamines
- Prior art date
Links
- 230000000844 anti-bacterial effect Effects 0.000 title abstract 3
- 238000004519 manufacturing process Methods 0.000 title abstract 3
- 239000000543 intermediate Substances 0.000 title abstract 2
- KDGKTJGPFXIBEB-UHFFFAOYSA-N n-hydroxyformamide Chemical class ONC=O KDGKTJGPFXIBEB-UHFFFAOYSA-N 0.000 abstract 1
- 239000000081 peptide deformylase inhibitor Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C239/00—Compounds containing nitrogen-to-halogen bonds; Hydroxylamino compounds or ethers or esters thereof
- C07C239/08—Hydroxylamino compounds or their ethers or esters
- C07C239/20—Hydroxylamino compounds or their ethers or esters having oxygen atoms of hydroxylamino groups etherified
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
- C07C259/04—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
- C07C259/06—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to hydrogen atoms or to acyclic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- C07D263/26—Oxygen atoms attached in position 2 with hetero atoms or acyl radicals directly attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
- C07F7/1872—Preparation; Treatments not provided for in C07F7/20
- C07F7/1892—Preparation; Treatments not provided for in C07F7/20 by reactions not provided for in C07F7/1876 - C07F7/1888
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
"PROCESSO PARA PREPARAR INTERMEDIáRIOS úTEIS PARA PREPARAR DETERMINADAS HIDROXILAMINAS DE NFORMILA ANTIBACTERIANAS". A presente invenção refere-se a um processo para preparar intermediários que são úteis para preparar determinados compostos de hidroxilamina de N-formila antibacterianos, que são inibidores de deformilase de peptídeos.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US48268603P | 2003-06-26 | 2003-06-26 | |
PCT/EP2004/006915 WO2005000835A1 (en) | 2003-06-26 | 2004-06-25 | Process for preparing intermediates useful to prepare certain antibacterial n-formyl hydroxylamines |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0411921A true BRPI0411921A (pt) | 2006-08-15 |
Family
ID=33552002
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0411921-5A BRPI0411921A (pt) | 2003-06-26 | 2004-06-25 | processo para preparar intermediários úteis para preparar determinadas hidroxilaminas de n-formila antibacterianas |
Country Status (11)
Country | Link |
---|---|
US (2) | US20070060753A1 (pt) |
EP (1) | EP1641778A1 (pt) |
JP (1) | JP2009513485A (pt) |
KR (1) | KR20060026445A (pt) |
CN (1) | CN100410251C (pt) |
AU (2) | AU2004251876A1 (pt) |
BR (1) | BRPI0411921A (pt) |
CA (1) | CA2530142A1 (pt) |
IL (1) | IL172681A0 (pt) |
MX (1) | MXPA05014217A (pt) |
WO (1) | WO2005000835A1 (pt) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE360014T1 (de) | 2001-06-15 | 2007-05-15 | Vicuron Pharm Inc | Bicyclische pyrrolidinverbindungen |
KR20050057429A (ko) | 2002-09-19 | 2005-06-16 | 노파르티스 아게 | 중간체의 제조 방법 |
AU2004216178B2 (en) | 2003-02-21 | 2008-07-03 | Novartis Ag | Chemical process for the preparation of intermediates to obtain N-formyl hydroxylamine compounds |
GT200600196A (es) * | 2005-05-23 | 2007-01-15 | Compuestos n-formil de hidroxilamina | |
US11174288B2 (en) | 2016-12-06 | 2021-11-16 | Northeastern University | Heparin-binding cationic peptide self-assembling peptide amphiphiles useful against drug-resistant bacteria |
CN112538058B (zh) * | 2020-12-26 | 2022-05-27 | 温州大学新材料与产业技术研究院 | 含恶唑环砜类化合物的制备方法 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4613676A (en) * | 1983-11-23 | 1986-09-23 | Ciba-Geigy Corporation | Substituted 5-amino-4-hydroxyvaleryl derivatives |
ATE189814T1 (de) * | 1996-04-15 | 2000-03-15 | Takeda Chemical Industries Ltd | Hydroxypyridin-derivate, ihre herstellung und ihre pharmazeutische verwendung |
JP2002502815A (ja) * | 1998-02-07 | 2002-01-29 | ブリティッシュ バイオテック ファーマシューティカルズ リミテッド | 抗菌剤 |
GB9907055D0 (en) * | 1999-03-29 | 1999-05-19 | British Biotech Pharm | Antibacterial agents |
AR036053A1 (es) * | 2001-06-15 | 2004-08-04 | Versicor Inc | Compuestos de n-formil-hidroxilamina, un proceso para su preparacion y composiciones farmaceuticas |
-
2004
- 2004-06-25 CA CA002530142A patent/CA2530142A1/en not_active Abandoned
- 2004-06-25 EP EP04740324A patent/EP1641778A1/en not_active Withdrawn
- 2004-06-25 JP JP2006516061A patent/JP2009513485A/ja active Pending
- 2004-06-25 CN CNB2004800214382A patent/CN100410251C/zh not_active Expired - Fee Related
- 2004-06-25 KR KR1020057024908A patent/KR20060026445A/ko not_active Application Discontinuation
- 2004-06-25 WO PCT/EP2004/006915 patent/WO2005000835A1/en active Application Filing
- 2004-06-25 BR BRPI0411921-5A patent/BRPI0411921A/pt not_active IP Right Cessation
- 2004-06-25 AU AU2004251876A patent/AU2004251876A1/en not_active Abandoned
- 2004-06-25 US US10/561,754 patent/US20070060753A1/en not_active Abandoned
- 2004-06-25 MX MXPA05014217A patent/MXPA05014217A/es unknown
-
2005
- 2005-12-19 IL IL172681A patent/IL172681A0/en unknown
-
2008
- 2008-11-03 US US12/263,992 patent/US20090118515A1/en not_active Abandoned
-
2009
- 2009-03-13 AU AU2009201025A patent/AU2009201025A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP1641778A1 (en) | 2006-04-05 |
IL172681A0 (en) | 2006-04-10 |
KR20060026445A (ko) | 2006-03-23 |
JP2009513485A (ja) | 2009-04-02 |
US20090118515A1 (en) | 2009-05-07 |
CA2530142A1 (en) | 2005-01-06 |
US20070060753A1 (en) | 2007-03-15 |
CN100410251C (zh) | 2008-08-13 |
CN1829710A (zh) | 2006-09-06 |
AU2009201025A1 (en) | 2009-04-02 |
AU2004251876A1 (en) | 2005-01-06 |
MXPA05014217A (es) | 2006-03-09 |
WO2005000835A1 (en) | 2005-01-06 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE 7A. ANUIDADE(S). |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE A 7A ANUIDADE. |