BR9910696A - Composições farmacêuticas - Google Patents

Composições farmacêuticas

Info

Publication number
BR9910696A
BR9910696A BR9910696-5A BR9910696A BR9910696A BR 9910696 A BR9910696 A BR 9910696A BR 9910696 A BR9910696 A BR 9910696A BR 9910696 A BR9910696 A BR 9910696A
Authority
BR
Brazil
Prior art keywords
pharmaceutical compositions
piperidine
asthma
antagonist
acyl
Prior art date
Application number
BR9910696-5A
Other languages
English (en)
Inventor
Steffen Lang
Kurt Liechti
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9811200.6A external-priority patent/GB9811200D0/en
Priority claimed from GBGB9818105.0A external-priority patent/GB9818105D0/en
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR9910696A publication Critical patent/BR9910696A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds

Abstract

Patente de Invenção: <B>"COMPOSIçõES FARMACêUTICAS"<D>. Composições farmacêuticas espontaneamente dispersáveis compreendendo uma piperidina, por exemplo, Antagonista de Substância P de 1-acil-piperidina e seu uso no tratamento de distúrbios de SNC, por exemplo, depressão e fobia social e doenças respiratórias, por exemplo, asma e bronquite crónica.
BR9910696-5A 1998-05-26 1999-05-26 Composições farmacêuticas BR9910696A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9811200.6A GB9811200D0 (en) 1998-05-26 1998-05-26 Organic compounds
GBGB9818105.0A GB9818105D0 (en) 1998-08-19 1998-08-19 Organic compounds
PCT/EP1999/003623 WO1999061025A1 (en) 1998-05-26 1999-05-26 Microemulsion preconcentrates containing a piperidine substance p antagonist

Publications (1)

Publication Number Publication Date
BR9910696A true BR9910696A (pt) 2001-01-30

Family

ID=26313736

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9910696-5A BR9910696A (pt) 1998-05-26 1999-05-26 Composições farmacêuticas

Country Status (31)

Country Link
US (2) US20020156099A1 (pt)
EP (1) EP1082119B1 (pt)
JP (1) JP4083985B2 (pt)
KR (1) KR20010043669A (pt)
CN (1) CN1270714C (pt)
AR (1) AR018376A1 (pt)
AT (1) ATE257380T1 (pt)
AU (1) AU755134B2 (pt)
BE (1) BE1012143A5 (pt)
BR (1) BR9910696A (pt)
CA (1) CA2333154C (pt)
DE (2) DE69914077T2 (pt)
DK (1) DK1082119T3 (pt)
ES (1) ES2214859T3 (pt)
FR (1) FR2779145B1 (pt)
GB (1) GB2353473A (pt)
HK (1) HK1035137A1 (pt)
HU (1) HUP0102202A3 (pt)
ID (1) ID27096A (pt)
IL (1) IL139501A0 (pt)
IT (1) IT1313551B1 (pt)
NO (1) NO20005920L (pt)
NZ (1) NZ508325A (pt)
PE (1) PE20000537A1 (pt)
PL (1) PL344245A1 (pt)
PT (1) PT1082119E (pt)
RU (1) RU2240121C2 (pt)
SK (1) SK17752000A3 (pt)
TR (1) TR200003502T2 (pt)
TW (1) TW537894B (pt)
WO (1) WO1999061025A1 (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW537894B (en) 1998-05-26 2003-06-21 Novartis Ag A spontaneously dispersible pharmaceutical composition comprising a piperidine substance P antagonist
AU2003225260A1 (en) * 2002-04-22 2003-11-03 University Of Florida Microemulsions for selective molecular separation
GB0220953D0 (en) 2002-09-10 2002-10-23 Novartis Ag Organic compounds
US7842791B2 (en) 2002-12-19 2010-11-30 Nancy Jean Britten Dispersible pharmaceutical compositions
FR2934953B1 (fr) 2008-08-14 2011-01-21 Commissariat Energie Atomique Nanoemulsions de nanocristaux
FR2934955B1 (fr) 2008-08-14 2011-07-08 Commissariat Energie Atomique Encapsulation d'agents therapeutiques lipophiles ou amphiphiles dans des nanoemulsions
FR2935001B1 (fr) * 2008-08-14 2011-12-30 Commissariat Energie Atomique Emulsion fluorescente
FR2934954B1 (fr) 2008-08-14 2011-07-22 Commissariat Energie Atomique Emulsion fluorescente de vert d'indocyanine
WO2014106048A2 (en) * 2012-12-31 2014-07-03 Jrx Biotechnology, Inc. Liquid topical pharmaceutical nano-emulsion formulations

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3305689A1 (de) 1983-02-18 1984-08-23 Mack Chem Pharm Pharmazeutische zubereitung mit retardwirkung
US5342625A (en) * 1988-09-16 1994-08-30 Sandoz Ltd. Pharmaceutical compositions comprising cyclosporins
MY110227A (en) 1991-08-12 1998-03-31 Ciba Geigy Ag 1-acylpiperindine compounds.
DE4220616C2 (de) 1992-06-24 1994-12-22 Byk Gulden Lomberg Chem Fab Dexniguldipin zur intravenösen Verabreichung
ES2168271T3 (es) 1992-09-25 2002-06-16 Novartis Ag Composiciones farmaceuticas que contienen ciclosporinas.
GB2278780B (en) * 1993-05-27 1998-10-14 Sandoz Ltd Macrolide formulations
US5952004A (en) * 1994-03-18 1999-09-14 Shire Laboratories Inc. Emulsified drug delivery systems
TW397825B (en) * 1994-10-14 2000-07-11 Novartis Ag Aroyl-piperidine derivatives
GB2308545B (en) 1994-10-26 1999-06-02 Novartis Ag Pharmaceutical microemulsion preconcentrates
FR2728169A1 (fr) 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des prurits et des dysesthesies oculaires ou palpebrales
FR2728165A1 (fr) * 1994-12-19 1996-06-21 Oreal Utilisation d'un antagoniste de substance p pour le traitement des rougeurs cutanees d'origine neurogene
AU696948B2 (en) * 1995-03-27 1998-09-24 Hisamitsu Pharmaceutical Co., Inc. Piperidine derivatives
NZ280689A (en) 1995-12-15 1997-08-22 Bernard Charles Sherma Sherman Pharmaceutical composition comprising a cyclosporipharmaceutical composition comprising a cyclosporin; a tocol, tocopherol or tocotrienol; and propylen; a tocol, tocopherol or tocotrienol; and propylene carbonate or polyethylene glycol ne carbonate or polyethylene glycol
GB9601120D0 (en) 1996-01-19 1996-03-20 Sandoz Ltd Organic compounds
WO1997045119A1 (en) 1996-05-24 1997-12-04 Novartis Ag Use of substance p antagonists for treating social phobia
TW537894B (en) 1998-05-26 2003-06-21 Novartis Ag A spontaneously dispersible pharmaceutical composition comprising a piperidine substance P antagonist

Also Published As

Publication number Publication date
PL344245A1 (en) 2001-10-08
WO1999061025A1 (en) 1999-12-02
TW537894B (en) 2003-06-21
NZ508325A (en) 2003-06-30
IT1313551B1 (it) 2002-09-09
ITMI991164A1 (it) 2000-11-26
CA2333154C (en) 2008-07-08
EP1082119B1 (en) 2004-01-07
PE20000537A1 (es) 2000-07-10
HUP0102202A3 (en) 2003-01-28
DE19983247T1 (de) 2001-05-31
AR018376A1 (es) 2001-11-14
DE69914077T2 (de) 2004-06-09
RU2240121C2 (ru) 2004-11-20
AU755134B2 (en) 2002-12-05
EP1082119A1 (en) 2001-03-14
ID27096A (id) 2001-03-01
HK1035137A1 (en) 2001-11-16
GB0028506D0 (en) 2001-01-10
JP2002516280A (ja) 2002-06-04
US20030152626A1 (en) 2003-08-14
US6949257B2 (en) 2005-09-27
DE69914077D1 (de) 2004-02-12
US20020156099A1 (en) 2002-10-24
HUP0102202A2 (hu) 2001-11-28
PT1082119E (pt) 2004-05-31
CA2333154A1 (en) 1999-12-02
GB2353473A (en) 2001-02-28
AU4500899A (en) 1999-12-13
CN1303285A (zh) 2001-07-11
TR200003502T2 (tr) 2001-04-20
KR20010043669A (ko) 2001-05-25
NO20005920D0 (no) 2000-11-23
FR2779145B1 (fr) 2004-07-30
ATE257380T1 (de) 2004-01-15
FR2779145A1 (fr) 1999-12-03
SK17752000A3 (sk) 2001-05-10
CN1270714C (zh) 2006-08-23
BE1012143A5 (fr) 2000-05-02
ES2214859T3 (es) 2004-09-16
JP4083985B2 (ja) 2008-04-30
DK1082119T3 (da) 2004-04-13
IL139501A0 (en) 2001-11-25
NO20005920L (no) 2001-01-25

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: ALTERADA DE INT.CL.8: A61K 9/107, A61K 9/48, A61K 31/4709, A61K 47/10, A61K 47/14, A61K 47/44, A61P 11/00, A61P 11/06, A61P 25/00, A61P 25/22, A61P 25/24, A61P 25/28, A61P 37/08, A61P 43/00

Ipc: A61K 9/107 (2008.01), A61K 9/48 (2008.01), A61K 31

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFERIMENTO DO PRESENTE PEDIDO, UMA VEZ QUE A MATERIA PLEITEADA NAO APRESENTA ATIVIDADE INVENTIVA CONFORME O ART. 13 DA LPI ( LEI 9279/96 ), NAO SENDO MATERIA PATENTEAVEL CONFORME O ART. 8O DA LPI ( LEI 9279/96

B12B Appeal against refusal [chapter 12.2 patent gazette]