BR9815670A - Compostos agonistas de exendina - Google Patents

Compostos agonistas de exendina

Info

Publication number
BR9815670A
BR9815670A BR9815670-5A BR9815670A BR9815670A BR 9815670 A BR9815670 A BR 9815670A BR 9815670 A BR9815670 A BR 9815670A BR 9815670 A BR9815670 A BR 9815670A
Authority
BR
Brazil
Prior art keywords
exendin agonist
agonist compounds
compounds
benefited
delaying
Prior art date
Application number
BR9815670-5A
Other languages
English (en)
Inventor
Nigel Robert Arnold Beeley
Kathryn S Prickett
Original Assignee
Amylin Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22062753&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9815670(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Amylin Pharmaceuticals Inc filed Critical Amylin Pharmaceuticals Inc
Publication of BR9815670A publication Critical patent/BR9815670A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/57563—Vasoactive intestinal peptide [VIP]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Vascular Medicine (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Patente de Invenção: <B>"COMPOSTOS AGONISTAS DE EXENDINA"<D>. A presente invenção refere-se a novos compostos que têm a atividade como agonistas de exendina. Estes compostos são úteis no tratamento da diabetes Tipo I e II, em tratamento de distúrbio que seriam beneficiados por agentes que reduzem os níveis de glicose de plasma e em tratamento de distúrbios que seriam beneficiados com agentes úteis para impedir e/ou retardar o esvaziamento gástrico. A presente invenção refere-se ainda a composição farmacêuticas compreendendo os referidos novos compostos e a métodos para o tratamento de diabetes melito.
BR9815670-5A 1997-11-14 1998-11-13 Compostos agonistas de exendina BR9815670A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6544297P 1997-11-14 1997-11-14
PCT/US1998/024210 WO1999025727A2 (en) 1997-11-14 1998-11-13 Novel exendin agonist compounds

Publications (1)

Publication Number Publication Date
BR9815670A true BR9815670A (pt) 2000-10-17

Family

ID=22062753

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9815670-5A BR9815670A (pt) 1997-11-14 1998-11-13 Compostos agonistas de exendina

Country Status (12)

Country Link
US (1) US7696161B2 (pt)
EP (1) EP1066314B1 (pt)
JP (1) JP2003522721A (pt)
AT (1) ATE381939T1 (pt)
AU (1) AU757748B2 (pt)
BR (1) BR9815670A (pt)
CA (1) CA2310097C (pt)
DE (1) DE69838916T2 (pt)
ES (1) ES2294822T3 (pt)
MX (1) MXPA00004670A (pt)
NZ (1) NZ504258A (pt)
WO (1) WO1999025727A2 (pt)

Families Citing this family (124)

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EP1066314A4 (en) 2002-04-10
EP1066314A1 (en) 2001-01-10
EP1066314B1 (en) 2007-12-26
DE69838916D1 (de) 2008-02-07
ATE381939T1 (de) 2008-01-15
WO1999025727A2 (en) 1999-05-27
DE69838916T2 (de) 2008-12-18
CA2310097C (en) 2014-07-29
NZ504258A (en) 2002-12-20
US20080119393A1 (en) 2008-05-22
ES2294822T3 (es) 2008-04-01
CA2310097A1 (en) 1999-05-27
AU757748B2 (en) 2003-03-06
US7696161B2 (en) 2010-04-13
AU1404699A (en) 1999-06-07
JP2003522721A (ja) 2003-07-29
MXPA00004670A (es) 2003-07-14

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