BR9813303A - Composto, processo para prepará-lo, utilização do mesmo, processos de preparação de um composto diaestereomericamente puro, e de preparação do sal deste, e, composição farmacêutica - Google Patents

Composto, processo para prepará-lo, utilização do mesmo, processos de preparação de um composto diaestereomericamente puro, e de preparação do sal deste, e, composição farmacêutica

Info

Publication number
BR9813303A
BR9813303A BR9813303-9A BR9813303A BR9813303A BR 9813303 A BR9813303 A BR 9813303A BR 9813303 A BR9813303 A BR 9813303A BR 9813303 A BR9813303 A BR 9813303A
Authority
BR
Brazil
Prior art keywords
preparing
compound
hydrogen atom
salt
processes
Prior art date
Application number
BR9813303-9A
Other languages
English (en)
Portuguese (pt)
Inventor
Patrice Mayer
Jean-Louis Vidaluc
Thierry Imbert
Marc Marien
Original Assignee
Pf Medicament
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pf Medicament filed Critical Pf Medicament
Publication of BR9813303A publication Critical patent/BR9813303A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D455/00Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/03Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/04Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine
    • C07D455/06Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine containing benzo [a] quinolizine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BR9813303-9A 1997-10-28 1998-10-26 Composto, processo para prepará-lo, utilização do mesmo, processos de preparação de um composto diaestereomericamente puro, e de preparação do sal deste, e, composição farmacêutica BR9813303A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9713499A FR2770215B1 (fr) 1997-10-28 1997-10-28 Derives d'aminomethyl-benzo[a]quinolizidine, leur preparation et leur application en therapeutique pour les maladies neurodegeneratives
PCT/FR1998/002281 WO1999021856A1 (fr) 1997-10-28 1998-10-26 Derives d'aminomethyl-benzo[a]quinolizidine, leur preparation et leur application en therapeutique pour les maladies neurodegeneratives

Publications (1)

Publication Number Publication Date
BR9813303A true BR9813303A (pt) 2000-08-29

Family

ID=9512729

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9813303-9A BR9813303A (pt) 1997-10-28 1998-10-26 Composto, processo para prepará-lo, utilização do mesmo, processos de preparação de um composto diaestereomericamente puro, e de preparação do sal deste, e, composição farmacêutica

Country Status (8)

Country Link
EP (1) EP1027350A1 (ja)
JP (1) JP2001521034A (ja)
CN (1) CN1278260A (ja)
AU (1) AU9751798A (ja)
BR (1) BR9813303A (ja)
CA (1) CA2307748A1 (ja)
FR (1) FR2770215B1 (ja)
WO (1) WO1999021856A1 (ja)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0016454D0 (en) 2000-07-04 2000-08-23 Hoffmann La Roche Thienopyrrolidinones
US8084492B2 (en) 2004-11-19 2011-12-27 The New Industry Research Organization Benzofuran compound and pharmaceutical composition containing the same
ES2525932T3 (es) * 2006-05-02 2015-01-02 The Trustees Of The University Of Pennsylvania Derivados de dihidrotetrabenazina radiomarcados y su uso como agentes de imagenología
GB2463451A (en) * 2008-09-08 2010-03-17 Cambridge Lab 3, 11b cis-dihydrotetrabenazine compounds for use in the treatment of dementia
FR2976287B1 (fr) * 2011-06-09 2013-07-05 Pf Medicament Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutique
US9115149B2 (en) * 2011-09-19 2015-08-25 Vitas Pharma Research Private Limited Heterocyclic compounds as inhibitors of fatty acid biosysnthesis for bacterial infections

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8416432D0 (en) * 1984-06-28 1984-08-01 Wyeth John & Brother Ltd Benzoquinolizines

Also Published As

Publication number Publication date
CA2307748A1 (fr) 1999-05-06
AU9751798A (en) 1999-05-17
FR2770215A1 (fr) 1999-04-30
JP2001521034A (ja) 2001-11-06
WO1999021856A1 (fr) 1999-05-06
FR2770215B1 (fr) 2000-01-14
EP1027350A1 (fr) 2000-08-16
CN1278260A (zh) 2000-12-27

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
B11Y Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired