FR2976287B1 - Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutique - Google Patents
Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutiqueInfo
- Publication number
- FR2976287B1 FR2976287B1 FR1155028A FR1155028A FR2976287B1 FR 2976287 B1 FR2976287 B1 FR 2976287B1 FR 1155028 A FR1155028 A FR 1155028A FR 1155028 A FR1155028 A FR 1155028A FR 2976287 B1 FR2976287 B1 FR 2976287B1
- Authority
- FR
- France
- Prior art keywords
- benzoquinolizidine
- derivatives
- preparation
- therapeutic applications
- therapeutic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/03—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/04—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine
- C07D455/06—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine containing benzo [a] quinolizine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Priority Applications (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR1155028A FR2976287B1 (fr) | 2011-06-09 | 2011-06-09 | Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutique |
EP12729076.5A EP2718291A1 (fr) | 2011-06-09 | 2012-06-07 | Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutique |
PCT/EP2012/060805 WO2012168368A1 (fr) | 2011-06-09 | 2012-06-07 | Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutique |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR1155028A FR2976287B1 (fr) | 2011-06-09 | 2011-06-09 | Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2976287A1 FR2976287A1 (fr) | 2012-12-14 |
FR2976287B1 true FR2976287B1 (fr) | 2013-07-05 |
Family
ID=46331276
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR1155028A Expired - Fee Related FR2976287B1 (fr) | 2011-06-09 | 2011-06-09 | Derives benzoquinolizidines, leur procede de preparation et leurs applications en therapeutique |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP2718291A1 (fr) |
FR (1) | FR2976287B1 (fr) |
WO (1) | WO2012168368A1 (fr) |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4686226A (en) * | 1985-09-03 | 1987-08-11 | Merck & Co., Inc. | Substituted benzo[b]furo- and benzo[b]thieno quinolizines |
FR2770215B1 (fr) * | 1997-10-28 | 2000-01-14 | Pf Medicament | Derives d'aminomethyl-benzo[a]quinolizidine, leur preparation et leur application en therapeutique pour les maladies neurodegeneratives |
KR20040038899A (ko) * | 2001-09-28 | 2004-05-08 | 교와 핫꼬 고교 가부시끼가이샤 | 수용체 길항제 |
AR052342A1 (es) | 2004-12-21 | 2007-03-14 | Janssen Pharmaceutica Nv | Derivados sustituidos de triazolona,tetrazolona e imidazolona con actividad selectiva antagonista de alfa2c-adenoreceptores |
CA2649707A1 (fr) | 2006-05-22 | 2007-11-29 | Janssen Pharmaceutica N.V. | Derives de pyrazinone substitues a utiliser comme medicament |
WO2008043775A1 (fr) | 2006-10-12 | 2008-04-17 | Janssen Pharmaceutica Nv | Dérivés de pyrazinone substitués pour une utilisation en tant que médicament |
-
2011
- 2011-06-09 FR FR1155028A patent/FR2976287B1/fr not_active Expired - Fee Related
-
2012
- 2012-06-07 WO PCT/EP2012/060805 patent/WO2012168368A1/fr active Application Filing
- 2012-06-07 EP EP12729076.5A patent/EP2718291A1/fr not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
EP2718291A1 (fr) | 2014-04-16 |
FR2976287A1 (fr) | 2012-12-14 |
WO2012168368A1 (fr) | 2012-12-13 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PLFP | Fee payment |
Year of fee payment: 6 |
|
ST | Notification of lapse |
Effective date: 20180228 |