PT82682B - Processo para a preparacao de derivados da quinazolina e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de derivados da quinazolina e de composicoes farmaceuticas que os contem

Info

Publication number
PT82682B
PT82682B PT82682A PT8268286A PT82682B PT 82682 B PT82682 B PT 82682B PT 82682 A PT82682 A PT 82682A PT 8268286 A PT8268286 A PT 8268286A PT 82682 B PT82682 B PT 82682B
Authority
PT
Portugal
Prior art keywords
group
heteroatom
quinazoline derivatives
preparation
pharmaceutical compositions
Prior art date
Application number
PT82682A
Other languages
English (en)
Other versions
PT82682A (en
Original Assignee
Nat Res Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nat Res Dev filed Critical Nat Res Dev
Publication of PT82682A publication Critical patent/PT82682A/pt
Publication of PT82682B publication Critical patent/PT82682B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
PT82682A 1985-05-31 1986-05-30 Processo para a preparacao de derivados da quinazolina e de composicoes farmaceuticas que os contem PT82682B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB858513754A GB8513754D0 (en) 1985-05-31 1985-05-31 Anti-cancer quinazoline derivatives

Publications (2)

Publication Number Publication Date
PT82682A PT82682A (en) 1986-06-01
PT82682B true PT82682B (pt) 1988-03-03

Family

ID=10579966

Family Applications (1)

Application Number Title Priority Date Filing Date
PT82682A PT82682B (pt) 1985-05-31 1986-05-30 Processo para a preparacao de derivados da quinazolina e de composicoes farmaceuticas que os contem

Country Status (17)

Country Link
US (1) US5236927A (pt)
EP (1) EP0204529B1 (pt)
JP (1) JPS61282368A (pt)
AT (1) ATE87621T1 (pt)
AU (1) AU592271B2 (pt)
DE (1) DE3688150T2 (pt)
DK (1) DK255786A (pt)
ES (1) ES8800911A1 (pt)
FI (1) FI862303A (pt)
GB (2) GB8513754D0 (pt)
GR (1) GR861418B (pt)
HU (1) HUT45512A (pt)
IL (1) IL78910A0 (pt)
NO (1) NO862170L (pt)
NZ (1) NZ216363A (pt)
PT (1) PT82682B (pt)
ZA (1) ZA864051B (pt)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8607683D0 (en) * 1986-03-27 1986-04-30 Ici Plc Anti-tumor agents
GB8707053D0 (en) * 1987-03-25 1987-04-29 Ici Plc Anti-tumour agents
US4857530A (en) * 1987-11-03 1989-08-15 Warner-Lambert Company Substituted quinazolinones as anticancer agents
GB8809978D0 (en) * 1988-04-27 1988-06-02 Ici Plc Anti-tumour agents
EP0365763A1 (en) * 1988-09-30 1990-05-02 Agouron Pharmaceuticals, Inc. Antiproliferative cyclic compounds
US5286726A (en) * 1990-04-12 1994-02-15 The Regents Of The University Of Michigan Difluoroglutamic acid conjugates with folates and anti-folates for the treatment of neoplastic diseases
US6762188B1 (en) 1990-06-19 2004-07-13 Smithkline Beecham Corporation Pharmaceutically active benzoquinazoline compounds
GB9013615D0 (en) * 1990-06-19 1990-08-08 Wellcome Found Pharmaceutical compounds
GB9105771D0 (en) * 1991-03-19 1991-05-01 Cancer Res Inst Royal Anti-cancer compounds
GB9205320D0 (en) * 1992-03-11 1992-04-22 Ici Plc Anti-tumour compounds
GB9205907D0 (en) * 1992-03-18 1992-04-29 Cancer Res Inst Royal Anti-cancer compounds
US5430148A (en) * 1992-03-31 1995-07-04 Agouron Pharmaceuticals, Inc. Antiproliferative quinazolines
GB9223352D0 (en) * 1992-11-06 1992-12-23 Ici Plc Tricyclic compounds
US7262058B2 (en) * 2001-03-09 2007-08-28 Nonda Katopodis Method for determining lipid associated sialoprotein in body fluids
KR20050061545A (ko) * 2002-10-18 2005-06-22 코닌클리케 필립스 일렉트로닉스 엔.브이. Ｔｖ-애니타임의 메타데이터 보호를 위한 방법 및 시스템
CA2502302A1 (en) * 2002-11-04 2004-05-21 Nps Pharmaceuticals, Inc. Quinazolinone compounds as calcilytics
MX2008000744A (es) * 2005-07-15 2008-03-10 Schering Corp Derivados de quinazolina utiles en el tratamiento del cancer.
CA2615380A1 (en) * 2005-07-15 2007-01-25 Schering Corporation Quinazoline derivatives useful in cancer treatment
AU2007303846B2 (en) 2006-10-04 2011-03-10 Pfizer Products Inc. Pyrido[4,3-d]pyrimidin-4(3H)-one derivatives as calcium receptor antagonists
JP5535925B2 (ja) 2007-10-26 2014-07-02 ザ リージェンツ オブ ザ ユニバーシティ オブ カリフォルニア アンドロゲン受容体調節物質としてのジアリールヒダントイン化合物
LT2445502T (lt) * 2009-06-25 2017-09-25 Alkermes Pharma Ireland Limited Heterocikliniai junginiai, skirti neurologinių ir fiziologinių susirgimų gydymui
ES2647361T3 (es) * 2010-01-07 2017-12-21 Alkermes Pharma Ireland Limited Profármacos de sales de amonio cuaternario
AU2011270701B2 (en) 2010-06-24 2015-05-14 Alkermes Pharma Ireland Limited Prodrugs of NH-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives
CA2830511C (en) 2011-03-18 2021-09-14 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising aripiprazole lauroxil and sorbitan laurate
US9999670B2 (en) 2012-03-19 2018-06-19 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising benzyl alcohol
CA2867121C (en) 2012-03-19 2021-05-25 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty acid esters
US9993556B2 (en) 2012-03-19 2018-06-12 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty glycerol esters
EP3718536A1 (en) 2012-09-19 2020-10-07 Alkermes Pharma Ireland Limited Pharmaceutical compositions having improved storage stability
MA39495A (fr) 2014-03-20 2015-09-24 Alkermes Pharma Ireland Ltd Formulations d'aripiprazole présentant des vitesses d'injection plus élevées
EP3761983A1 (en) 2018-03-05 2021-01-13 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy
WO2024028999A1 (ja) * 2022-08-03 2024-02-08 Ils株式会社 Ｎ－［４－メチルアミノベンゾイル］－ｌ－グルタミン酸ジエチルエステルの製造方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1021196A (en) * 1964-02-20 1966-03-02 Parke Davis & Co Novel amino acids and means for producing the same
US3471498A (en) * 1967-08-11 1969-10-07 Parke Davis & Co Certain n-p-((2,4-diamino-6-quinazolinyl)-methyl)benzoylamino acids
GB2065653B (en) 1979-12-19 1983-03-09 Nat Res Dev Anti-cancer quinazoline derivatives
GB8607683D0 (en) * 1986-03-27 1986-04-30 Ici Plc Anti-tumor agents

Also Published As

Publication number Publication date
ES555548A0 (es) 1987-12-01
ATE87621T1 (de) 1993-04-15
DK255786A (da) 1986-12-01
GB8513754D0 (en) 1985-07-03
JPS61282368A (ja) 1986-12-12
ES8800911A1 (es) 1987-12-01
NO862170L (no) 1986-12-01
GR861418B (en) 1986-09-26
EP0204529A2 (en) 1986-12-10
IL78910A0 (en) 1986-09-30
PT82682A (en) 1986-06-01
EP0204529A3 (en) 1987-11-19
AU5822086A (en) 1986-12-04
AU592271B2 (en) 1990-01-04
DK255786D0 (da) 1986-05-30
GB8613184D0 (en) 1986-07-02
FI862303A (fi) 1986-12-01
GB2175903B (en) 1988-10-12
GB2175903A (en) 1986-12-10
US5236927A (en) 1993-08-17
DE3688150D1 (de) 1993-05-06
EP0204529B1 (en) 1993-03-31
ZA864051B (en) 1987-01-28
NZ216363A (en) 1989-07-27
HUT45512A (en) 1988-07-28
DE3688150T2 (de) 1993-07-29
FI862303A0 (fi) 1986-05-30

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Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 19920329