BR9811658A - Polimorfos de 8-cloro-6,11-dihidro-11-(4-piperidilideno)-5h-benzo [5,6]-ciclo hepta[1,2-b] piridina - Google Patents

Polimorfos de 8-cloro-6,11-dihidro-11-(4-piperidilideno)-5h-benzo [5,6]-ciclo hepta[1,2-b] piridina

Info

Publication number
BR9811658A
BR9811658A BR9811658-4A BR9811658A BR9811658A BR 9811658 A BR9811658 A BR 9811658A BR 9811658 A BR9811658 A BR 9811658A BR 9811658 A BR9811658 A BR 9811658A
Authority
BR
Brazil
Prior art keywords
polymorphs
piperidylidene
benzo
dihydro
pyridine
Prior art date
Application number
BR9811658-4A
Other languages
English (en)
Portuguese (pt)
Inventor
Doris P Schumacher
Junning Lee
Lawrence R Rogers
Charles C Eckhart
Naneshwar S Sawant
Michael B Mitchell
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25389724&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9811658(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Publication of BR9811658A publication Critical patent/BR9811658A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BR9811658-4A 1997-07-02 1998-07-01 Polimorfos de 8-cloro-6,11-dihidro-11-(4-piperidilideno)-5h-benzo [5,6]-ciclo hepta[1,2-b] piridina BR9811658A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US88676697A 1997-07-02 1997-07-02
PCT/US1998/013433 WO1999001450A1 (en) 1997-07-02 1998-07-01 POLYMORPHS OF 8-CHLORO-6, 11-DIHYDRO-11- (4-PIPERIDYLIDENE) -5H-BENZO[5,6] CYCLOHEPTA[1,2-b]PYRIDINE

Publications (1)

Publication Number Publication Date
BR9811658A true BR9811658A (pt) 2000-09-05

Family

ID=25389724

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9811658-4A BR9811658A (pt) 1997-07-02 1998-07-01 Polimorfos de 8-cloro-6,11-dihidro-11-(4-piperidilideno)-5h-benzo [5,6]-ciclo hepta[1,2-b] piridina

Country Status (25)

Country Link
EP (1) EP0993455B1 (https=)
JP (2) JP2002507991A (https=)
KR (1) KR20010014316A (https=)
CN (1) CN1261886A (https=)
AR (1) AR013161A1 (https=)
AT (1) ATE239010T1 (https=)
AU (1) AU734487B2 (https=)
BR (1) BR9811658A (https=)
CA (1) CA2294352C (https=)
CO (1) CO4940423A1 (https=)
DE (1) DE69814076T2 (https=)
ES (1) ES2197480T3 (https=)
HU (1) HUP0004308A3 (https=)
IL (1) IL133387A (https=)
MY (1) MY132943A (https=)
NO (1) NO996547L (https=)
NZ (1) NZ501417A (https=)
PE (1) PE86399A1 (https=)
PL (1) PL337712A1 (https=)
RU (1) RU2197485C2 (https=)
SK (1) SK185299A3 (https=)
TR (1) TR199903308T2 (https=)
UA (1) UA62976C2 (https=)
WO (1) WO1999001450A1 (https=)
ZA (1) ZA985783B (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7405223B2 (en) 2000-02-03 2008-07-29 Schering Corporation Treating allergic and inflammatory conditions
US7678908B2 (en) * 2002-04-15 2010-03-16 Sun Pharmaceutical Industries Limited Process of preparing desaloratadine
WO2004012738A1 (en) * 2002-08-05 2004-02-12 Sandoz Ag Novel salt and polymorphs of desloratadine hemifumarate
US20060135547A1 (en) * 2003-03-12 2006-06-22 Toth Zoltan G Stable pharmaceutical compositions of desloratadine and processes for preparation of polymorphic forms of desloratadine
WO2004080461A2 (en) * 2003-03-12 2004-09-23 TEVA Gyógyszergyár Részvénytársaság Stable pharmaceutical compositions of desloratadine
SK50112007A3 (sk) * 2004-07-07 2007-07-06 Egis Gy�gyszergy�r Nyrt. Nový pseudopolymorf desloratadínu vytvorený s oxidom uhličitým
TW200735871A (en) * 2005-11-17 2007-10-01 Teva Pharma Desloratadine crystalline forms mixtures having a low level of residual solvents
HU230417B1 (hu) * 2006-10-26 2016-05-30 Egis Gyógyszergyár Zrt Eljárás desloratadine szén-dioxiddal képezett adduktjának előállítására
EP2164470A1 (en) * 2007-05-11 2010-03-24 ratiopharm GmbH Pharmaceutical composition comprising desloratadine
EP2269586B1 (en) 2009-07-01 2011-09-21 Alfred E. Tiefenbacher (GmbH & Co. KG) Pharmaceutical composition comprising desloratadine
PT2568970T (pt) 2010-05-10 2019-02-11 Lesvi Laboratorios Sl Formulações farmacêuticas estáveis contendo um anti-histamínico
EP2727592A1 (en) 2012-11-05 2014-05-07 Kücükgüzel, Sükriye Güniz A combination of desloratadine and paracetamol
CN103755682A (zh) * 2013-12-30 2014-04-30 山东达因海洋生物制药股份有限公司 一种地氯雷他定新晶型及制备方法
CN108358892A (zh) * 2018-04-11 2018-08-03 常州方圆制药有限公司 一种地氯雷他定粗品的提纯方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1985003707A1 (en) * 1984-02-15 1985-08-29 Schering Corporation 8-CHLORO-6,11-DIHYDRO-11-(4-PIPERIDYLIDENE)-5H-BENZO AD5,6 BDCYCLOHEPTA AD1,2-b BDPYRIDINE AND ITS SALTS, PROCESSES FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS
EP0208855B1 (en) * 1985-05-13 1991-03-06 Schering Corporation process for preparing piperidylidene dihydrodibenzo(a,d)cycloheptenes and aza derivatives thereof, compounds obtained by such process and the use of such compounds for preparing useful pharmaceutical compositions
IE68935B1 (en) * 1990-06-22 1996-07-24 Schering Corp Bis-benzo or benzopyrido cyclohepta piperidene piperidylidene and piperazine compounds compositions and methods of use

Also Published As

Publication number Publication date
HUP0004308A3 (en) 2004-07-28
EP0993455A1 (en) 2000-04-19
DE69814076T2 (de) 2004-02-26
SK185299A3 (en) 2000-07-11
AR013161A1 (es) 2000-12-13
PL337712A1 (en) 2000-08-28
PE86399A1 (es) 1999-10-23
ES2197480T3 (es) 2004-01-01
ATE239010T1 (de) 2003-05-15
UA62976C2 (en) 2004-01-15
HUP0004308A2 (hu) 2001-10-28
CN1261886A (zh) 2000-08-02
MY132943A (en) 2007-10-31
JP2002507991A (ja) 2002-03-12
CO4940423A1 (es) 2000-07-24
NO996547L (no) 2000-03-01
ZA985783B (en) 1999-01-19
AU8271098A (en) 1999-01-25
NZ501417A (en) 2000-10-27
NO996547D0 (no) 1999-12-29
TR199903308T2 (xx) 2000-11-21
KR20010014316A (ko) 2001-02-26
WO1999001450A1 (en) 1999-01-14
IL133387A (en) 2004-02-08
DE69814076D1 (de) 2003-06-05
HK1024687A1 (en) 2000-10-20
AU734487B2 (en) 2001-06-14
JP2009242436A (ja) 2009-10-22
IL133387A0 (en) 2001-04-30
CA2294352A1 (en) 1999-01-14
CA2294352C (en) 2008-05-06
RU2197485C2 (ru) 2003-01-27
EP0993455B1 (en) 2003-05-02

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A, 8A E 9A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1909 DE 07/08/2007.