BR9710366A - Derivados de taxane e drogas que os contêm - Google Patents

Derivados de taxane e drogas que os contêm

Info

Publication number
BR9710366A
BR9710366A BR9710366A BR9710366A BR9710366A BR 9710366 A BR9710366 A BR 9710366A BR 9710366 A BR9710366 A BR 9710366A BR 9710366 A BR9710366 A BR 9710366A BR 9710366 A BR9710366 A BR 9710366A
Authority
BR
Brazil
Prior art keywords
drugs
contain
taxane derivatives
taxane
derivatives
Prior art date
Application number
BR9710366A
Other languages
English (en)
Inventor
Hideaki Shimizu
Atsuhiro Abe
Takashi Yaegashi
Seigo Sawada
Hiroshi Nagata
Original Assignee
Yakult Honsha Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Yakult Honsha Kk filed Critical Yakult Honsha Kk
Publication of BR9710366A publication Critical patent/BR9710366A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
BR9710366A 1996-07-15 1997-07-14 Derivados de taxane e drogas que os contêm BR9710366A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP18474296 1996-07-15
JP18474196 1996-07-15
PCT/JP1997/002431 WO1998002426A1 (fr) 1996-07-15 1997-07-14 Derives de taxane et medicaments les contenant

Publications (1)

Publication Number Publication Date
BR9710366A true BR9710366A (pt) 1999-08-17

Family

ID=26502676

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9710366A BR9710366A (pt) 1996-07-15 1997-07-14 Derivados de taxane e drogas que os contêm

Country Status (9)

Country Link
US (1) US6025385A (pt)
EP (1) EP0930309A4 (pt)
JP (1) JP3942197B2 (pt)
KR (1) KR100476247B1 (pt)
CN (1) CN1097044C (pt)
AU (1) AU710156B2 (pt)
BR (1) BR9710366A (pt)
CA (1) CA2259977C (pt)
WO (1) WO1998002426A1 (pt)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH1192468A (ja) * 1997-09-17 1999-04-06 Yakult Honsha Co Ltd 新規なタキサン誘導体
KR100551945B1 (ko) 1997-12-19 2006-02-20 가부시키가이샤 야쿠루트 혼샤 택산 유도체
MXPA02001396A (es) * 1999-08-11 2002-08-12 Bristol & Minus Proceso para la preparacion de un analogo de carbonato de metilo del carbono 4, del paclitaxel.
HK1049787B (en) 1999-10-01 2014-07-25 Immunogen, Inc. Compositions and methods for treating cancer using immunoconjugates and chemotherapeutic agents
US6649632B2 (en) 2000-02-02 2003-11-18 Fsu Research Foundation, Inc. C10 ester substituted taxanes
WO2001057013A1 (en) * 2000-02-02 2001-08-09 Florida State University Research Foundation, Inc. Taxane formulations having improved solubility
CA2368541A1 (en) * 2000-02-02 2001-08-09 Florida State University Research Foundation, Inc. C10 carbamoyloxy substituted taxanes as antitumor agents
TR200102855T1 (tr) 2000-02-02 2002-06-21 Florida State University Research Foundation, Inc Antitümör ajanları olarak C10 karbonat ikameli taksanlar.
EP1165068B1 (en) 2000-02-02 2007-12-19 Florida State University Research Foundation, Inc. C10 heterosubstituted acetate taxanes as antitumor agents
CA2354471A1 (en) * 2001-07-31 2003-01-31 Florida State University Research Foundation, Inc. C10 ester substituted taxanes
SV2006002010A (es) 2004-02-13 2006-08-23 Univ Florida State Res Found Taxanos sustituidos con esteres de ciclopentilo en c10
EP1792927B1 (en) * 2004-09-22 2013-03-06 Nippon Kayaku Kabushiki Kaisha Novel block copolymer, micelle preparation, and anticancer agent containing the same as active ingredient
US7095150B2 (en) * 2004-10-21 2006-08-22 Shop Vac Corporation Apparatus for securing a bobbin of a reluctance machine
JP2008530122A (ja) * 2005-02-14 2008-08-07 フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド C10シクロプロピルエステル置換タキサン組成物
JP4954983B2 (ja) 2005-05-18 2012-06-20 ファーマサイエンス・インコーポレイテッド Birドメイン結合化合物
KR20080106254A (ko) 2006-03-28 2008-12-04 니폰 가야꾸 가부시끼가이샤 탁산류의 고분자 결합체
JP5419685B2 (ja) 2006-05-16 2014-02-19 ファーマサイエンス・インコーポレイテッド Iapbirドメイン結合タンパク質
JP5181347B2 (ja) 2006-05-18 2013-04-10 日本化薬株式会社 ポドフィロトキシン類の高分子結合体
WO2008041610A1 (fr) * 2006-10-03 2008-04-10 Nippon Kayaku Kabushiki Kaisha Mélange d'un dérivé de résorcinol avec un polymère
JP5503872B2 (ja) 2006-11-06 2014-05-28 日本化薬株式会社 核酸系代謝拮抗剤の高分子誘導体
US8188222B2 (en) 2006-11-08 2012-05-29 Nippon Kayaku Kabushiki Kaisha High molecular weight derivative of nucleic acid antimetabolite
KR100847331B1 (ko) * 2006-12-14 2008-07-21 한미약품 주식회사 도세탁셀의 제조방법 및 이에 사용되는 중간체
EP2206502B1 (en) 2007-09-28 2018-09-12 Nippon Kayaku Kabushiki Kaisha Polymer conjugate of steroid
EP2258397B1 (en) * 2008-03-18 2017-10-11 Nippon Kayaku Kabushiki Kaisha Polymer conjugate of physiologically active substance
JP2011517455A (ja) 2008-03-31 2011-06-09 フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド C(10)エチルエステルおよびc(10)シクロプロピルエステル置換タキサン
EP2284209B1 (en) 2008-05-08 2016-08-31 Nippon Kayaku Kabushiki Kaisha Polymer conjugate of folic acid or folic acid derivative
EP2431403B1 (en) 2009-05-15 2016-09-28 Nipponkayaku Kabushikikaisha Polymer conjugate of bioactive substance having hydroxy group
US9284350B2 (en) 2010-02-12 2016-03-15 Pharmascience Inc. IAP BIR domain binding compounds
JP5856069B2 (ja) 2010-11-17 2016-02-09 日本化薬株式会社 新規なシチジン系代謝拮抗剤の高分子誘導体
PT2754682T (pt) 2011-09-11 2017-08-29 Nippon Kayaku Kk Método para o fabrico de copolímero de bloco

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4942184A (en) * 1988-03-07 1990-07-17 The United States Of America As Represented By The Department Of Health And Human Services Water soluble, antineoplastic derivatives of taxol
FR2679230B1 (fr) * 1991-07-16 1993-11-19 Rhone Poulenc Rorer Sa Nouveaux derives d'analogues du taxol, leur preparation et les compositions qui les contiennent.
FR2687151B1 (fr) * 1992-02-07 1994-03-25 Rhone Poulenc Rorer Sa Nouveaux derives de la baccatine iii et de la desacetyl-10 baccatine iii, leur preparation et les compositions pharmaceutiques qui les contiennent.
US5880131A (en) * 1993-10-20 1999-03-09 Enzon, Inc. High molecular weight polymer-based prodrugs
JPH08253465A (ja) * 1995-03-17 1996-10-01 Dai Ichi Seiyaku Co Ltd 四環性化合物

Also Published As

Publication number Publication date
EP0930309A4 (en) 2001-09-26
KR20000023664A (ko) 2000-04-25
JP3942197B2 (ja) 2007-07-11
CA2259977A1 (en) 1998-01-22
KR100476247B1 (ko) 2005-03-10
CN1097044C (zh) 2002-12-25
CA2259977C (en) 2005-06-28
US6025385A (en) 2000-02-15
AU3460297A (en) 1998-02-09
AU710156B2 (en) 1999-09-16
WO1998002426A1 (fr) 1998-01-22
EP0930309A1 (en) 1999-07-21
CN1225633A (zh) 1999-08-11

Similar Documents

Publication Publication Date Title
BR9710366A (pt) Derivados de taxane e drogas que os contêm
PT1112251E (pt) Derivados de azetidina sua preparacao e medicamentos que os contem
PT835246E (pt) Compostos aromaticos e composicoes farmaceuticas que os contem
PT944614E (pt) Derivados da benzotiofenocarboxamida e antagonistas de pgd2 que os contem
FI973243A0 (fi) Uusi farmaseuttinen yhdistelmä
FI953479A7 (fi) 1-aryylipyrimidiinijohdannaiset ja niiden farmaseuttinen käyttö
DK0783302T3 (da) Lægemidler
PT1038874E (pt) Derivados de oxima e produtos agro-quimicos que os contem
PT879814E (pt) Compostos tri-aromaticos composicoes que os contem e utilizacoes
FR11C0020I2 (fr) Dérives difluoroprostaglandines et leur application
ATE367150T1 (de) Arzneimittel
NO20002359L (no) Adenosinderivater og farmasoytisk sammensetning inneholdende derivatene
FI961599A7 (fi) 1N-alkyyli-N-aryylipyrimidiiniamiineja ja niiden johdannaisia
BR9607851B1 (pt) combinaÇço e formulaÇço farmacÊutica.
FI973733L (fi) Farmaseuttinen valmiste ja menetelmä sen valmistamiseksi
EE04277B1 (et) Taksoidide klassi kuuluvate derivaatide valmistamismeetod
LV12624B (lv) Tienilazolilalkosietanamini to iegusanas panemiens un pielietojums medikamentu legusana
DE69614718D1 (de) Behälter und darin befestigtes drehendes Teil
FR2738176B1 (fr) Decoupeuse non rotative et indexable
BR9707812A (pt) Composto composto farmacêutica e uso do composto
EE9800378A (et) Alküülaminobensotiasooli ja -bensoksasooli derivaadid
NO982874D0 (no) Farmas°ytiske preparater med vitamin D-analoger
PT1187847E (pt) Derivados de estreptograminas sua preparacao e as composicoes que os contem
DE69415570D1 (de) Esculetin Derivate und pharmazeutische Zusammenstellung
FI942294A7 (fi) Bentsopyraanijohdannaiset ja niiden käyttö

Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PRESENTE PEDIDO, UMA VEZ QUE NAO ATENDE AO REQUISITO DE NOVIDADE ( ART. 8O COMBINADO COM ART. 11 DA LPI ); NAO ATENDE AO REQUISITO DE ATIVIDADE INVENTIVA ( ART. 8O COMBINADO COM ART. 13 DA LPI); NAO APRESENTA SUFUCIENCIA DESCRITIVA ( ART. 24 DA LPI ); AS REIVINDICACOES ESTAO INDEFINIDAS E/OU NAO ESTAO FUNDAMENTADAS NO RELATORIO DESCRITIVO ( ART. 25 DA LPI )

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.