BR112021002523A2 - método para preparar um composto - Google Patents
método para preparar um composto Download PDFInfo
- Publication number
- BR112021002523A2 BR112021002523A2 BR112021002523-5A BR112021002523A BR112021002523A2 BR 112021002523 A2 BR112021002523 A2 BR 112021002523A2 BR 112021002523 A BR112021002523 A BR 112021002523A BR 112021002523 A2 BR112021002523 A2 BR 112021002523A2
- Authority
- BR
- Brazil
- Prior art keywords
- formula
- compound
- 7alkyl
- halogen
- 7alkoxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
- C07H7/06—Heterocyclic radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Furan Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR10-2018-0094261 | 2018-08-13 | ||
| KR20180094261 | 2018-08-13 | ||
| PCT/KR2019/010123 WO2020036382A1 (ko) | 2018-08-13 | 2019-08-09 | Sglt 저해제의 합성에 유용한 중간체의 제조 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR112021002523A2 true BR112021002523A2 (pt) | 2021-05-04 |
Family
ID=69525610
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR112021002523-5A BR112021002523A2 (pt) | 2018-08-13 | 2019-08-09 | método para preparar um composto |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US11661406B2 (de) |
| EP (1) | EP3838894B1 (de) |
| JP (1) | JP7146067B2 (de) |
| KR (1) | KR102307475B1 (de) |
| CN (1) | CN112585124B (de) |
| BR (1) | BR112021002523A2 (de) |
| CA (1) | CA3109107C (de) |
| CO (1) | CO2021001857A2 (de) |
| ES (1) | ES2980368T3 (de) |
| MX (1) | MX2021001732A (de) |
| PE (1) | PE20211206A1 (de) |
| PH (1) | PH12021550297A1 (de) |
| WO (1) | WO2020036382A1 (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102572714B1 (ko) * | 2020-02-27 | 2023-08-31 | 주식회사 대웅제약 | Sglt 저해제의 합성에 유용한 중간체 및 이를 이용한 sglt 저해제의 제조 방법 |
| KR102693201B1 (ko) * | 2020-09-10 | 2024-08-08 | 주식회사 대웅제약 | Sglt 저해제 중간체의 합성 방법 |
| KR20230110001A (ko) * | 2022-01-14 | 2023-07-21 | 주식회사 대웅제약 | Ssglt 저해제의 합성에 유용한 중간체의 제조 방법 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009014970A1 (en) | 2007-07-26 | 2009-01-29 | Lexicon Pharmaceuticals, Inc. | Methods and compounds useful for the preparation of sodium glucose co-transporter 2 inhibitors |
| ES2719656T3 (es) * | 2011-06-01 | 2019-07-11 | Green Cross Corp | Derivados de difenilmetano novedosos como inhibidores del SGLT2 |
| US9340521B2 (en) * | 2013-03-18 | 2016-05-17 | Green Cross Corporation | Method for dual inhibition of SGLT1 and SGLT2 using diphenylmethane derivatives |
| AU2014317663B2 (en) | 2013-09-09 | 2018-02-08 | Youngene Therapeutics Co., Ltd. | C-aryl glucoside derivative, preparation method for same, and medical applications thereof |
| HRP20211670T8 (hr) | 2016-06-17 | 2022-03-18 | Daewoong Pharmaceutical Co., Ltd. | Derivat difenilmetana u kristalnom obliku |
| KR101770302B1 (ko) | 2016-06-28 | 2017-08-22 | 주식회사 녹십자 | 다이페닐메탄 유도체의 제조방법 |
| CN110337442B (zh) * | 2017-02-24 | 2023-05-12 | 东亚St株式会社 | 作为2型钠依赖性葡萄糖转运蛋白抑制剂的新型葡萄糖衍生物 |
-
2019
- 2019-08-09 US US17/266,844 patent/US11661406B2/en active Active
- 2019-08-09 BR BR112021002523-5A patent/BR112021002523A2/pt unknown
- 2019-08-09 KR KR1020190097311A patent/KR102307475B1/ko active IP Right Grant
- 2019-08-09 WO PCT/KR2019/010123 patent/WO2020036382A1/ko unknown
- 2019-08-09 ES ES19850413T patent/ES2980368T3/es active Active
- 2019-08-09 CN CN201980054448.2A patent/CN112585124B/zh active Active
- 2019-08-09 PE PE2021000202A patent/PE20211206A1/es unknown
- 2019-08-09 EP EP19850413.6A patent/EP3838894B1/de active Active
- 2019-08-09 CA CA3109107A patent/CA3109107C/en active Active
- 2019-08-09 JP JP2021507818A patent/JP7146067B2/ja active Active
- 2019-08-09 MX MX2021001732A patent/MX2021001732A/es unknown
-
2021
- 2021-02-10 PH PH12021550297A patent/PH12021550297A1/en unknown
- 2021-02-16 CO CONC2021/0001857A patent/CO2021001857A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP3838894A1 (de) | 2021-06-23 |
| CN112585124A (zh) | 2021-03-30 |
| PE20211206A1 (es) | 2021-07-05 |
| CO2021001857A2 (es) | 2021-02-26 |
| EP3838894B1 (de) | 2024-03-13 |
| WO2020036382A1 (ko) | 2020-02-20 |
| JP7146067B2 (ja) | 2022-10-03 |
| CA3109107A1 (en) | 2020-02-20 |
| US11661406B2 (en) | 2023-05-30 |
| EP3838894A4 (de) | 2022-04-20 |
| PH12021550297A1 (en) | 2021-10-11 |
| MX2021001732A (es) | 2021-06-23 |
| KR102307475B1 (ko) | 2021-09-30 |
| US20210292291A1 (en) | 2021-09-23 |
| JP2021534174A (ja) | 2021-12-09 |
| CN112585124B (zh) | 2024-04-19 |
| CA3109107C (en) | 2023-04-25 |
| KR20200019092A (ko) | 2020-02-21 |
| ES2980368T3 (es) | 2024-10-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B15K | Others concerning applications: alteration of classification |
Free format text: AS CLASSIFICACOES ANTERIORES ERAM: C07D 307/82 , C07D 409/04 , C07H 7/06 , C07H 1/00 Ipc: C07D 307/82 (2006.01), C07D 409/04 (2006.01), C07H |
|
| B06W | Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette] |