BR112018011830A2 - cristal de 2-(3-etanossulfonilpiridina-2-il)-5-(trifluorometanossulfonil)benzoxazol - Google Patents

cristal de 2-(3-etanossulfonilpiridina-2-il)-5-(trifluorometanossulfonil)benzoxazol

Info

Publication number
BR112018011830A2
BR112018011830A2 BR112018011830-3A BR112018011830A BR112018011830A2 BR 112018011830 A2 BR112018011830 A2 BR 112018011830A2 BR 112018011830 A BR112018011830 A BR 112018011830A BR 112018011830 A2 BR112018011830 A2 BR 112018011830A2
Authority
BR
Brazil
Prior art keywords
crystal
trifluoromethanesulfonyl
benzoxazole
ethanesulfonylpyridine
ethanesulfonylpyridin
Prior art date
Application number
BR112018011830-3A
Other languages
English (en)
Japanese (ja)
Inventor
Miyamoto Takashi
Takebayashi Kosuke
Original Assignee
Sumitomo Chemical Company, Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Company, Limited filed Critical Sumitomo Chemical Company, Limited
Publication of BR112018011830A2 publication Critical patent/BR112018011830A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/76—1,3-Oxazoles; Hydrogenated 1,3-oxazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/46—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom rings with more than six members
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N23/00—Investigating or analysing materials by the use of wave or particle radiation, e.g. X-rays or neutrons, not covered by groups G01N3/00 – G01N17/00, G01N21/00 or G01N22/00
    • G01N23/20—Investigating or analysing materials by the use of wave or particle radiation, e.g. X-rays or neutrons, not covered by groups G01N3/00 – G01N17/00, G01N21/00 or G01N22/00 by using diffraction of the radiation by the materials, e.g. for investigating crystal structure; by using scattering of the radiation by the materials, e.g. for investigating non-crystalline materials; by using reflection of the radiation by the materials
    • G01N23/20075—Investigating or analysing materials by the use of wave or particle radiation, e.g. X-rays or neutrons, not covered by groups G01N3/00 – G01N17/00, G01N21/00 or G01N22/00 by using diffraction of the radiation by the materials, e.g. for investigating crystal structure; by using scattering of the radiation by the materials, e.g. for investigating non-crystalline materials; by using reflection of the radiation by the materials by measuring interferences of X-rays, e.g. Borrmann effect
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Analytical Chemistry (AREA)
  • Biochemistry (AREA)
  • General Physics & Mathematics (AREA)
  • Immunology (AREA)
  • Pathology (AREA)
  • Physics & Mathematics (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

um cristal do tipo 2 de 2-(3-etanossulfonilpiridin-2-il)-5-(trifluorometanossulfonil)benzoxazol tendo picos de difração a 2¿ = 14,0 ± 0,2°, 14,3 ± 0,2°, 16,5 ± 0,2°, 16,9 ± 0,2°, 17,6 ± 0,2°, 18,8 ± 0,2°, 19,9 ± 0,2°, e 22,3 ± 0,2° em difração de raio x de pó usando radiação de cu-ka é um cristal estável.
BR112018011830-3A 2015-12-16 2016-12-12 cristal de 2-(3-etanossulfonilpiridina-2-il)-5-(trifluorometanossulfonil)benzoxazol BR112018011830A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2015244909 2015-12-16
JP2015-244909 2015-12-16
PCT/JP2016/086849 WO2017104592A1 (ja) 2015-12-16 2016-12-12 ２－（３－エタンスルホニルピリジン－２－イル）－５－（トリフルオロメタンスルホニル）ベンズオキサゾールの結晶

Publications (1)

Publication Number Publication Date
BR112018011830A2 true BR112018011830A2 (pt) 2018-12-04

Family

ID=59056594

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112018011830-3A BR112018011830A2 (pt) 2015-12-16 2016-12-12 cristal de 2-(3-etanossulfonilpiridina-2-il)-5-(trifluorometanossulfonil)benzoxazol

Country Status (11)

Country Link
US (1) US10448640B2 (pt)
EP (1) EP3392248B1 (pt)
JP (2) JP6665869B2 (pt)
KR (1) KR102627208B1 (pt)
CN (1) CN108401430B (pt)
AU (1) AU2016371984A1 (pt)
BR (1) BR112018011830A2 (pt)
IL (1) IL259698B (pt)
PH (1) PH12018501180A1 (pt)
TW (1) TW201726667A (pt)
WO (1) WO2017104592A1 (pt)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN108401430B (zh) * 2015-12-16 2021-06-29 住友化学株式会社 2-(3-乙磺酰基吡啶-2-基)-5-(三氟甲磺酰基)苯并噁唑晶体
CA3054591A1 (en) 2017-03-31 2018-10-04 Basf Se Pyrimidinium compounds and their mixtures for combating animal pests
RU2019136972A (ru) 2017-04-26 2021-05-26 Басф Се Замещенные сукцинимидные производные в качестве пестицидов
WO2019121143A1 (en) 2017-12-20 2019-06-27 Basf Se Substituted cyclopropyl derivatives
KR20200108007A (ko) 2018-01-09 2020-09-16 바스프 에스이 질화작용 저해제로서의 실릴에티닐 헤타릴 화합물
WO2019137995A1 (en) 2018-01-11 2019-07-18 Basf Se Novel pyridazine compounds for controlling invertebrate pests
JP7444780B2 (ja) 2018-02-28 2024-03-06 ビーエーエスエフ ソシエタス・ヨーロピア 硝化阻害剤としてのｎ－官能化アルコキシピラゾール化合物の使用
EP3758491A1 (en) 2018-02-28 2021-01-06 Basf Se Use of pyrazole propargyl ethers as nitrification inhibitors
CN111683529B (zh) 2018-02-28 2022-10-14 巴斯夫欧洲公司 烷氧基吡唑作为硝化抑制剂的用途
KR20210008036A (ko) 2018-05-15 2021-01-20 바스프 에스이 벤즈피리목산 및 옥사조술필을 포함하는 혼합물 및 이의 용도 및 이의 적용 방법
WO2019224092A1 (en) 2018-05-22 2019-11-28 Basf Se Pesticidally active c15-derivatives of ginkgolides
WO2020002472A1 (en) 2018-06-28 2020-01-02 Basf Se Use of alkynylthiophenes as nitrification inhibitors
EP3826983B1 (en) 2018-07-23 2024-05-15 Basf Se Use of substituted 2-thiazolines as nitrification inhibitors
PL3826982T3 (pl) 2018-07-23 2024-04-02 Basf Se Zastosowanie podstawionych związków tiazolidynowych jako inhibitora nitryfikacji
TWI800674B (zh) * 2018-08-20 2023-05-01 日商住友化學股份有限公司 唑化合物及其用途
EP3613736A1 (en) 2018-08-22 2020-02-26 Basf Se Substituted glutarimide derivatives
EP3628156A1 (en) 2018-09-28 2020-04-01 Basf Se Method for controlling pests of sugarcane, citrus, rapeseed, and potato plants
EP3628157A1 (en) 2018-09-28 2020-04-01 Basf Se Method of controlling insecticide resistant insects and virus transmission to plants
EP3628158A1 (en) 2018-09-28 2020-04-01 Basf Se Pesticidal mixture comprising a mesoionic compound and a biopesticide
US20220046925A1 (en) 2018-09-28 2022-02-17 Basf Se Method of controlling pests by seed treatment application of a mesoionic compound or mixture thereof
EP3643705A1 (en) 2018-10-24 2020-04-29 Basf Se Pesticidal compounds
EP3696177A1 (en) 2019-02-12 2020-08-19 Basf Se Heterocyclic compounds for the control of invertebrate pests
US20220202017A1 (en) 2019-05-29 2022-06-30 Basf Se Mesoionic imidazolium compounds and derivatives for combating animal pests
EP3769623A1 (en) 2019-07-22 2021-01-27 Basf Se Mesoionic imidazolium compounds and derivatives for combating animal pests
CN112056318B (zh) * 2019-06-10 2023-10-20 东莞市东阳光菌阳氢专利农药有限公司 一种含有Oxazosulfyl与抑食肼的杀虫组合物
EP3766879A1 (en) 2019-07-19 2021-01-20 Basf Se Pesticidal pyrazole derivatives
JP7388125B2 (ja) * 2019-10-28 2023-11-29 住友化学株式会社 農薬粒剤
US20240101496A1 (en) 2021-02-02 2024-03-28 Basf Se Synergistic action of dcd and alkoxypyrazoles as nitrification inhibitors
CA3219128A1 (en) 2021-05-21 2022-11-24 Barbara Nave Use of an n-functionalized alkoxy pyrazole compound as nitrification inhibitor
CA3219022A1 (en) 2021-05-21 2022-11-24 Barbara Nave Use of ethynylpyridine compounds as nitrification inhibitors
CA3223077A1 (en) 2021-06-21 2022-12-29 Barbara Nave Metal-organic frameworks with pyrazole-based building blocks
WO2023203066A1 (en) 2022-04-21 2023-10-26 Basf Se Synergistic action as nitrification inhibitors of dcd oligomers with alkoxypyrazole and its oligomers
WO2024028243A1 (en) 2022-08-02 2024-02-08 Basf Se Pyrazolo pesticidal compounds

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2938601B1 (en) * 2012-12-27 2018-05-16 Sumitomo Chemical Company Limited Fused oxazole compounds and use thereof for pest control
CN105142403B (zh) * 2013-01-31 2018-06-19 住友化学株式会社 用于防治害虫的方法
ES2693320T3 (es) * 2014-06-26 2018-12-11 Sumitomo Chemical Company, Limited Método para la producción compuestos heterocíclicos condensados
CN106572657B (zh) * 2014-07-04 2019-08-23 住友化学株式会社 有害生物防治组合物及其用途
JP2017025014A (ja) * 2015-07-21 2017-02-02 住友化学株式会社 ベンゾオキサゾール化合物の製造方法
CN108401430B (zh) * 2015-12-16 2021-06-29 住友化学株式会社 2-(3-乙磺酰基吡啶-2-基)-5-(三氟甲磺酰基)苯并噁唑晶体
JP2016056197A (ja) 2016-01-12 2016-04-21 住友化学株式会社 有害生物防除組成物及びその用途

Also Published As

Publication number Publication date
AU2016371984A1 (en) 2018-07-05
TW201726667A (zh) 2017-08-01
WO2017104592A1 (ja) 2017-06-22
JP2020100634A (ja) 2020-07-02
CN108401430A (zh) 2018-08-14
PH12018501180A1 (en) 2019-01-28
JPWO2017104592A1 (ja) 2018-10-04
US20180368407A1 (en) 2018-12-27
JP6863493B2 (ja) 2021-04-21
KR102627208B1 (ko) 2024-01-19
EP3392248A4 (en) 2019-05-22
JP6665869B2 (ja) 2020-03-13
CN108401430B (zh) 2021-06-29
EP3392248A1 (en) 2018-10-24
US10448640B2 (en) 2019-10-22
IL259698A (en) 2018-07-31
KR20180095855A (ko) 2018-08-28
EP3392248B1 (en) 2020-05-06
IL259698B (en) 2020-10-29

Similar Documents

Publication Publication Date Title
BR112018011830A2 (pt) cristal de 2-(3-etanossulfonilpiridina-2-il)-5-(trifluorometanossulfonil)benzoxazol
CO6430432A2 (es) Cristales
EP2956064A4 (en) LARGE VIEW FIELD OF X-RAY FIELD PHASE CONTRAST IMAGING AND CT IN HIGH ENERGY
NI201600022A (es) Compuestos terapéuticamente activos y sus métodos de uso
HUE045353T2 (hu) N-((4,6-dimetil-2-oxo-1,2-dihidropiridin-3-il)-metil)-5-(etil-(tetrahidro-2H-pirán-4-il) -amino)-4-metil-4'-(morfolino-metil)-[1,1'-bifenil]-3-karboxamid-hidrobromid a hematológiai rendszer egy sejtszaporodásos rendellenességének kezelésében való alkalmazásra
PL3220916T3 (pl) Sposób leczenia raka n-((4,6-dimetylo-2-okso-1,2-dihydropirydyn-3-ylo)metylo)-5-(etylo(tetrahydro-2h-piran-4-ylo)amino)-4-metylo-4'-(morfolinometylo)-[1,1'-bifenylo]-3-karboksyamidem
GT201700023A (es) Derivados de heterociclico opcionalmente condensados de piridimina útiles para el tratamiento de enfermedades inflamatorias, metabolicas, oncológicas y autoinmunitarias
DK3240538T3 (da) Anvendelse af masitinib til behandling af en underpopulation af patienter med amyotrofisk lateralsklerose
BR112016019592A8 (pt) Composto, uso de um composto, e, composição farmacêutica
FI20135204L (fi) Testihallinta
DK3603524T3 (da) Indretning til digital billeddannelse i hovedregionen af en patient
BR112019009172A2 (pt) formulações para radioterapia e diagnóstico por imagem.
DK3193978T3 (da) Lægemiddelinjektor af hudplastertypen til voluminøs bolus med medikamentforvarmning
ZA201906541B (en) Isoxazole derivatives as nuclear receptor agonists and uses thereof
MA43361A (fr) Composition pour le soin et la protection de cultures
CL2017001164A1 (es) Compuesto de diaril isoxazolina
TR201901516T4 (tr) Nöroprotektif ajanlar ve bunların kullanımları.
UA117933C2 (uk) Поліпептид, здатний зв'язувати с5-компонент комплементу людини
MX2015012318A (es) Formas de estado solido de un derivado de quinazolina y su uso como un inhibidor de braf.
MA40524A (fr) Dérivés d'adrénomédulline stabilisés et leur utilisation
DK3141088T3 (da) Feedback-billeddannelse med ultralav dosis ved hjælp af laser-compton-røntgen- og laser-compton-gamma-strålekilder
BR112017016396A2 (pt) composto, composição farmacêutica, uso de um composto, e, método.
AR095346A1 (es) Compuesto de hidrato de fluoreno y sus cristales
MX2017003607A (es) Sales de clorhidrato de aluminio que exhiben un pico 1 sec alto.
IL281229A (en) Salts of cycloserine compounds and their applications

Legal Events

Date Code Title Description
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.