BR112015026685A2 - agente de diminuição de ácido úrico - Google Patents
agente de diminuição de ácido úricoInfo
- Publication number
- BR112015026685A2 BR112015026685A2 BR112015026685A BR112015026685A BR112015026685A2 BR 112015026685 A2 BR112015026685 A2 BR 112015026685A2 BR 112015026685 A BR112015026685 A BR 112015026685A BR 112015026685 A BR112015026685 A BR 112015026685A BR 112015026685 A2 BR112015026685 A2 BR 112015026685A2
- Authority
- BR
- Brazil
- Prior art keywords
- tyrosine
- uric acid
- lowering agent
- acid lowering
- cyclothyrosyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/005—Enzyme inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/01—Hydrolysed proteins; Derivatives thereof
- A61K38/011—Hydrolysed proteins; Derivatives thereof from plants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/05—Dipeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/12—Cyclic peptides with only normal peptide bonds in the ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Abstract
resumo patente de invenção: "agente de diminuição de ácido úrico". trata-se de um agente de diminuição de ácido úrico que contém, como um ingrediente ativo, um dipeptídeo cíclico contendo tirosina selecionado a partir de um grupo que consiste em ciclotriptofaniltirosina, cicloseriltirosina, cicloproliltirosina, ciclotirosilglicina, ciclotirosiltirosina, ciclofenilalaniltirosina, cicloleuciltirosina, ciclolisiltirosina, ciclohistidiltirosina, cicloalaniltirosina, cicloglutamiltirosina, ciclovaliltirosina, cicloisoleuciltirosina, ciclotreoniltirosina, cicloaspartiltirosina, cicloasparaginiltirosina, cicloglutaminiltirosina, cicloarginiltirosina, ciclometioniltirosina e ciclotirosilcisteína ou um sal dos mesmos. o agente de diminuição de ácido úrico da presente invenção tem uma excelente ação de diminuição de um nível de ácido úrico, e o agente de diminuição de ácido úrico é útil, por exemplo, na prevenção ou no tratamento de hiperuricemia, gota ou similar. 1/1
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/JP2014/066424 WO2015194034A1 (ja) | 2014-06-20 | 2014-06-20 | 尿酸値低下剤 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112015026685A2 true BR112015026685A2 (pt) | 2017-07-25 |
Family
ID=52823346
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112015026685A BR112015026685A2 (pt) | 2014-06-20 | 2014-06-20 | agente de diminuição de ácido úrico |
Country Status (13)
Country | Link |
---|---|
US (1) | US9650415B2 (pt) |
EP (1) | EP3159005A1 (pt) |
JP (1) | JP5690028B1 (pt) |
KR (1) | KR20160022292A (pt) |
CN (1) | CN105407907A (pt) |
AU (1) | AU2014386720B2 (pt) |
BR (1) | BR112015026685A2 (pt) |
CA (1) | CA2904493A1 (pt) |
HK (1) | HK1215797A1 (pt) |
MX (1) | MX2015015162A (pt) |
SG (1) | SG11201507823RA (pt) |
TW (1) | TWI564018B (pt) |
WO (1) | WO2015194034A1 (pt) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2014200000A1 (ja) | 2013-06-10 | 2014-12-18 | サントリーホールディングス株式会社 | ジケトピペラジンを含有する植物エキス及びその製造方法 |
JP6772133B2 (ja) * | 2015-07-02 | 2020-10-21 | サントリーホールディングス株式会社 | Glp−2分泌促進用組成物 |
WO2017002906A1 (ja) * | 2015-07-02 | 2017-01-05 | サントリーホールディングス株式会社 | アルコール吸収抑制用組成物 |
JP6669750B2 (ja) * | 2015-07-16 | 2020-03-18 | サントリーホールディングス株式会社 | 環状ジペプチド含有血清カルノシン分解酵素阻害用組成物 |
WO2017014120A1 (ja) * | 2015-07-17 | 2017-01-26 | サントリーホールディングス株式会社 | Trpv1刺激用組成物 |
SG10201912392SA (en) * | 2015-07-27 | 2020-02-27 | Suntory Holdings Ltd | Composition containing cyclic dipeptide and sweetening agent |
JP6719475B2 (ja) * | 2015-09-04 | 2020-07-08 | サントリーホールディングス株式会社 | ウレアーゼ活性阻害剤 |
CN109562110A (zh) | 2016-05-26 | 2019-04-02 | 株式会社日本阿明诺化学 | 睡眠改善剂 |
JP2019011303A (ja) * | 2017-07-03 | 2019-01-24 | サントリーホールディングス株式会社 | 環状ジペプチドの製造方法 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5973574A (ja) * | 1982-10-21 | 1984-04-25 | Grelan Pharmaceut Co Ltd | 環状ジペプチド類 |
PT1311269E (pt) * | 2000-08-04 | 2012-05-10 | Dmi Biosciences Inc | Método de utilização de dicetopiperazinas e composição que contém as mesmas |
ES2297142T3 (es) | 2002-03-28 | 2008-05-01 | Eli Lilly And Company | Arilbenzodiazepinas sustituidas con piperazina y su uso como antagonistas del receptor de dopamina para el tratamiento de trastornos psicoticos. |
EP2537524B1 (en) * | 2003-05-15 | 2016-07-06 | Ampio Pharmaceuticals, Inc. | Treatment of T-cell mediated diseases |
JP2006111541A (ja) | 2004-10-12 | 2006-04-27 | Toyo Shinyaku:Kk | 葛花処理物を含有する経口用肌質改善剤 |
EP2088143A1 (en) * | 2008-01-24 | 2009-08-12 | Commissariat A L'energie Atomique | Novel inhibitors of mycobacterium tuberculosis complex cytochrome P450 CYP121 |
JP5058379B2 (ja) | 2009-12-25 | 2012-10-24 | サントリーホールディングス株式会社 | 学習意欲改善剤 |
JP2013053115A (ja) * | 2011-09-06 | 2013-03-21 | Josho Gakuen | α環状ジペプチドの製造方法 |
WO2014200000A1 (ja) * | 2013-06-10 | 2014-12-18 | サントリーホールディングス株式会社 | ジケトピペラジンを含有する植物エキス及びその製造方法 |
-
2014
- 2014-06-20 AU AU2014386720A patent/AU2014386720B2/en not_active Ceased
- 2014-06-20 CA CA2904493A patent/CA2904493A1/en not_active Abandoned
- 2014-06-20 EP EP14894840.9A patent/EP3159005A1/en not_active Withdrawn
- 2014-06-20 US US14/787,677 patent/US9650415B2/en not_active Expired - Fee Related
- 2014-06-20 KR KR1020157031132A patent/KR20160022292A/ko not_active Application Discontinuation
- 2014-06-20 SG SG11201507823RA patent/SG11201507823RA/en unknown
- 2014-06-20 MX MX2015015162A patent/MX2015015162A/es unknown
- 2014-06-20 CN CN201480005474.3A patent/CN105407907A/zh active Pending
- 2014-06-20 BR BR112015026685A patent/BR112015026685A2/pt not_active IP Right Cessation
- 2014-06-20 WO PCT/JP2014/066424 patent/WO2015194034A1/ja active Application Filing
- 2014-06-20 JP JP2014545991A patent/JP5690028B1/ja active Active
- 2014-09-26 TW TW103133548A patent/TWI564018B/zh not_active IP Right Cessation
-
2016
- 2016-04-01 HK HK16103771.1A patent/HK1215797A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
AU2014386720B2 (en) | 2016-07-21 |
TWI564018B (zh) | 2017-01-01 |
CN105407907A (zh) | 2016-03-16 |
KR20160022292A (ko) | 2016-02-29 |
JPWO2015194034A1 (ja) | 2017-04-20 |
US9650415B2 (en) | 2017-05-16 |
CA2904493A1 (en) | 2015-12-20 |
MX2015015162A (es) | 2016-03-15 |
AU2014386720A1 (en) | 2016-01-21 |
US20160159858A1 (en) | 2016-06-09 |
JP5690028B1 (ja) | 2015-03-25 |
EP3159005A1 (en) | 2017-04-26 |
TW201600103A (zh) | 2016-01-01 |
HK1215797A1 (zh) | 2016-09-15 |
SG11201507823RA (en) | 2016-01-28 |
WO2015194034A1 (ja) | 2015-12-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: application dismissed [chapter 8.6 patent gazette] | ||
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] | ||
B350 | Update of information on the portal [chapter 15.35 patent gazette] |