BR112014026266A2 - derivado de quinazolidinadiona - Google Patents
derivado de quinazolidinadionaInfo
- Publication number
- BR112014026266A2 BR112014026266A2 BR112014026266A BR112014026266A BR112014026266A2 BR 112014026266 A2 BR112014026266 A2 BR 112014026266A2 BR 112014026266 A BR112014026266 A BR 112014026266A BR 112014026266 A BR112014026266 A BR 112014026266A BR 112014026266 A2 BR112014026266 A2 BR 112014026266A2
- Authority
- BR
- Brazil
- Prior art keywords
- quinazolidinedione
- derivative
- formula
- pharmaceutically acceptable
- relates
- Prior art date
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- A61P19/04—Drugs for skeletal disorders for non-specific disorders of the connective tissue
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- C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
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- C07C321/24—Thiols, sulfides, hydropolysulfides, or polysulfides having thio groups bound to carbon atoms of six-membered aromatic rings
- C07C321/28—Sulfides, hydropolysulfides, or polysulfides having thio groups bound to carbon atoms of six-membered aromatic rings
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
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- A61K31/18—Sulfonamides
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- C07C317/32—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C317/34—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring
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- C07C317/34—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring
- C07C317/38—Sulfones; Sulfoxides having sulfone or sulfoxide groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having sulfone or sulfoxide groups and amino groups bound to carbon atoms of six-membered aromatic rings being part of the same non-condensed ring or of a condensed ring system containing that ring with the nitrogen atom of at least one amino group being part of any of the groups, X being a hetero atom, Y being any atom, e.g. N-acylaminosulfones
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- C07C323/39—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02W—CLIMATE CHANGE MITIGATION TECHNOLOGIES RELATED TO WASTEWATER TREATMENT OR WASTE MANAGEMENT
- Y02W30/00—Technologies for solid waste management
- Y02W30/50—Reuse, recycling or recovery technologies
- Y02W30/62—Plastics recycling; Rubber recycling
Abstract
abstract the present invention relates to benzamide derivatives represented by formula (i) or pharmaceutically acceptable salts thereof. (i) tradução do resumo resumo patente de invenção: "derivado de quinazolidinadiona". a presente invenção refere-se a um derivado de quinazolidinadiona ou um sal farmaceuticamente aceitável do mesmo o qual é representado pela fórmula (i). (i)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2012098953 | 2012-04-24 | ||
PCT/JP2013/062003 WO2013161851A1 (ja) | 2012-04-24 | 2013-04-24 | ベンズアミド誘導体 |
Publications (1)
Publication Number | Publication Date |
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BR112014026266A2 true BR112014026266A2 (pt) | 2017-06-27 |
Family
ID=49483159
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112014026266A BR112014026266A2 (pt) | 2012-04-24 | 2013-04-24 | derivado de quinazolidinadiona |
Country Status (15)
Country | Link |
---|---|
US (1) | US9695118B2 (pt) |
EP (1) | EP2842939B1 (pt) |
JP (1) | JP6177768B2 (pt) |
KR (1) | KR20150013563A (pt) |
CN (1) | CN104379560A (pt) |
AR (1) | AR090836A1 (pt) |
AU (1) | AU2013253539A1 (pt) |
BR (1) | BR112014026266A2 (pt) |
CA (1) | CA2871237A1 (pt) |
HK (1) | HK1203926A1 (pt) |
MX (1) | MX2014012991A (pt) |
RU (1) | RU2014147017A (pt) |
SG (1) | SG11201406871UA (pt) |
TW (1) | TW201348187A (pt) |
WO (1) | WO2013161851A1 (pt) |
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AU2013253541A1 (en) | 2012-04-24 | 2014-11-20 | Chugai Seiyaku Kabushiki Kaisha | Quinazolinedione derivative |
CN105829285A (zh) | 2013-10-23 | 2016-08-03 | 中外制药株式会社 | 喹唑啉酮和异喹啉酮衍生物 |
KR101810378B1 (ko) * | 2014-11-07 | 2017-12-20 | 론자 리미티드 | 균일 촉매작용에 의한 플루오로 알킬화 화합물의 제조 방법 |
EP3101009A1 (en) * | 2015-06-05 | 2016-12-07 | Lead Pharma Cel Models IP B.V. | Ror gamma (rory) modulators |
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EP3414247B1 (en) * | 2016-02-08 | 2021-04-21 | F. Hoffmann-La Roche AG | Spiroindolinones as ddr1 inhibitors |
CN106397174B (zh) * | 2016-08-24 | 2018-12-21 | 河北诚信集团有限公司 | 一种制备3,6-二氯-2-甲氧基苯甲酸的方法 |
BR112021016564A2 (pt) * | 2019-02-22 | 2021-11-03 | Pi Ind Ltd | Processo para a síntese de compostos de diamida antranílica e intermediários dos mesmos |
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AU2022330732A1 (en) * | 2021-08-17 | 2024-02-15 | Cyrus Therapeutics Inc. | Sos1 inhibitor and use thereof |
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-
2013
- 2013-04-24 TW TW102114528A patent/TW201348187A/zh unknown
- 2013-04-24 RU RU2014147017A patent/RU2014147017A/ru unknown
- 2013-04-24 BR BR112014026266A patent/BR112014026266A2/pt not_active Application Discontinuation
- 2013-04-24 AR ARP130101382A patent/AR090836A1/es unknown
- 2013-04-24 CN CN201380033232.0A patent/CN104379560A/zh active Pending
- 2013-04-24 SG SG11201406871UA patent/SG11201406871UA/en unknown
- 2013-04-24 WO PCT/JP2013/062003 patent/WO2013161851A1/ja active Application Filing
- 2013-04-24 JP JP2014512632A patent/JP6177768B2/ja not_active Expired - Fee Related
- 2013-04-24 KR KR1020147032532A patent/KR20150013563A/ko not_active Application Discontinuation
- 2013-04-24 AU AU2013253539A patent/AU2013253539A1/en not_active Withdrawn
- 2013-04-24 US US14/396,678 patent/US9695118B2/en not_active Expired - Fee Related
- 2013-04-24 CA CA2871237A patent/CA2871237A1/en not_active Abandoned
- 2013-04-24 EP EP13782636.8A patent/EP2842939B1/en not_active Not-in-force
- 2013-04-24 MX MX2014012991A patent/MX2014012991A/es unknown
-
2015
- 2015-05-07 HK HK15104329.7A patent/HK1203926A1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
RU2014147017A (ru) | 2016-06-10 |
JPWO2013161851A1 (ja) | 2015-12-24 |
AU2013253539A1 (en) | 2014-11-13 |
CN104379560A (zh) | 2015-02-25 |
EP2842939B1 (en) | 2018-05-30 |
EP2842939A1 (en) | 2015-03-04 |
US9695118B2 (en) | 2017-07-04 |
AR090836A1 (es) | 2014-12-10 |
TW201348187A (zh) | 2013-12-01 |
CA2871237A1 (en) | 2013-10-31 |
MX2014012991A (es) | 2015-08-14 |
WO2013161851A1 (ja) | 2013-10-31 |
HK1203926A1 (en) | 2015-11-06 |
US20150152047A1 (en) | 2015-06-04 |
EP2842939A4 (en) | 2015-11-11 |
SG11201406871UA (en) | 2014-11-27 |
KR20150013563A (ko) | 2015-02-05 |
JP6177768B2 (ja) | 2017-08-09 |
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