BR112021016564A2 - Processo para a síntese de compostos de diamida antranílica e intermediários dos mesmos - Google Patents

Processo para a síntese de compostos de diamida antranílica e intermediários dos mesmos

Info

Publication number
BR112021016564A2
BR112021016564A2 BR112021016564A BR112021016564A BR112021016564A2 BR 112021016564 A2 BR112021016564 A2 BR 112021016564A2 BR 112021016564 A BR112021016564 A BR 112021016564A BR 112021016564 A BR112021016564 A BR 112021016564A BR 112021016564 A2 BR112021016564 A2 BR 112021016564A2
Authority
BR
Brazil
Prior art keywords
formula
compound
synthesis
intermediates
anthranilic
Prior art date
Application number
BR112021016564A
Other languages
English (en)
Inventor
G M Klausener Alexander
Dnyaneshwar Kalwaghe Amol
Uttamrao Shinde Bharat
Shankar panmand Deepak
Jagadish Pabba
Maruti Madhavrao Kamble
Phaneendrasai Karri
Original Assignee
Pi Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pi Industries Ltd filed Critical Pi Industries Ltd
Publication of BR112021016564A2 publication Critical patent/BR112021016564A2/pt

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/68—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton
    • C07C209/74—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton by halogenation, hydrohalogenation, dehalogenation, or dehydrohalogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/44—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring
    • C07C211/52—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/02—Formation of carboxyl groups in compounds containing amino groups, e.g. by oxidation of amino alcohols
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
    • C07C227/18—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions involving amino or carboxyl groups, e.g. hydrolysis of esters or amides, by formation of halides, salts or esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/52—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
    • C07C229/54—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/14—Preparation of carboxylic acid nitriles by reaction of cyanides with halogen-containing compounds with replacement of halogen atoms by cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C07C255/60—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Toxicology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

processo para a síntese de compostos de diamida antranílica e intermediários dos mesmos. a presente invenção revelou um processo para a síntese de composto de diamida antranílica da fórmula (i), em que, r1, r2, r3a, r3b, r3c, r4, r5, r6 e z são como definido na descrição detalhada. o processo compreende a etapa de obter um composto de anilina substituída por mono ou diciano da fórmula (iv) que é, então, convertido em um composto de ácido antranílico da fórmula (v) ou um composto de amida antranílica da fórmula (va). adicionalmente, o composto da fórmula (vi) pode ser opcionalmente sintetizado a partir do composto da fórmula (iv ou v ou va).
BR112021016564A 2019-02-22 2020-02-20 Processo para a síntese de compostos de diamida antranílica e intermediários dos mesmos BR112021016564A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN201911007091 2019-02-22
PCT/IB2020/051410 WO2020170178A1 (en) 2019-02-22 2020-02-20 A process for the synthesis anthranilic diamide compounds and intermediates thereof

Publications (1)

Publication Number Publication Date
BR112021016564A2 true BR112021016564A2 (pt) 2021-11-03

Family

ID=72144001

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112021016564A BR112021016564A2 (pt) 2019-02-22 2020-02-20 Processo para a síntese de compostos de diamida antranílica e intermediários dos mesmos

Country Status (9)

Country Link
US (1) US11718584B2 (pt)
EP (1) EP3927685A4 (pt)
KR (1) KR20210130738A (pt)
CN (1) CN113614063A (pt)
BR (1) BR112021016564A2 (pt)
CA (1) CA3129950A1 (pt)
IL (1) IL285377B1 (pt)
MX (1) MX2021010098A (pt)
WO (1) WO2020170178A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR123526A1 (es) * 2020-09-17 2022-12-14 Pi Industries Ltd Un proceso para la síntesis de compuestos antranílicos de ácido / amida e intermediarios de los mismos
AR126248A1 (es) * 2021-06-28 2023-10-04 Pi Industries Ltd Un proceso para la preparación de diamidas antranílicas bicíclicas de fórmula (i) e intermediarios de las mismas
CN113444004B (zh) * 2021-06-29 2023-06-23 江西荣兴药业有限公司 3,5-二溴邻氨基苯甲醛生产工艺
WO2024186513A1 (en) * 2023-03-03 2024-09-12 Fmc Corporation Photochemical systems and methods for preparing cyanobenzamides

Family Cites Families (22)

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Publication number Priority date Publication date Assignee Title
TWI325302B (en) 2001-08-13 2010-06-01 Du Pont Benzoxazinone compounds
AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
RU2343151C3 (ru) 2003-01-28 2019-10-01 ЭфЭмСи Корпорейшн Цианоантраниламидные инсектициды
EP1717237B1 (en) 2004-02-18 2010-12-29 Ishihara Sangyo Kaisha, Ltd. Anthranilamides, process for the production thereof, and pest controllers containing the same
MY140912A (en) 2004-07-26 2010-01-29 Du Pont Mixtures of anthranilamide invertebrate pest control agents
TWI363756B (en) * 2004-12-07 2012-05-11 Du Pont Method for preparing n-phenylpyrazole-1-carboxamides
DK2394983T3 (en) 2006-07-19 2014-12-15 Du Pont Process for the preparation of 3-substituted 2-amino-5- halobenzamider
TWI395728B (zh) 2006-12-06 2013-05-11 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
TWI415827B (zh) 2006-12-21 2013-11-21 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
TWI430980B (zh) 2007-06-29 2014-03-21 Du Pont 製備２－胺基－5－氰基苯甲酸衍生物之方法
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TWI432421B (zh) 2007-12-19 2014-04-01 Du Pont 製備２－胺基－５－氰基苯甲酸衍生物之方法
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EP2668153B1 (en) 2011-01-28 2015-03-04 E.I. Du Pont De Nemours And Company Method for preparing 2-aminobenzamide derivatives
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BR112014026266A2 (pt) * 2012-04-24 2017-06-27 Chugai Pharmaceutical Co Ltd derivado de quinazolidinadiona
BR112015027591A2 (pt) * 2013-05-17 2017-07-25 Basf Se processos para a preparação de um ácido, de um cloreto e de um composto de sulfimina
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CN106146414A (zh) 2016-07-07 2016-11-23 浙江大学 喹唑啉二酮类衍生物及其制备方法和用途

Also Published As

Publication number Publication date
CN113614063A (zh) 2021-11-05
EP3927685A4 (en) 2022-11-23
KR20210130738A (ko) 2021-11-01
WO2020170178A1 (en) 2020-08-27
US11718584B2 (en) 2023-08-08
EP3927685A1 (en) 2021-12-29
US20220185782A1 (en) 2022-06-16
MX2021010098A (es) 2021-09-28
IL285377B1 (en) 2024-09-01
IL285377A (en) 2021-09-30
CA3129950A1 (en) 2020-08-27

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B06W Patent application suspended after preliminary examination (for patents with searches from other patent authorities) chapter 6.23 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]