MX2021010098A - Un proceso para la sintesis de compuestos de diamida antranilica y compuestos intermedios de los mismos. - Google Patents

Un proceso para la sintesis de compuestos de diamida antranilica y compuestos intermedios de los mismos.

Info

Publication number
MX2021010098A
MX2021010098A MX2021010098A MX2021010098A MX2021010098A MX 2021010098 A MX2021010098 A MX 2021010098A MX 2021010098 A MX2021010098 A MX 2021010098A MX 2021010098 A MX2021010098 A MX 2021010098A MX 2021010098 A MX2021010098 A MX 2021010098A
Authority
MX
Mexico
Prior art keywords
formula
compound
synthesis
intermediates
anthranilic
Prior art date
Application number
MX2021010098A
Other languages
English (en)
Inventor
Jagadish Pabba
Alexander G M Klausener
Phaneendrasai Karri
Amol Dnyaneshwar Kalwaghe
Bharat Uttamrao Shinde
Deepak Shankar Panmand
Kamble Maruti Madhavrao
Original Assignee
Pi Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pi Industries Ltd filed Critical Pi Industries Ltd
Publication of MX2021010098A publication Critical patent/MX2021010098A/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/68—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton
    • C07C209/74—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton by halogenation, hydrohalogenation, dehalogenation, or dehydrohalogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/44—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring
    • C07C211/52—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/02—Formation of carboxyl groups in compounds containing amino groups, e.g. by oxidation of amino alcohols
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
    • C07C227/18—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions involving amino or carboxyl groups, e.g. hydrolysis of esters or amides, by formation of halides, salts or esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/52—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
    • C07C229/54—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton with amino and carboxyl groups bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/14—Preparation of carboxylic acid nitriles by reaction of cyanides with halogen-containing compounds with replacement of halogen atoms by cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C07C255/60—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Toxicology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

La presente invención divulgó un proceso para la síntesis de compuesto de diamida antranílica de fórmula (I), en donde, R1, R2, R3a, R3b, R3c, R4, R5, R6 y Z son como se definen en la descripción detallada. El proceso 5 que comprende la etapa de obtener un compuesto de anilina monociano- o diciano-sustituida de fórmula (IV) que luego se convierte en un compuesto de ácido antranílico de fórmula (V) o un compuesto de amida antranílica de fórmula (Va). Además, el compuesto de fórmula (VI) se puede sintetizar opcionalmente a partir del compuesto de fórmula (IV o V o Va).
MX2021010098A 2019-02-22 2020-02-20 Un proceso para la sintesis de compuestos de diamida antranilica y compuestos intermedios de los mismos. MX2021010098A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN201911007091 2019-02-22
PCT/IB2020/051410 WO2020170178A1 (en) 2019-02-22 2020-02-20 A process for the synthesis anthranilic diamide compounds and intermediates thereof

Publications (1)

Publication Number Publication Date
MX2021010098A true MX2021010098A (es) 2021-09-28

Family

ID=72144001

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2021010098A MX2021010098A (es) 2019-02-22 2020-02-20 Un proceso para la sintesis de compuestos de diamida antranilica y compuestos intermedios de los mismos.

Country Status (9)

Country Link
US (1) US11718584B2 (es)
EP (1) EP3927685A4 (es)
KR (1) KR20210130738A (es)
CN (1) CN113614063A (es)
BR (1) BR112021016564A2 (es)
CA (1) CA3129950A1 (es)
IL (1) IL285377A (es)
MX (1) MX2021010098A (es)
WO (1) WO2020170178A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022058916A1 (en) * 2020-09-17 2022-03-24 Pi Industries Limited A process for the synthesis of anthranilic acid/amide compounds and intermediates thereof
WO2023275705A1 (en) * 2021-06-28 2023-01-05 Pi Industries Ltd. A process for the preparation of pyrazolopyridine-diamides of formula (i) and intermediates thereof
CN113444004B (zh) * 2021-06-29 2023-06-23 江西荣兴药业有限公司 3,5-二溴邻氨基苯甲醛生产工艺

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AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
TWI325302B (en) 2001-08-13 2010-06-01 Du Pont Benzoxazinone compounds
NZ541112A (en) 2003-01-28 2008-01-31 Du Pont Cyano anthranilamide insecticides
KR100963370B1 (ko) 2004-02-18 2010-06-14 이시하라 산교 가부시끼가이샤 안트라닐아미드계 화합물, 그의 제조 방법 및 그것을함유하는 유해 생물 방제제
MY140912A (en) 2004-07-26 2010-01-29 Du Pont Mixtures of anthranilamide invertebrate pest control agents
TWI363756B (en) 2004-12-07 2012-05-11 Du Pont Method for preparing n-phenylpyrazole-1-carboxamides
CA2656357C (en) 2006-07-19 2014-05-06 E.I. Du Pont De Nemours And Company Process for making 3-substituted 2-amino-5-halobenzamides
TWI395728B (zh) 2006-12-06 2013-05-11 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
TWI415827B (zh) 2006-12-21 2013-11-21 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
TWI430980B (zh) 2007-06-29 2014-03-21 Du Pont 製備２－胺基－5－氰基苯甲酸衍生物之方法
KR20100098382A (ko) 2007-11-08 2010-09-06 이 아이 듀폰 디 네모아 앤드 캄파니 2-아미노-5-시아노벤조산 유도체의 제조 방법
TWI432421B (zh) 2007-12-19 2014-04-01 Du Pont 製備２－胺基－５－氰基苯甲酸衍生物之方法
EP2484676B1 (de) 2008-12-18 2015-01-21 Bayer CropScience AG Tetrazolsubstituierte Anthranilsäureamide als Pestizide
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CN105189477A (zh) * 2013-05-17 2015-12-23 巴斯夫欧洲公司 制备n-取代的1h-吡唑-5-甲酸化合物及其衍生物的方法
MD3259253T2 (ro) 2015-02-16 2020-06-30 Univ Queensland Sulfoniluree și compuși înrudiți și utilizări ale acestora
CN106928216A (zh) * 2015-12-31 2017-07-07 中国科学院上海药物研究所 具有erk激酶抑制活性的化合物、其制备方法和用途
CN106146414A (zh) 2016-07-07 2016-11-23 浙江大学 喹唑啉二酮类衍生物及其制备方法和用途

Also Published As

Publication number Publication date
US11718584B2 (en) 2023-08-08
BR112021016564A2 (pt) 2021-11-03
EP3927685A1 (en) 2021-12-29
CN113614063A (zh) 2021-11-05
WO2020170178A1 (en) 2020-08-27
IL285377A (en) 2021-09-30
US20220185782A1 (en) 2022-06-16
CA3129950A1 (en) 2020-08-27
KR20210130738A (ko) 2021-11-01
EP3927685A4 (en) 2022-11-23

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