BR0311266A - Processo para a preparação de derivados de tioalquilamina - Google Patents

Processo para a preparação de derivados de tioalquilamina

Info

Publication number
BR0311266A
BR0311266A BR0311266-7A BR0311266A BR0311266A BR 0311266 A BR0311266 A BR 0311266A BR 0311266 A BR0311266 A BR 0311266A BR 0311266 A BR0311266 A BR 0311266A
Authority
BR
Brazil
Prior art keywords
formula
preparation
sulfuric acid
thioalkylamine
derivatives
Prior art date
Application number
BR0311266-7A
Other languages
English (en)
Inventor
Joern Stoelting
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of BR0311266A publication Critical patent/BR0311266A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/36—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/24—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of esters of sulfuric acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C323/24—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/25—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

"PROCESSO PARA A PREPARAçãO DE DERIVADOS DE TIOALQUILAMINA". A presente invenção refere-se a um novo processo para a preparação de compostos de fórmula (I) por reação em uma primeira etapa de aminoálcoois de fórmula (II) com oleum para dar ésteres de ácido sulfúrico de fórmula geral (III) e por reação destes ésteres de ácido sulfúrico em uma segunda etapa com mercaptanos ou sais dos mesmos da fórmula geral (IV) em cada fórmula, onde aplicável, R1, R2, R3, R4, R5, R6, R, n e M tem os significados dados na descrição na presença de um diluente e na presença de uma base.
BR0311266-7A 2002-05-24 2003-05-12 Processo para a preparação de derivados de tioalquilamina BR0311266A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP02011545 2002-05-24
PCT/EP2003/004911 WO2003099777A1 (en) 2002-05-24 2003-05-12 Process for the preparation of thioalkylamine derivatives

Publications (1)

Publication Number Publication Date
BR0311266A true BR0311266A (pt) 2005-02-22

Family

ID=29558291

Family Applications (2)

Application Number Title Priority Date Filing Date
BR0311266-7A BR0311266A (pt) 2002-05-24 2003-05-12 Processo para a preparação de derivados de tioalquilamina
BRPI0311266-7A BRPI0311266B1 (pt) 2002-05-24 2003-05-12 Processo para a preparação de derivados de tioalquilamina

Family Applications After (1)

Application Number Title Priority Date Filing Date
BRPI0311266-7A BRPI0311266B1 (pt) 2002-05-24 2003-05-12 Processo para a preparação de derivados de tioalquilamina

Country Status (12)

Country Link
US (1) US7235668B2 (pt)
EP (1) EP1511724B1 (pt)
JP (1) JP4522851B2 (pt)
KR (1) KR100994169B1 (pt)
CN (1) CN100475789C (pt)
AU (1) AU2003245880A1 (pt)
BR (2) BR0311266A (pt)
DK (1) DK1511724T3 (pt)
ES (1) ES2471240T3 (pt)
IL (1) IL165137A (pt)
MX (1) MXPA04011479A (pt)
WO (1) WO2003099777A1 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1919860A1 (en) * 2005-08-24 2008-05-14 Bayer CropScience AG Preparation of thioalkylamines with high yields
EP1981841A1 (en) * 2005-08-24 2008-10-22 Bayer CropScience AG Preparation of thioalkylamines using chlorosulfonic acid
DE102006004063A1 (de) * 2006-01-28 2007-08-02 Degussa Gmbh Verfahren zur Herstellung von Methionin aus Homoserin
WO2009066749A1 (ja) * 2007-11-22 2009-05-28 Nihon Nohyaku Co., Ltd. チオアルキルアミン類の製造方法
CN101481321B (zh) 2009-02-27 2012-04-18 上海医药工业研究院 阿戈美拉汀卤化氢复合物及其制备方法
RU2466986C1 (ru) * 2011-05-30 2012-11-20 Учреждение Российской Академии Наук Институт Нефтехимии И Катализа Ран Способ получения n,n,-дизамещенных n-{[алкил(бензил)сульфанил]метил}аминов
TW201329025A (zh) 2011-11-01 2013-07-16 Astex Therapeutics Ltd 醫藥化合物
HUE036238T2 (hu) 2012-07-17 2018-06-28 Glaxosmithkline Ip No 2 Ltd Szelektív androgén receptor modulátorokként ható indolkarbonitril vegyületek

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2689867A (en) * 1948-12-03 1954-09-21 Phillips Petroleum Co Preparation of alkyl aminosulfides
US2912357A (en) * 1956-03-29 1959-11-10 Monsanto Chemicals Aminoalkylthiazoles
NL124622C (pt) * 1963-05-02
DE2045905A1 (de) 1970-09-17 1972-03-23 Badische Anilin- & Soda-Fabrik Ag, 6700 Ludwigshafen Substituierte Thioätherverbindungen
JPS59231064A (ja) 1983-06-13 1984-12-25 Mitsui Toatsu Chem Inc ２−メルカプトエチルアミン類の製造法
TW211595B (pt) * 1991-12-07 1993-08-21 Hoechst Ag
DE4214740A1 (de) * 1992-05-04 1993-11-11 Bayer Ag Reaktivfarbstoffe, deren Herstellung und Verwendung
JPH0616618A (ja) * 1992-07-03 1994-01-25 Retsuku Tec Lab Kk β−アミノエチル酸性硫酸エステルの製造方法
JP2001163854A (ja) * 1999-09-28 2001-06-19 Nippon Nohyaku Co Ltd チオアルキルアミン誘導体及びその製造方法
WO2001023350A1 (en) 1999-09-28 2001-04-05 Nihon Nohyaku Co., Ltd. Thioalkylamine derivatives and process for the preparation thereof

Also Published As

Publication number Publication date
IL165137A (en) 2009-02-11
US20050182275A1 (en) 2005-08-18
US7235668B2 (en) 2007-06-26
MXPA04011479A (es) 2005-02-14
EP1511724B1 (en) 2014-04-30
EP1511724A1 (en) 2005-03-09
BRPI0311266B1 (pt) 2019-08-20
KR20050003444A (ko) 2005-01-10
JP2005526858A (ja) 2005-09-08
IL165137A0 (en) 2005-12-18
WO2003099777A1 (en) 2003-12-04
JP4522851B2 (ja) 2010-08-11
CN100475789C (zh) 2009-04-08
KR100994169B1 (ko) 2010-11-15
CN1671656A (zh) 2005-09-21
DK1511724T3 (da) 2014-06-16
AU2003245880A1 (en) 2003-12-12
ES2471240T3 (es) 2014-06-25

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8O E 13 DA LPI.

B12B Appeal against refusal [chapter 12.2 patent gazette]
B25A Requested transfer of rights approved

Owner name: BAYER INTELLECTUAL PROPERTY GMBH (DE)

B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 20/08/2019, OBSERVADAS AS CONDICOES LEGAIS. (CO) 10 (DEZ) ANOS CONTADOS A PARTIR DE 20/08/2019, OBSERVADAS AS CONDICOES LEGAIS